DK171350B1 - 4-(2-Pyridyloxy)-2-butenylenderivater og medicinsk acceptable salte, hydrater og solvater heraf samt farmaceutisk produkt omfattende samme - Google Patents
4-(2-Pyridyloxy)-2-butenylenderivater og medicinsk acceptable salte, hydrater og solvater heraf samt farmaceutisk produkt omfattende samme Download PDFInfo
- Publication number
- DK171350B1 DK171350B1 DK448885A DK448885A DK171350B1 DK 171350 B1 DK171350 B1 DK 171350B1 DK 448885 A DK448885 A DK 448885A DK 448885 A DK448885 A DK 448885A DK 171350 B1 DK171350 B1 DK 171350B1
- Authority
- DK
- Denmark
- Prior art keywords
- cis
- oxy
- pyridyl
- piperidinomethyl
- solvates
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP20669084A JPS6185365A (ja) | 1984-10-02 | 1984-10-02 | アミノアルキルピリジルオキシ誘導体 |
| JP20669084 | 1984-10-02 | ||
| JP5020785A JPS61207375A (ja) | 1985-03-12 | 1985-03-12 | ピリジルオキシ誘導体 |
| JP5020785 | 1985-03-12 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK448885D0 DK448885D0 (da) | 1985-10-02 |
| DK448885A DK448885A (da) | 1986-04-03 |
| DK171350B1 true DK171350B1 (da) | 1996-09-16 |
Family
ID=26390658
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK448885A DK171350B1 (da) | 1984-10-02 | 1985-10-02 | 4-(2-Pyridyloxy)-2-butenylenderivater og medicinsk acceptable salte, hydrater og solvater heraf samt farmaceutisk produkt omfattende samme |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US4710498A (de) |
| EP (1) | EP0177016B1 (de) |
| AU (1) | AU583536B2 (de) |
| CA (1) | CA1275097A (de) |
| DE (2) | DE177016T1 (de) |
| DK (1) | DK171350B1 (de) |
| ES (1) | ES8701161A1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4772704A (en) * | 1983-09-21 | 1988-09-20 | Bristol-Myers Company | 2,5-disubstituted-4(3H)-pyrimidones having histamine H2 -receptor antagonist activity |
| US4912101A (en) * | 1987-03-13 | 1990-03-27 | Fujirebio Kabushiki Kaisha | 4-aminomethyl-pyridyl-2-oxy derivatives having anti-ulcer activity |
| JPH0613486B2 (ja) * | 1987-12-07 | 1994-02-23 | 株式会社池田模範堂 | ピリミドン誘導体及びその医薬的に許容される塩 |
| WO1992013854A1 (fr) * | 1991-01-30 | 1992-08-20 | Central Glass Company, Limited | Compose de phtalimide et sa production |
| DE69317714T2 (de) * | 1992-08-07 | 1998-07-30 | Fujirebio Kk | Verfahren zur Herstellung von Aminobutene-Derivate |
| US5872139A (en) * | 1996-06-17 | 1999-02-16 | American Home Products Corporation | Heterocyclymethylamino derivatives of cyclobutene-3,4-diones |
| US6436972B1 (en) | 2000-04-10 | 2002-08-20 | Dalhousie University | Pyridones and their use as modulators of serine hydrolase enzymes |
| WO2022034121A1 (en) | 2020-08-11 | 2022-02-17 | Université De Strasbourg | H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4166857A (en) * | 1975-07-03 | 1979-09-04 | Smith Kline & French Laboratories Limited | N-Hetero substituted cyclobutenones |
| US4120968A (en) * | 1975-07-31 | 1978-10-17 | Smith Kline & French Laboratories Limited | Heterocyclic alkylaminocyclobutenediones |
| NZ186511A (en) | 1977-03-19 | 1980-11-14 | Smith Kline French Lab | 3-substituted alkylamino-6-substituted alkyl-1,2,4-triazin-5-ones and pharmaceutical compositions 3-substituted thio-1,2,4-triazin-5-ones |
| FR2437392A1 (fr) | 1978-06-30 | 1980-04-25 | Rhone Poulenc Ind | Stabilisation du trichloro-1,1,1 ethane |
| IL60944A (en) | 1979-09-04 | 1987-11-30 | Bristol Myers Co | 3,4-disubstituted-1,2,5-thiadiazole-1-oxides and 1,1 dioxides,process for their preparation and pharmaceutical compositions comprising them |
| CA1155842A (en) * | 1980-03-29 | 1983-10-25 | Thomas H. Brown | Compounds |
| ZW21281A1 (en) * | 1980-10-01 | 1981-11-18 | Smith Kline French Lab | Amine derivatives |
| US4503051A (en) * | 1981-05-18 | 1985-03-05 | Bristol-Myers Company | Substituted 3-cyclobutene-1,2-diones, pharmaceutical compositions thereof and methods of use |
| US4808589A (en) * | 1982-02-20 | 1989-02-28 | Smith Kline & French Laboratories Limited | Pyrimidone derivatives |
| KR840004100A (ko) | 1982-03-17 | 1984-10-06 | 데비드 마틴 워터스 | 피리딘 유도체 |
| EP0089153B1 (de) * | 1982-03-17 | 1986-09-24 | Smith Kline & French Laboratories Limited | Pyridin-Derivate |
| JPS5984867A (ja) * | 1982-10-02 | 1984-05-16 | スミス・クライン・アンド・フレンチ・ラボラトリ−ス・リミテツド | ジオキソシクロブテン誘導体 |
| AU1956283A (en) * | 1982-10-02 | 1984-04-05 | Smith Kline & French Laboratories Limited | 1-(3-(4-(substited aminomethyl)pyrid-2-yl-oxy)-prop-1-yl- amino) - 2-aminocyclobut-i-ene-3,4-diones |
| ZA839248B (en) * | 1982-12-14 | 1984-10-31 | Smith Kline French Lab | Pyridine derivatives |
| JO1279B1 (en) * | 1982-12-23 | 1985-04-20 | جون ايف روبرت | Pyridine derivatives |
| US4440933A (en) * | 1983-03-16 | 1984-04-03 | Bristol-Myers Company | Process for preparing 1,2,5-thiadiazoles |
| DE3513184A1 (de) * | 1985-04-12 | 1986-10-16 | Ludwig Heumann & Co GmbH, 8500 Nürnberg | 1,3,4-thiadiazolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
-
1985
- 1985-09-27 CA CA000491789A patent/CA1275097A/en not_active Expired - Fee Related
- 1985-09-30 US US06/781,881 patent/US4710498A/en not_active Expired - Lifetime
- 1985-09-30 AU AU48136/85A patent/AU583536B2/en not_active Ceased
- 1985-10-01 DE DE198585112416T patent/DE177016T1/de active Pending
- 1985-10-01 ES ES547458A patent/ES8701161A1/es not_active Expired
- 1985-10-01 EP EP85112416A patent/EP0177016B1/de not_active Expired - Lifetime
- 1985-10-01 DE DE85112416T patent/DE3587416T2/de not_active Expired - Fee Related
- 1985-10-02 DK DK448885A patent/DK171350B1/da not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES8701161A1 (es) | 1986-11-16 |
| AU583536B2 (en) | 1989-05-04 |
| CA1275097A (en) | 1990-10-09 |
| ES547458A0 (es) | 1986-11-16 |
| AU4813685A (en) | 1986-04-10 |
| DE3587416T2 (de) | 1993-09-30 |
| DK448885A (da) | 1986-04-03 |
| EP0177016A3 (en) | 1986-12-03 |
| DE3587416D1 (de) | 1993-07-29 |
| EP0177016B1 (de) | 1993-06-23 |
| DE177016T1 (de) | 1986-11-06 |
| DK448885D0 (da) | 1985-10-02 |
| US4710498A (en) | 1987-12-01 |
| EP0177016A2 (de) | 1986-04-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B1 | Patent granted (law 1993) | ||
| PBP | Patent lapsed |