DK72282A - Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf - Google Patents

Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf Download PDF

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Publication number
DK72282A
DK72282A DK72282A DK72282A DK72282A DK 72282 A DK72282 A DK 72282A DK 72282 A DK72282 A DK 72282A DK 72282 A DK72282 A DK 72282A DK 72282 A DK72282 A DK 72282A
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DK
Denmark
Prior art keywords
methyl
penam
acetoxymethyl
dioxide
esters
Prior art date
Application number
DK72282A
Other languages
Danish (da)
English (en)
Inventor
W E Barth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK72282A publication Critical patent/DK72282A/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK72282A 1981-02-20 1982-02-19 Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf DK72282A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/236,407 US4364957A (en) 1979-09-26 1981-02-20 Bis-esters of alkanediols as antibacterial agents

Publications (1)

Publication Number Publication Date
DK72282A true DK72282A (da) 1982-08-21

Family

ID=22889370

Family Applications (1)

Application Number Title Priority Date Filing Date
DK72282A DK72282A (da) 1981-02-20 1982-02-19 Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf

Country Status (11)

Country Link
US (1) US4364957A (es)
EP (1) EP0059046B1 (es)
JP (1) JPS57154192A (es)
AT (1) ATE15044T1 (es)
AU (1) AU527894B2 (es)
CA (1) CA1176242A (es)
DE (1) DE3265503D1 (es)
DK (1) DK72282A (es)
ES (1) ES8304992A1 (es)
GR (1) GR75173B (es)
IE (1) IE52902B1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4478748A (en) * 1981-02-20 1984-10-23 Pfizer Inc. Bis-esters of alkanediols
US4530792A (en) * 1982-11-01 1985-07-23 Pfizer Inc. Process and intermediates for preparation of 1,1-dioxopenicillanoyloxymethyl 6-beta-aminopenicillanate
US4462934A (en) 1983-03-31 1984-07-31 Pfizer Inc. Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides
JPS60214792A (ja) * 1984-04-06 1985-10-28 Taiho Yakuhin Kogyo Kk ペナム酸エステル誘導体
JPH0410174Y2 (es) * 1986-09-24 1992-03-13
CN104650119B (zh) * 2015-02-10 2017-04-05 中国科学院长春应用化学研究所 一种β‑内酰胺化合物的制备方法
IT202000031070A1 (it) 2020-12-16 2022-06-16 Paolo Bonomi Procedimento di sintesi di derivati ammidici dell’acido 8-idrossi penicillanico

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
IE49371B1 (en) * 1979-02-13 1985-09-18 Leo Pharm Prod Ltd 6-(azacycloalkyl-or azabicycloalkyl-methyl imino)penicillanic acid esters
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4256733A (en) * 1979-09-26 1981-03-17 Pfizer Inc. Acetoxymethyl penam compounds as β-lactamase inhibitors

Also Published As

Publication number Publication date
ES509782A0 (es) 1983-03-16
GR75173B (es) 1984-07-13
DE3265503D1 (en) 1985-09-26
ATE15044T1 (de) 1985-09-15
JPS6330312B2 (es) 1988-06-17
IE820342L (en) 1982-08-20
CA1176242A (en) 1984-10-16
ES8304992A1 (es) 1983-03-16
EP0059046B1 (en) 1985-08-21
JPS57154192A (en) 1982-09-22
US4364957A (en) 1982-12-21
EP0059046A1 (en) 1982-09-01
AU8062382A (en) 1982-11-04
AU527894B2 (en) 1983-03-31
IE52902B1 (en) 1988-04-13

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