DK0807630T3 - Heterocykliske forbindelser - Google Patents

Heterocykliske forbindelser

Info

Publication number
DK0807630T3
DK0807630T3 DK96901518T DK96901518T DK0807630T3 DK 0807630 T3 DK0807630 T3 DK 0807630T3 DK 96901518 T DK96901518 T DK 96901518T DK 96901518 T DK96901518 T DK 96901518T DK 0807630 T3 DK0807630 T3 DK 0807630T3
Authority
DK
Denmark
Prior art keywords
heterocyclic compounds
chem
halogen atom
formula
halogenocyclopropyl
Prior art date
Application number
DK96901518T
Other languages
English (en)
Inventor
Makoto Takemura
Youichi Kimura
Katsuhiro Kawakami
Kenichi Kimura
Hitoshi Ohki
Norikazu Matsuhashi
Haruko Kawato
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Application granted granted Critical
Publication of DK0807630T3 publication Critical patent/DK0807630T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
DK96901518T 1995-02-02 1996-02-01 Heterocykliske forbindelser DK0807630T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP1561495 1995-02-02
JP1948195 1995-02-07
JP1947895 1995-02-07
PCT/JP1996/000208 WO1996023782A1 (fr) 1995-02-02 1996-02-01 Composes heterocycliques

Publications (1)

Publication Number Publication Date
DK0807630T3 true DK0807630T3 (da) 2003-09-01

Family

ID=27281082

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96901518T DK0807630T3 (da) 1995-02-02 1996-02-01 Heterocykliske forbindelser

Country Status (13)

Country Link
US (1) US5849757A (da)
EP (2) EP0807630B1 (da)
KR (1) KR100389773B1 (da)
AT (2) ATE239720T1 (da)
CA (1) CA2212007C (da)
DE (2) DE69637717D1 (da)
DK (1) DK0807630T3 (da)
ES (2) ES2315432T3 (da)
FI (1) FI973207A (da)
NO (1) NO314546B1 (da)
PT (1) PT807630E (da)
TW (1) TW487701B (da)
WO (1) WO1996023782A1 (da)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA003321B1 (ru) * 1995-11-22 2003-04-24 Дайити Фармасьютикал Ко., Лтд. Производные аминоциклоалкилпирролидона и антибактериальное лекарственное средство на их основе
US6121285A (en) 1995-11-22 2000-09-19 Daiichi Pharmaceutical Co., Ltd. Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
TW519542B (en) * 1996-09-27 2003-02-01 Daiichi Seiyaku Co Bicyclic amine derivative
MY119816A (en) * 1997-05-30 2005-07-29 Daiichi Seiyaku Co Substituted cyclobutylamine derivatives
PL339408A1 (en) 1997-09-15 2000-12-18 Procter & Gamble Antimicrobial quinolones, agents containing them and their applications
GB9822440D0 (en) * 1998-10-14 1998-12-09 Smithkline Beecham Plc Medicaments
EP1167344A4 (en) * 1999-03-17 2004-06-16 Daiichi Seiyaku Co PROCESS FOR THE PRODUCTION OF 5-AMINO-8-ALKYLQUINOLO NECARBOXYLIC ACID DERIVATIVES AND INTERMEDIATE PRODUCTS IN THE PRODUCTION
CA2408806A1 (en) * 2000-03-31 2001-10-04 Masayasu Sekiguchi Quinolonecarboxylic acid derivative
CA2429440C (en) * 2000-11-20 2009-12-29 Daiichi Pharmaceutical Co., Ltd. Dehalogeno-compounds
GB0112834D0 (en) * 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
KR101041277B1 (ko) * 2002-05-17 2011-06-14 다이이찌 세이야꾸 가부시기가이샤 퀴놀론카르복실산 유도체의 제조방법
US6875784B2 (en) 2002-10-09 2005-04-05 Pharmacia & Upjohn Company Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
WO2004108680A1 (ja) * 2003-06-06 2004-12-16 Daiichi Pharmaceutical Co., Ltd. 光学活性なキノロンカルボン酸誘導体の製造中間体およびその製造法
EP1634879A4 (en) * 2003-06-19 2007-09-05 Daiichi Seiyaku Co METHOD FOR THE SELECTIVE INTRODUCTION OF AN AMINO SUBSTITUENT
WO2005030752A1 (ja) * 2003-09-29 2005-04-07 Daiichi Pharmaceutical Co., Ltd. 8−シアノキノロンカルボン酸誘導体
HUE025625T2 (en) 2003-12-12 2016-04-28 Daiichi Sankyo Co Ltd Intermediates for the preparation of optically active cyclopropylamine derivatives and a process for the preparation of intermediates
MX2008012328A (es) 2006-03-28 2008-10-09 Procter & Gamble Sales de malato, y polimorfos de acido (3s,5s)-7-[3-amino-5-metil- piperidinil]-1-ciclopropil-1,4-dihidro-8-metoxi-4-oxo-3-quinolinc arboxilico.
JP2009531418A (ja) 2006-03-28 2009-09-03 ザ プロクター アンド ギャンブル カンパニー キノロン中間体調製のためのカップリング方法
PL2097400T3 (pl) 2007-01-05 2013-11-29 Daiichi Sankyo Co Ltd Skondensowane podstawione pochodne aminopirolidyny
US8278313B2 (en) 2008-03-11 2012-10-02 Abbott Laboratories Macrocyclic spiro pyrimidine derivatives
US8436005B2 (en) 2008-04-03 2013-05-07 Abbott Laboratories Macrocyclic pyrimidine derivatives
US10300155B2 (en) 2015-12-31 2019-05-28 Washington University Alpha-synuclein ligands

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5772981A (en) * 1980-10-22 1982-05-07 Dainippon Pharmaceut Co Ltd 1,8-naphthyridine derivative and its salt
CS274601B2 (en) * 1983-07-27 1991-09-15 Dainippon Pharmaceutical Co Method of 1,8-naphthyridine derivative production
JPS60260577A (ja) * 1984-06-06 1985-12-23 Dainippon Pharmaceut Co Ltd 1,8−ナフチリジン誘導体
IL79189A (en) * 1985-06-26 1990-07-12 Daiichi Seiyaku Co Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
IL90062A (en) * 1988-04-27 1994-10-07 Daiichi Seiyaku Co History of pyridonecarboxylic acid, their preparation and pharmaceutical preparations containing them
JP2844079B2 (ja) * 1988-05-23 1999-01-06 塩野義製薬株式会社 ピリドンカルボン酸系抗菌剤
HU219403B (hu) * 1989-08-16 2001-04-28 Pfizer Inc. Azabiciklo-csoporttal helyettesített kinolon- és naftiridon-karbonsavak és eljárás ezek előállítására
RU2100351C1 (ru) * 1991-05-28 1997-12-27 Дайити Фармасьютикал Ко., Лтд. Производные пиридонкарбоновой кислоты и композиция на их основе
KR960011370B1 (ko) * 1991-12-31 1996-08-22 재단법인 한국화학연구소 스피로알킬아민 유도체와 그의 제조방법
EP0550016A1 (en) * 1991-12-31 1993-07-07 Korea Research Institute Of Chemical Technology Novel quinolone carboxylic acid derivatives and processes for preparing same
US5990106A (en) * 1994-02-04 1999-11-23 Dainippon Pharmaceutical Co., Ltd. Bicyclic amino group-substituted pyridonecarboxylic acid derivatives, esters thereof and salts thereof, and bicyclic amines useful as intermediates thereof
EA003321B1 (ru) * 1995-11-22 2003-04-24 Дайити Фармасьютикал Ко., Лтд. Производные аминоциклоалкилпирролидона и антибактериальное лекарственное средство на их основе

Also Published As

Publication number Publication date
ATE239720T1 (de) 2003-05-15
ATE411309T1 (de) 2008-10-15
EP1304329A2 (en) 2003-04-23
DE69627985T2 (de) 2004-02-19
CA2212007C (en) 2004-09-14
FI973207A (fi) 1997-10-01
WO1996023782A1 (fr) 1996-08-08
DE69637717D1 (de) 2008-11-27
EP0807630A1 (en) 1997-11-19
US5849757A (en) 1998-12-15
CA2212007A1 (en) 1996-08-08
EP1304329B1 (en) 2008-10-15
NO973530L (no) 1997-10-02
KR19980701860A (ko) 1998-06-25
ES2315432T3 (es) 2009-04-01
KR100389773B1 (ko) 2003-10-23
NO314546B1 (no) 2003-04-07
EP0807630A4 (en) 1998-05-13
EP1304329A3 (en) 2004-09-15
TW487701B (en) 2002-05-21
FI973207A0 (fi) 1997-08-01
EP0807630B1 (en) 2003-05-07
NO973530D0 (no) 1997-07-31
ES2198474T3 (es) 2004-02-01
PT807630E (pt) 2003-08-29
DE69627985D1 (de) 2003-06-12

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