DK12084A - Substituerede carboxy-thiazolo(3,2-a)pyrimidinderivater samt fremgangsmaade til fremstilling heraf - Google Patents

Substituerede carboxy-thiazolo(3,2-a)pyrimidinderivater samt fremgangsmaade til fremstilling heraf Download PDF

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Publication number
DK12084A
DK12084A DK12084A DK12084A DK12084A DK 12084 A DK12084 A DK 12084A DK 12084 A DK12084 A DK 12084A DK 12084 A DK12084 A DK 12084A DK 12084 A DK12084 A DK 12084A
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DK
Denmark
Prior art keywords
thiazolo
procedures
preparing
pyrimidine derivatives
substituted carboxy
Prior art date
Application number
DK12084A
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English (en)
Other versions
DK12084D0 (da
Inventor
Gianfederico Doria
Carlo Passarotti
Maria Luisa Corno
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of DK12084D0 publication Critical patent/DK12084D0/da
Publication of DK12084A publication Critical patent/DK12084A/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK12084A 1983-01-12 1984-01-11 Substituerede carboxy-thiazolo(3,2-a)pyrimidinderivater samt fremgangsmaade til fremstilling heraf DK12084A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB838300728A GB8300728D0 (en) 1983-01-12 1983-01-12 Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives

Publications (2)

Publication Number Publication Date
DK12084D0 DK12084D0 (da) 1984-01-11
DK12084A true DK12084A (da) 1984-07-13

Family

ID=10536219

Family Applications (1)

Application Number Title Priority Date Filing Date
DK12084A DK12084A (da) 1983-01-12 1984-01-11 Substituerede carboxy-thiazolo(3,2-a)pyrimidinderivater samt fremgangsmaade til fremstilling heraf

Country Status (27)

Country Link
US (2) US4558046A (da)
JP (1) JPS59130891A (da)
KR (1) KR840007420A (da)
AT (1) AT386601B (da)
AU (1) AU568527B2 (da)
BE (1) BE898641A (da)
CA (1) CA1232604A (da)
CH (1) CH660011A5 (da)
CS (1) CS27984A2 (da)
DE (1) DE3400733A1 (da)
DK (1) DK12084A (da)
ES (1) ES8505357A1 (da)
FI (1) FI77869C (da)
FR (1) FR2539131B1 (da)
GB (1) GB8300728D0 (da)
GR (1) GR81735B (da)
HU (1) HU190945B (da)
IL (1) IL70651A (da)
IT (1) IT1185050B (da)
NL (1) NL8400099A (da)
NO (1) NO840092L (da)
NZ (1) NZ206816A (da)
PH (1) PH22448A (da)
PT (1) PT77946B (da)
SE (1) SE456996B (da)
SU (1) SU1355131A3 (da)
ZA (1) ZA84227B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4921854A (en) * 1986-12-30 1990-05-01 Egis Gyogyszergyar Condensed thiazolopyrimidine, pyrimido-thiazine or thiazepine pyrimidine compounds
US6121300A (en) 1998-11-10 2000-09-19 Wagle; Dilip R. Reversing advanced glycosylation cross-links using heterocyclic-substituted thiazolium salts
AU2009220825A1 (en) * 2008-01-11 2012-01-19 Glenmark Pharmaceuticals, S.A. Fused pyrimidine derivatives as TRPV3 modulators
US8119647B2 (en) * 2008-04-23 2012-02-21 Glenmark Pharmaceuticals S.A. Fused pyrimidineone compounds as TRPV3 modulators

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3594378A (en) * 1969-10-24 1971-07-20 Ayerst Mckenna & Harrison Thiazolopyrimidine derivatives and preparation thereof
US3888983A (en) * 1970-08-14 1975-06-10 Seperic Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia
GB1334628A (en) * 1972-02-02 1973-10-24 Seperic Thiazolino-pyrimidinone derivatives their preparation and appli cations
DE2557425C2 (de) * 1975-12-19 1987-03-19 C.H. Boehringer Sohn, 6507 Ingelheim 11-Oxo-11-H-pyrido[2,1-b]-chinazolin-2-carbonsäure und ihre Salze, Verfahren zu ihrer Herstellung und Arzneimittel
US4041163A (en) * 1976-03-29 1977-08-09 Pfizer Inc. N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
US4168380A (en) * 1978-04-21 1979-09-18 Hoffmann-La Roche Inc. 7-Methoxy-5-oxo-5H-thiazolo[2,3-b]quinazoline-2-carboxylic acid
US4223031A (en) * 1978-05-05 1980-09-16 Mead Johnson & Company Azolopyrimidinones
AU527931B2 (en) * 1979-05-08 1983-03-31 Farmitalia Carlo Erba S.P.A. Substituted pyrido(1,2-a)pyrimidines
US4282360A (en) * 1979-10-12 1981-08-04 Hoffmann-La Roche Inc. 7-Methylthio or methylsulfinyl-5-oxo-5H-thiazolo[2,3-b]quinazoline-2-carboxylic acid
DK151811C (da) * 1979-11-23 1988-06-06 Pfizer Analogifremgangsmaade til fremstilling af n-(5-tetrazolyl)-1-oxo-1h-thiazolooe3,2-aaa-pyrimidin-2-carboxamider eller farmaceutisk acceptable kationsalte deraf samt 1-oxo-1h-thiazolooe3,2-aaapyrimidin-2-carboxylsyrer til anvendelse som udgangsmaterialer ved fremgangsmaaden
PL129612B1 (en) * 1980-07-24 1984-05-31 Rhone Poulenc Ind Process for preparing novel derivatives of 2,3,6,7-tetrahydrothiazole/3,2-a/pirymidin-5-one
US4340734A (en) * 1980-11-14 1982-07-20 American Cyanamid Company 3-(α-Substituted-benzyl)-2,3-dihydrothiazolo [3,2-a][1,3]diazacyclan-3-ol derivatives
US4443451A (en) * 1981-07-15 1984-04-17 Janssen Pharmaceutica N.V. Bicyclic pyrimidin-5-one derivatives
US4325955A (en) * 1981-03-23 1982-04-20 American Cyanamid Company Substituted 3-benzhydrylthiazolo(3,2-a)pyrimidines
US4347248A (en) * 1981-03-23 1982-08-31 American Cyanamid Company 2,3-Disubstituted-thiazolo[3,2-a]pyrimidines
NL8202706A (nl) * 1981-07-15 1983-02-01 Erba Farmitalia Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.
AU553266B2 (en) * 1982-02-04 1986-07-10 Farmitalia Carlo Erba S.P.A. Substituted 1,3,4-thiadiazolo(3,2-a) pyrimidines

Also Published As

Publication number Publication date
SE456996B (sv) 1988-11-21
SE8400118L (sv) 1984-07-13
AU568527B2 (en) 1988-01-07
IL70651A0 (en) 1984-04-30
IL70651A (en) 1986-10-31
KR840007420A (ko) 1984-12-07
FI77869C (fi) 1989-05-10
US4609660A (en) 1986-09-02
BE898641A (fr) 1984-07-10
PT77946B (en) 1986-04-16
US4558046A (en) 1985-12-10
FR2539131B1 (fr) 1987-01-30
ZA84227B (en) 1984-08-29
IT8419085A0 (it) 1984-01-10
JPS59130891A (ja) 1984-07-27
AT386601B (de) 1988-09-26
ES528662A0 (es) 1985-05-16
FI840088A (fi) 1984-07-13
CS27984A2 (en) 1991-03-12
GB8300728D0 (en) 1983-02-16
NO840092L (no) 1984-07-13
DK12084D0 (da) 1984-01-11
GR81735B (da) 1984-12-12
HU190945B (en) 1986-12-28
FI77869B (fi) 1989-01-31
ES8505357A1 (es) 1985-05-16
CH660011A5 (de) 1987-03-13
DE3400733A1 (de) 1984-07-12
AU2322184A (en) 1984-07-19
IT1185050B (it) 1987-11-04
FR2539131A1 (fr) 1984-07-13
FI840088A0 (fi) 1984-01-11
CA1232604A (en) 1988-02-09
SE8400118D0 (sv) 1984-01-11
PH22448A (en) 1988-09-12
NL8400099A (nl) 1984-08-01
ATA8084A (de) 1988-02-15
NZ206816A (en) 1985-09-13
SU1355131A3 (ru) 1987-11-23
PT77946A (en) 1984-02-01

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