DK141604B - Fremgangsmåde til fremstilling af 1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-on-derivater. - Google Patents

Fremgangsmåde til fremstilling af 1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-on-derivater. Download PDF

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Publication number
DK141604B
DK141604B DK372871AA DK372871A DK141604B DK 141604 B DK141604 B DK 141604B DK 372871A A DK372871A A DK 372871AA DK 372871 A DK372871 A DK 372871A DK 141604 B DK141604 B DK 141604B
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DK
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Prior art keywords
tetrahydro
derivatives
benzodiazepin
amino
compounds
Prior art date
Application number
DK372871AA
Other languages
Danish (da)
English (en)
Other versions
DK141604C (de
Inventor
Lajos Kisfaludy
Istvan Szakolczay
Juliana Roehricht
Ferenc Korenczki
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of DK141604B publication Critical patent/DK141604B/da
Application granted granted Critical
Publication of DK141604C publication Critical patent/DK141604C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/28Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK372871AA 1970-07-30 1971-07-29 Fremgangsmåde til fremstilling af 1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-on-derivater. DK141604B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HURI000403 1970-07-30
HURI000403 1970-07-30

Publications (2)

Publication Number Publication Date
DK141604B true DK141604B (da) 1980-05-05
DK141604C DK141604C (de) 1980-10-06

Family

ID=11000846

Family Applications (1)

Application Number Title Priority Date Filing Date
DK372871AA DK141604B (da) 1970-07-30 1971-07-29 Fremgangsmåde til fremstilling af 1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-on-derivater.

Country Status (10)

Country Link
JP (1) JPS5432792B1 (de)
AT (1) AT311356B (de)
CH (1) CH558370A (de)
CS (1) CS171708B2 (de)
DK (1) DK141604B (de)
ES (1) ES393521A1 (de)
NL (1) NL7110356A (de)
PL (1) PL70872B1 (de)
SE (1) SE385888B (de)
SU (1) SU461503A3 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU187262B (en) * 1979-08-16 1985-12-28 Richter Gedeon Vegyeszet Process for preparing new tetrahydro-1,4-benzodiazepin-2-ones

Also Published As

Publication number Publication date
SE385888B (sv) 1976-07-26
NL7110356A (de) 1972-02-01
DK141604C (de) 1980-10-06
CS171708B2 (de) 1976-10-29
SU461503A3 (ru) 1975-02-25
CH558370A (de) 1975-01-31
ES393521A1 (es) 1973-08-16
AT311356B (de) 1973-11-12
PL70872B1 (de) 1974-04-30
JPS5432792B1 (de) 1979-10-16

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