DOP2013000051A - Compuestos heterociclico y sus usos - Google Patents
Compuestos heterociclico y sus usosInfo
- Publication number
- DOP2013000051A DOP2013000051A DO2013000051A DO2013000051A DOP2013000051A DO P2013000051 A DOP2013000051 A DO P2013000051A DO 2013000051 A DO2013000051 A DO 2013000051A DO 2013000051 A DO2013000051 A DO 2013000051A DO P2013000051 A DOP2013000051 A DO P2013000051A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- heterociclical
- compounds
- heterociclical compounds
- activity
- secretase
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención proporciona un derivado heterociclo que tiene una actividad inhibidora de la producción de amiloide ß superior y/o una actividad de modulación de ¿-secretasa superior, y el uso del mismo. Un compuesto representado por la fórmula (I): donde cada símbolo es como se define en la presente memoria descriptiva, o una sal del mismo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2010197064 | 2010-09-02 | ||
JP2011143548 | 2011-06-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2013000051A true DOP2013000051A (es) | 2013-04-30 |
Family
ID=45094181
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2013000051A DOP2013000051A (es) | 2010-09-02 | 2013-03-01 | Compuestos heterociclico y sus usos |
Country Status (21)
Country | Link |
---|---|
US (3) | US8822699B2 (es) |
EP (1) | EP2611805A1 (es) |
JP (1) | JP5871909B2 (es) |
KR (1) | KR20130139895A (es) |
CN (1) | CN103249733A (es) |
AR (1) | AR082865A1 (es) |
AU (1) | AU2011296887A1 (es) |
BR (1) | BR112013004746A2 (es) |
CA (1) | CA2809779A1 (es) |
CL (1) | CL2013000575A1 (es) |
DO (1) | DOP2013000051A (es) |
EA (1) | EA201390333A1 (es) |
EC (1) | ECSP13012535A (es) |
MA (1) | MA34556B1 (es) |
MX (1) | MX2013002511A (es) |
PE (1) | PE20131305A1 (es) |
SG (1) | SG187917A1 (es) |
TW (1) | TW201213327A (es) |
UY (1) | UY33586A (es) |
WO (1) | WO2012029991A1 (es) |
ZA (1) | ZA201301929B (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20120142672A1 (en) * | 2009-07-13 | 2012-06-07 | Tatsuki Koike | Heterocyclic compound and use thereof |
WO2012029991A1 (en) * | 2010-09-02 | 2012-03-08 | Takeda Pharmaceutical Company Limited | Fused triazoles for the treatment or prophylaxis of mild cognitive impairment |
EP2687528A1 (en) * | 2012-07-17 | 2014-01-22 | Ares Trading S.A. | Fused triazole derivatives as gamma secretase modulators |
RU2563254C2 (ru) * | 2013-07-08 | 2015-09-20 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Московский государственный университет имени М.В. Ломоносова" (МГУ) | Способ получения производных 7-(гетеро)арил-4,5,6,7-тетрагидро[1,2,3]триазоло[1,5-a]пиридина |
CN113402394B (zh) * | 2015-05-12 | 2024-04-26 | Fmc公司 | 作为除草剂的芳基取代的双环化合物 |
US20210079182A1 (en) * | 2019-09-12 | 2021-03-18 | Dupont Electronics, Inc. | Polyimide films and electronic devices |
TW202339756A (zh) * | 2021-12-17 | 2023-10-16 | 美商雅斯娜製藥公司 | 雙環化合物用於治療疾病之用途 |
Family Cites Families (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2003523345A (ja) | 2000-02-17 | 2003-08-05 | ブリストル−マイヤーズ スクイブ ファーマ カンパニー | Aβタンパク質産生の阻害剤としてのスクシノイルアミノ炭素環および複素環 |
JP4847868B2 (ja) | 2003-05-14 | 2011-12-28 | ニューロジェネティック ファーマシューティカルズ、 インコーポレイテッド | 化合物、及び、アミロイドベータの調節におけるその使用 |
JP2007533641A (ja) * | 2003-10-15 | 2007-11-22 | ターガセプト,インコーポレイテッド | 疼痛緩和および中枢神経系障害治療のためのアザビシクロ化合物 |
MXPA06013534A (es) | 2004-05-26 | 2007-05-10 | Eisai R&D Man Co Ltd | Compuesto de cinamida. |
CA2580119A1 (en) | 2004-10-26 | 2006-05-04 | Eisai R & D Management Co., Ltd. | Amorphous object of cinnamide compound |
EP1976527A4 (en) | 2006-01-11 | 2009-04-22 | Merck & Co Inc | CONDENSED TRIAZOL TACHYKININE RECEPTOR ANTAGONISTS |
KR101464651B1 (ko) * | 2006-03-09 | 2014-11-24 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 다환식 신나미드 유도체 |
TWI378091B (en) | 2006-03-09 | 2012-12-01 | Eisai R&D Man Co Ltd | Multi-cyclic cinnamide derivatives |
TW200808800A (en) | 2006-05-05 | 2008-02-16 | Astrazeneca Ab | MGluR5 modulators V |
EP2119719A1 (en) | 2006-12-26 | 2009-11-18 | Daiichi Sankyo Company, Limited | Thiazepine derivative |
WO2008077649A1 (en) | 2006-12-26 | 2008-07-03 | Gilead Sciences, Inc. | Pyrido(3,2-d)pyrimidines useful for treating viral infectons |
EP2117311A4 (en) | 2007-02-08 | 2011-05-11 | Merck Sharp & Dohme | THERAPEUTICS |
AU2008333865A1 (en) | 2007-12-06 | 2009-06-11 | Schering Corporation | Gamma secretase modulators |
TW201030002A (en) | 2009-01-16 | 2010-08-16 | Bristol Myers Squibb Co | Bicyclic compounds for the reduction of beta-amyloid production |
JP2010197064A (ja) | 2009-02-23 | 2010-09-09 | Chugoku Electric Power Co Inc:The | 直下位置測定装置 |
JP2012051806A (ja) * | 2009-02-26 | 2012-03-15 | Eisai R & D Management Co Ltd | イミダゾリルピラジン誘導体 |
JP2012051807A (ja) | 2009-02-26 | 2012-03-15 | Eisai R & D Management Co Ltd | アリールイミダゾール化合物 |
CA2753696A1 (en) * | 2009-02-26 | 2010-09-02 | Noritaka Kitazawa | Nitrogen-containing fused heterocyclic compounds and their use as beta amyloid production inhibitors |
WO2011002067A1 (ja) | 2009-07-02 | 2011-01-06 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
US20120142672A1 (en) * | 2009-07-13 | 2012-06-07 | Tatsuki Koike | Heterocyclic compound and use thereof |
KR20120050450A (ko) | 2009-07-15 | 2012-05-18 | 얀센 파마슈티칼즈, 인코포레이티드 | 감마 세크레타제 조절제로서의 치환된 트리아졸 및 이미다졸 유도체 |
US8637525B2 (en) | 2009-07-31 | 2014-01-28 | Bristol-Myers Squibb Company | Compounds for the reduction of beta-amyloid production |
TWI468402B (zh) | 2009-07-31 | 2015-01-11 | 必治妥美雅史谷比公司 | 降低β-類澱粉生成之化合物 |
WO2011016559A1 (ja) | 2009-08-07 | 2011-02-10 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
JP2011143548A (ja) | 2010-01-12 | 2011-07-28 | Panasonic Corp | スクリーン印刷機及びスクリーン印刷方法 |
MX2012008259A (es) | 2010-01-15 | 2012-08-17 | Janssen Pharmaceuticals Inc | Novedosos derivados biciclicos de triazol sustituidos como moduladores de gamma secretasa. |
WO2012029991A1 (en) * | 2010-09-02 | 2012-03-08 | Takeda Pharmaceutical Company Limited | Fused triazoles for the treatment or prophylaxis of mild cognitive impairment |
-
2011
- 2011-09-01 WO PCT/JP2011/070419 patent/WO2012029991A1/en active Application Filing
- 2011-09-01 KR KR1020137008170A patent/KR20130139895A/ko not_active Application Discontinuation
- 2011-09-01 JP JP2013510386A patent/JP5871909B2/ja not_active Expired - Fee Related
- 2011-09-01 BR BR112013004746A patent/BR112013004746A2/pt not_active IP Right Cessation
- 2011-09-01 MA MA35785A patent/MA34556B1/fr unknown
- 2011-09-01 TW TW100131443A patent/TW201213327A/zh unknown
- 2011-09-01 AU AU2011296887A patent/AU2011296887A1/en not_active Abandoned
- 2011-09-01 MX MX2013002511A patent/MX2013002511A/es not_active Application Discontinuation
- 2011-09-01 CN CN2011800518621A patent/CN103249733A/zh active Pending
- 2011-09-01 UY UY0001033586A patent/UY33586A/es unknown
- 2011-09-01 SG SG2013012604A patent/SG187917A1/en unknown
- 2011-09-01 EP EP11791058.8A patent/EP2611805A1/en not_active Withdrawn
- 2011-09-01 EA EA201390333A patent/EA201390333A1/ru unknown
- 2011-09-01 PE PE2013000360A patent/PE20131305A1/es not_active Application Discontinuation
- 2011-09-01 US US13/223,455 patent/US8822699B2/en not_active Expired - Fee Related
- 2011-09-01 AR ARP110103195A patent/AR082865A1/es unknown
- 2011-09-01 US US13/819,239 patent/US8901309B2/en not_active Expired - Fee Related
- 2011-09-01 CA CA2809779A patent/CA2809779A1/en not_active Abandoned
-
2013
- 2013-02-28 CL CL2013000575A patent/CL2013000575A1/es unknown
- 2013-03-01 DO DO2013000051A patent/DOP2013000051A/es unknown
- 2013-03-14 ZA ZA2013/01929A patent/ZA201301929B/en unknown
- 2013-03-28 EC ECSP13012535 patent/ECSP13012535A/es unknown
-
2014
- 2014-08-08 US US14/454,993 patent/US20140350260A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2809779A1 (en) | 2012-03-08 |
US8901309B2 (en) | 2014-12-02 |
MX2013002511A (es) | 2013-07-29 |
BR112013004746A2 (pt) | 2016-06-07 |
SG187917A1 (en) | 2013-04-30 |
ZA201301929B (en) | 2013-11-27 |
KR20130139895A (ko) | 2013-12-23 |
JP2013536798A (ja) | 2013-09-26 |
UY33586A (es) | 2012-03-30 |
US20120059030A1 (en) | 2012-03-08 |
EA201390333A1 (ru) | 2013-08-30 |
ECSP13012535A (es) | 2013-06-28 |
US20130178497A1 (en) | 2013-07-11 |
EP2611805A1 (en) | 2013-07-10 |
CL2013000575A1 (es) | 2013-08-23 |
PE20131305A1 (es) | 2013-10-31 |
AU2011296887A1 (en) | 2013-04-11 |
TW201213327A (en) | 2012-04-01 |
JP5871909B2 (ja) | 2016-03-01 |
MA34556B1 (fr) | 2013-09-02 |
WO2012029991A1 (en) | 2012-03-08 |
US20140350260A1 (en) | 2014-11-27 |
AR082865A1 (es) | 2013-01-16 |
US8822699B2 (en) | 2014-09-02 |
CN103249733A (zh) | 2013-08-14 |
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