DK1084129T3 - Cykliske boroProlinforbindelser - Google Patents
Cykliske boroProlinforbindelserInfo
- Publication number
- DK1084129T3 DK1084129T3 DK99923113T DK99923113T DK1084129T3 DK 1084129 T3 DK1084129 T3 DK 1084129T3 DK 99923113 T DK99923113 T DK 99923113T DK 99923113 T DK99923113 T DK 99923113T DK 1084129 T3 DK1084129 T3 DK 1084129T3
- Authority
- DK
- Denmark
- Prior art keywords
- cyclic boroproline
- boroproline compounds
- compounds
- cyclic
- boroproline
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 125000004122 cyclic group Chemical group 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/04—Esters of boric acids
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Physical Education & Sports Medicine (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8854098P | 1998-06-05 | 1998-06-05 | |
PCT/US1999/010777 WO1999062914A1 (en) | 1998-06-05 | 1999-05-14 | Cyclic boroproline compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1084129T3 true DK1084129T3 (da) | 2003-05-19 |
Family
ID=22211956
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK99923113T DK1084129T3 (da) | 1998-06-05 | 1999-05-14 | Cykliske boroProlinforbindelser |
Country Status (19)
Country | Link |
---|---|
US (1) | US6355614B1 (da) |
EP (1) | EP1084129B1 (da) |
JP (1) | JP2002517401A (da) |
KR (1) | KR100704814B1 (da) |
AR (1) | AR018440A1 (da) |
AT (1) | ATE231512T1 (da) |
AU (1) | AU765370B2 (da) |
BR (1) | BR9910907A (da) |
CA (1) | CA2334155C (da) |
DE (1) | DE69905038T2 (da) |
DK (1) | DK1084129T3 (da) |
ES (1) | ES2189423T3 (da) |
IL (1) | IL139885A (da) |
MY (1) | MY122383A (da) |
NO (1) | NO20006169L (da) |
NZ (1) | NZ508642A (da) |
PT (1) | PT1084129E (da) |
TW (1) | TW575574B (da) |
WO (1) | WO1999062914A1 (da) |
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US20060014697A1 (en) * | 2001-08-22 | 2006-01-19 | Travis Mickle | Pharmaceutical compositions for prevention of overdose or abuse |
US6844316B2 (en) | 2001-09-06 | 2005-01-18 | Probiodrug Ag | Inhibitors of dipeptidyl peptidase I |
AU2002357767C1 (en) * | 2001-11-26 | 2009-03-19 | Trustees Of Tufts College | Peptidomimetic inhibitors of post-proline cleaving enzymes |
CA2466870A1 (en) * | 2001-11-26 | 2003-06-05 | Trustees Of Tufts College | Methods for treating autoimmune disorders, and reagents related thereto |
KR20040095241A (ko) | 2002-02-28 | 2004-11-12 | 프로시디온 리미티드 | 글루타미닐계 dpiv 억제제 |
US7691967B2 (en) | 2002-04-30 | 2010-04-06 | Trustees Of Tufts College | Smart pro-drugs of serine protease inhibitors |
IL166157A0 (en) * | 2002-07-09 | 2006-01-15 | Point Therapeutics Inc | Methods and compositions relating to isoleucine boroproline compounds |
JP4887139B2 (ja) * | 2003-03-25 | 2012-02-29 | 武田薬品工業株式会社 | ジペプチジルペプチダーゼインヒビター |
JP4806628B2 (ja) | 2003-05-05 | 2011-11-02 | プロビオドルグ エージー | グルタミニルシクラーゼ阻害剤 |
US7381537B2 (en) | 2003-05-05 | 2008-06-03 | Probiodrug Ag | Use of inhibitors of glutaminyl cyclases for treatment and prevention of disease |
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US20040247574A1 (en) * | 2003-05-27 | 2004-12-09 | Christopherson Kent W. | Methods for enhancing stem cell engraftment during transplantation |
US7169926B1 (en) | 2003-08-13 | 2007-01-30 | Takeda Pharmaceutical Company Limited | Dipeptidyl peptidase inhibitors |
DE602004010206T2 (de) * | 2003-08-13 | 2008-10-09 | Takeda Pharmaceutical Co. Ltd. | Dipeptidyl Peptidase Inhibitoren. |
US7678909B1 (en) | 2003-08-13 | 2010-03-16 | Takeda Pharmaceutical Company Limited | Dipeptidyl peptidase inhibitors |
JP2007502991A (ja) | 2003-08-20 | 2007-02-15 | バイオサイト インコーポレイテッド | 生物活性ナトリウム利尿ペプチドを測定するための、およびその治療可能性を向上させるための方法および組成物 |
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-
1999
- 1999-05-14 EP EP99923113A patent/EP1084129B1/en not_active Expired - Lifetime
- 1999-05-14 JP JP2000552125A patent/JP2002517401A/ja active Pending
- 1999-05-14 IL IL13988599A patent/IL139885A/en not_active IP Right Cessation
- 1999-05-14 ES ES99923113T patent/ES2189423T3/es not_active Expired - Lifetime
- 1999-05-14 AU AU39958/99A patent/AU765370B2/en not_active Ceased
- 1999-05-14 DK DK99923113T patent/DK1084129T3/da active
- 1999-05-14 AT AT99923113T patent/ATE231512T1/de not_active IP Right Cessation
- 1999-05-14 KR KR1020007013697A patent/KR100704814B1/ko not_active IP Right Cessation
- 1999-05-14 CA CA002334155A patent/CA2334155C/en not_active Expired - Fee Related
- 1999-05-14 NZ NZ508642A patent/NZ508642A/en unknown
- 1999-05-14 DE DE69905038T patent/DE69905038T2/de not_active Expired - Fee Related
- 1999-05-14 BR BR9910907-7A patent/BR9910907A/pt not_active IP Right Cessation
- 1999-05-14 US US09/312,565 patent/US6355614B1/en not_active Expired - Fee Related
- 1999-05-14 WO PCT/US1999/010777 patent/WO1999062914A1/en not_active Application Discontinuation
- 1999-05-14 PT PT99923113T patent/PT1084129E/pt unknown
- 1999-05-25 MY MYPI99002058A patent/MY122383A/en unknown
- 1999-05-28 TW TW88108803A patent/TW575574B/zh not_active IP Right Cessation
- 1999-06-02 AR ARP990102605A patent/AR018440A1/es not_active Application Discontinuation
-
2000
- 2000-12-04 NO NO20006169A patent/NO20006169L/no unknown
Also Published As
Publication number | Publication date |
---|---|
EP1084129A1 (en) | 2001-03-21 |
IL139885A (en) | 2004-05-12 |
MY122383A (en) | 2006-04-29 |
AU765370B2 (en) | 2003-09-18 |
AR018440A1 (es) | 2001-11-14 |
KR100704814B1 (ko) | 2007-04-10 |
NO20006169D0 (no) | 2000-12-04 |
NZ508642A (en) | 2003-10-31 |
CA2334155C (en) | 2005-04-19 |
BR9910907A (pt) | 2002-02-13 |
NO20006169L (no) | 2001-02-05 |
AU3995899A (en) | 1999-12-20 |
ES2189423T3 (es) | 2003-07-01 |
KR20010052548A (ko) | 2001-06-25 |
DE69905038D1 (de) | 2003-02-27 |
TW575574B (en) | 2004-02-11 |
US6355614B1 (en) | 2002-03-12 |
JP2002517401A (ja) | 2002-06-18 |
ATE231512T1 (de) | 2003-02-15 |
WO1999062914A1 (en) | 1999-12-09 |
CA2334155A1 (en) | 1999-12-09 |
PT1084129E (pt) | 2003-06-30 |
DE69905038T2 (de) | 2003-06-05 |
EP1084129B1 (en) | 2003-01-22 |
IL139885A0 (en) | 2002-02-10 |
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