EA200501736A1 - 2-замещённые пиримидины - Google Patents

2-замещённые пиримидины

Info

Publication number
EA200501736A1
EA200501736A1 EA200501736A EA200501736A EA200501736A1 EA 200501736 A1 EA200501736 A1 EA 200501736A1 EA 200501736 A EA200501736 A EA 200501736A EA 200501736 A EA200501736 A EA 200501736A EA 200501736 A1 EA200501736 A1 EA 200501736A1
Authority
EA
Eurasian Patent Office
Prior art keywords
substituted pyrimidines
pyrimidines
substituents
index
compounds
Prior art date
Application number
EA200501736A
Other languages
English (en)
Inventor
Хорди Тормо И Бласко
Карстен Блеттнер
Бернд МЮЛЛЕР
Маркус Гевер
Вассилиос Грамменос
Томас Гроте
Андреас Гипзер
Йоахим Райнхаймер
Петер Шэфер
Франк Шивек
Аня Швёглер
Оливер Вагнер
Зигфрид Штратманн
Ульрих Шёфль
Мария Шерер
Райнхард Штирль
Original Assignee
Басф Акциенгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Басф Акциенгезельшафт filed Critical Басф Акциенгезельшафт
Publication of EA200501736A1 publication Critical patent/EA200501736A1/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Изобретение относится к пиримидинам формулы Iв которой индекс n и заместители L, R-Rимеют приведенное в описании значение и Rсоответствует формулама также к способу получения и промежуточным продуктам для получения этих соединений, к содержащим их средствам, а также к их применению для борьбы с фитопатогенными грибами.
EA200501736A 2003-05-20 2004-05-10 2-замещённые пиримидины EA200501736A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10323026 2003-05-20
PCT/EP2004/004957 WO2004103978A1 (de) 2003-05-20 2004-05-10 2-substituierte pyrimidine

Publications (1)

Publication Number Publication Date
EA200501736A1 true EA200501736A1 (ru) 2006-04-28

Family

ID=33461831

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200501736A EA200501736A1 (ru) 2003-05-20 2004-05-10 2-замещённые пиримидины

Country Status (13)

Country Link
US (1) US20070054929A1 (ru)
EP (1) EP1633728A1 (ru)
JP (1) JP2007502846A (ru)
KR (1) KR20060013665A (ru)
CN (1) CN100453535C (ru)
AU (1) AU2004240717A1 (ru)
BR (1) BRPI0410482A (ru)
CA (1) CA2525762A1 (ru)
CO (1) CO5630009A2 (ru)
CR (1) CR8078A (ru)
EA (1) EA200501736A1 (ru)
MX (1) MXPA05011549A (ru)
WO (1) WO2004103978A1 (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004003428A1 (de) * 2004-01-23 2005-08-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue langwirksame Beta-2-Agonisten, und deren Verwendung als Arzneimittel
EP1751132B1 (de) * 2004-05-19 2008-03-26 Basf Se 2-substituierte pyrimidine und ihre verwendung als pestizide
TW200637556A (en) 2005-01-31 2006-11-01 Basf Ag Substituted 5-phenyl pyrimidines I in therapy
DE102005046592A1 (de) * 2005-09-28 2007-03-29 Basf Ag 2-Substituierte Hydroxylaminopyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Pestizid
EP1987011A1 (de) * 2006-02-15 2008-11-05 Basf Se 2-substituierte pyrimidine und ihre verwendung als pestizide
EP2001298A2 (de) * 2006-03-27 2008-12-17 Basf Se Substituierte 5-hetaryl-4-aminopyrimidine
CL2007002231A1 (es) * 2006-08-02 2008-04-11 Basf Ag Uso de compuestos derivados de 5-(het) arilpirimidina para combatir hongos daninos; compuestos derivados de 5-(het) arilpirimidina; agente fungicida; y agente farmaceutico.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4663327A (en) * 1984-05-23 1987-05-05 Bayer Aktiengesellschaft 1-heteroaryl-4-aryl-pyrazolin-5-ones
DE3419127A1 (de) * 1984-05-23 1985-11-28 Bayer Ag, 5090 Leverkusen 1-heteroaryl-4-aryl-pyrazolin-5-one
CN1178792A (zh) * 1996-10-07 1998-04-15 美国氰胺公司 五氟苯基唑类并嘧啶
KR20030011894A (ko) * 2000-06-13 2003-02-11 바스프 악티엔게젤샤프트 5-페닐 치환된 2-(시아노아미노)피리미딘 살균제
CA2440405A1 (en) * 2001-03-15 2002-09-26 Basf Aktiengesellschaft 5-phenylpyrimidine, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
BR0214253A (pt) * 2001-11-19 2004-12-14 Basf Aktengesellschaft Composto, processo para preparar o mesmo, agente fungicida, e, processo para combater fungos fitopatogênicos

Also Published As

Publication number Publication date
CO5630009A2 (es) 2006-04-28
CN100453535C (zh) 2009-01-21
BRPI0410482A (pt) 2006-06-13
CR8078A (es) 2006-07-14
MXPA05011549A (es) 2005-12-15
CN1791583A (zh) 2006-06-21
WO2004103978A1 (de) 2004-12-02
CA2525762A1 (en) 2004-12-02
JP2007502846A (ja) 2007-02-15
KR20060013665A (ko) 2006-02-13
US20070054929A1 (en) 2007-03-08
AU2004240717A1 (en) 2004-12-02
EP1633728A1 (de) 2006-03-15

Similar Documents

Publication Publication Date Title
NO20060230L (no) Nye aminobenzofenonforbindelser
EA200870116A1 (ru) Бициклические гетероарильные соединения
EA200700557A1 (ru) Замещенные гетероароилом серин-амиды
ATE384061T1 (de) Imidazo- und thiazolopyridine als jak3-kinase- inhibitoren
EA200601105A1 (ru) Замещённые бензоилом фенилаланин-амиды
NO20074093L (no) Fremgangsmater for fremstilling av glukopyranosyl-substituerte benzyl-benzenderivater og mellomprodukter derav
HRP20070076A2 (en) Pyrimidine derivatives
CY1106752T1 (el) Διϋδροπτεριδινονες, μεθοδος για την παραγωγη τους και χρηση τους ως φαρμακων
WO2006021379A8 (de) Dihydropteridinonderivate, verfahren zu deren herstellung und deren verwendung als arzneimittel
NO20062950L (no) 5,7-diaminopyrazolo `43-Dlpyrimidiner med PDE-5 inhiberende aktivitet
WO2006021378A8 (de) Dihydropteridinonderivate, verfahren zu deren herstellung und deren verwendung als arzneimittel
ATE362932T1 (de) Azaindolverbindungen als kinaseinhibitoren
CY1116885T1 (el) Υποκατεστημενα παραγωγα κυκλοεξυλομεθυλιου
EA200701930A1 (ru) Производные пиримидина для лечения гиперпролиферативных нарушений
EA200801608A1 (ru) Производные бензимидазолонкарбоновой кислоты
ATE411296T1 (de) Imidazolinderivate mit cb1-antagonistischer wirkung
NO20055632L (no) Aromatiske oksyfenyl- og aromatiske sulfanylfenylderivater
NO20054361D0 (no) Benzensylfonamidderivater, fremgangsmate for fremstilling og anvendelse derav for behandlig av smerte
EA200700166A1 (ru) 4-замещённые производные хинолина, способ получения и промежуточные вещества для их приготовления и содержащие их фармацевтические композиции
EA200601796A1 (ru) Пиримидиновые производные для лечения аномального клеточного роста
CY1106391T1 (el) 2-υποκατεστημενες πυριμιδινες
EA200601065A1 (ru) Производные имидазола, способы их получения и применения
EA200501399A1 (ru) Производные бензопирана, которые могут использоваться при лечении воспалительных заболеваний
BRPI0519267A2 (pt) derivado de quinolina, seu uso, produÇço e medicamento contendo o mesmo
EA200600605A1 (ru) Перегруппированные пентанолы, способ их получения и их применение в качестве противовоспалительных средств