DK166675B1 - Mycophenolsyrederivater, fremgangsmaade til fremstilling deraf, farmaceutisk praeparat indeholdende disse samt anvendelse af disse derivater til fremstilling af et laegemiddel - Google Patents

Mycophenolsyrederivater, fremgangsmaade til fremstilling deraf, farmaceutisk praeparat indeholdende disse samt anvendelse af disse derivater til fremstilling af et laegemiddel Download PDF

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Publication number
DK166675B1
DK166675B1 DK658787A DK658787A DK166675B1 DK 166675 B1 DK166675 B1 DK 166675B1 DK 658787 A DK658787 A DK 658787A DK 658787 A DK658787 A DK 658787A DK 166675 B1 DK166675 B1 DK 166675B1
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DK
Denmark
Prior art keywords
formula
compound
methyl
pharmaceutically acceptable
hydrogen
Prior art date
Application number
DK658787A
Other languages
Danish (da)
English (en)
Other versions
DK658787A (da
DK658787D0 (da
Inventor
Peter H Nelson
Chee-Liang Leo Gu
Anthony C Allison
Elsie M Eugui
William A Lee
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21733252&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK166675(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of DK658787D0 publication Critical patent/DK658787D0/da
Publication of DK658787A publication Critical patent/DK658787A/da
Application granted granted Critical
Publication of DK166675B1 publication Critical patent/DK166675B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Furan Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Saccharide Compounds (AREA)
DK658787A 1987-01-30 1987-12-15 Mycophenolsyrederivater, fremgangsmaade til fremstilling deraf, farmaceutisk praeparat indeholdende disse samt anvendelse af disse derivater til fremstilling af et laegemiddel DK166675B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US871787 1987-01-30
US07/008,717 US4753935A (en) 1987-01-30 1987-01-30 Morpholinoethylesters of mycophenolic acid and pharmaceutical compositions

Publications (3)

Publication Number Publication Date
DK658787D0 DK658787D0 (da) 1987-12-15
DK658787A DK658787A (da) 1988-07-31
DK166675B1 true DK166675B1 (da) 1993-06-28

Family

ID=21733252

Family Applications (1)

Application Number Title Priority Date Filing Date
DK658787A DK166675B1 (da) 1987-01-30 1987-12-15 Mycophenolsyrederivater, fremgangsmaade til fremstilling deraf, farmaceutisk praeparat indeholdende disse samt anvendelse af disse derivater til fremstilling af et laegemiddel

Country Status (26)

Country Link
US (7) US4753935A (hu)
EP (1) EP0281713B1 (hu)
JP (1) JPS63188672A (hu)
KR (1) KR940003758B1 (hu)
AT (1) ATE68180T1 (hu)
AU (1) AU599728B2 (hu)
CA (1) CA1333285C (hu)
DE (2) DE19675020I2 (hu)
DK (1) DK166675B1 (hu)
ES (1) ES2038190T3 (hu)
FI (1) FI85141C (hu)
GE (1) GEP20094816B (hu)
GR (1) GR3002866T3 (hu)
HK (1) HK125893A (hu)
HU (2) HU201927B (hu)
IE (1) IE60750B1 (hu)
IL (1) IL84833A (hu)
LU (1) LU88795I2 (hu)
LV (1) LV5748B4 (hu)
MX (1) MX9203163A (hu)
NL (1) NL960019I2 (hu)
NO (2) NO171680C (hu)
NZ (1) NZ222922A (hu)
PH (1) PH23819A (hu)
PT (1) PT86343B (hu)
ZA (1) ZA879414B (hu)

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Also Published As

Publication number Publication date
IE873397L (en) 1988-07-30
LV5748A4 (lv) 1996-10-20
US4948793A (en) 1990-08-14
ATE68180T1 (de) 1991-10-15
US4952579A (en) 1990-08-28
US4808592A (en) 1989-02-28
IL84833A (en) 1992-03-29
US4992467A (en) 1991-02-12
NZ222922A (en) 1990-09-26
HU201927B (en) 1991-01-28
FI875502A0 (fi) 1987-12-15
HUT47567A (en) 1989-03-28
FI85141C (fi) 1992-03-10
AU8254087A (en) 1988-08-04
LU88795I2 (fr) 1996-11-05
KR940003758B1 (ko) 1994-04-30
MX9203163A (es) 1992-07-31
HK125893A (en) 1993-11-19
PT86343A (en) 1988-01-01
FI85141B (fi) 1991-11-29
AU599728B2 (en) 1990-07-26
PT86343B (pt) 1991-02-08
US4868153A (en) 1989-09-19
JPH0571591B2 (hu) 1993-10-07
EP0281713B1 (en) 1991-10-09
NL960019I2 (nl) 1997-06-02
NO875240D0 (no) 1987-12-15
EP0281713A1 (en) 1988-09-14
US4786637A (en) 1988-11-22
US4753935A (en) 1988-06-28
GR3002866T3 (en) 1993-01-25
CA1333285C (en) 1994-11-29
KR880009016A (ko) 1988-09-13
IL84833A0 (en) 1988-06-30
HU210350A9 (en) 1995-03-28
LV5748B4 (lv) 1997-02-20
ZA879414B (en) 1989-08-30
NO171680C (no) 1993-04-21
NO171680B (no) 1993-01-11
NO1997007I1 (no) 1997-07-01
DE19675020I2 (de) 2002-11-07
FI875502A (fi) 1988-07-31
GEP20094816B (en) 2009-11-10
ES2038190T3 (es) 1993-07-16
DE3773660D1 (de) 1991-11-14
NO875240L (no) 1988-08-01
NL960019I1 (nl) 1996-10-01
IE60750B1 (en) 1994-08-10
PH23819A (en) 1989-11-23
DK658787A (da) 1988-07-31
DK658787D0 (da) 1987-12-15
JPS63188672A (ja) 1988-08-04

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