DK0807630T3 - Heterocykliske forbindelser - Google Patents
Heterocykliske forbindelserInfo
- Publication number
- DK0807630T3 DK0807630T3 DK96901518T DK96901518T DK0807630T3 DK 0807630 T3 DK0807630 T3 DK 0807630T3 DK 96901518 T DK96901518 T DK 96901518T DK 96901518 T DK96901518 T DK 96901518T DK 0807630 T3 DK0807630 T3 DK 0807630T3
- Authority
- DK
- Denmark
- Prior art keywords
- heterocyclic compounds
- chem
- halogen atom
- formula
- halogenocyclopropyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1561495 | 1995-02-02 | ||
JP1948195 | 1995-02-07 | ||
JP1947895 | 1995-02-07 | ||
PCT/JP1996/000208 WO1996023782A1 (fr) | 1995-02-02 | 1996-02-01 | Composes heterocycliques |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0807630T3 true DK0807630T3 (da) | 2003-09-01 |
Family
ID=27281082
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK96901518T DK0807630T3 (da) | 1995-02-02 | 1996-02-01 | Heterocykliske forbindelser |
Country Status (13)
Country | Link |
---|---|
US (1) | US5849757A (da) |
EP (2) | EP0807630B1 (da) |
KR (1) | KR100389773B1 (da) |
AT (2) | ATE239720T1 (da) |
CA (1) | CA2212007C (da) |
DE (2) | DE69637717D1 (da) |
DK (1) | DK0807630T3 (da) |
ES (2) | ES2315432T3 (da) |
FI (1) | FI973207A (da) |
NO (1) | NO314546B1 (da) |
PT (1) | PT807630E (da) |
TW (1) | TW487701B (da) |
WO (1) | WO1996023782A1 (da) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA003321B1 (ru) * | 1995-11-22 | 2003-04-24 | Дайити Фармасьютикал Ко., Лтд. | Производные аминоциклоалкилпирролидона и антибактериальное лекарственное средство на их основе |
US6121285A (en) | 1995-11-22 | 2000-09-19 | Daiichi Pharmaceutical Co., Ltd. | Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives |
TW519542B (en) * | 1996-09-27 | 2003-02-01 | Daiichi Seiyaku Co | Bicyclic amine derivative |
MY119816A (en) * | 1997-05-30 | 2005-07-29 | Daiichi Seiyaku Co | Substituted cyclobutylamine derivatives |
PL339408A1 (en) | 1997-09-15 | 2000-12-18 | Procter & Gamble | Antimicrobial quinolones, agents containing them and their applications |
GB9822440D0 (en) * | 1998-10-14 | 1998-12-09 | Smithkline Beecham Plc | Medicaments |
EP1167344A4 (en) * | 1999-03-17 | 2004-06-16 | Daiichi Seiyaku Co | PROCESS FOR THE PRODUCTION OF 5-AMINO-8-ALKYLQUINOLO NECARBOXYLIC ACID DERIVATIVES AND INTERMEDIATE PRODUCTS IN THE PRODUCTION |
CA2408806A1 (en) * | 2000-03-31 | 2001-10-04 | Masayasu Sekiguchi | Quinolonecarboxylic acid derivative |
CA2429440C (en) * | 2000-11-20 | 2009-12-29 | Daiichi Pharmaceutical Co., Ltd. | Dehalogeno-compounds |
GB0112834D0 (en) * | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
KR101041277B1 (ko) * | 2002-05-17 | 2011-06-14 | 다이이찌 세이야꾸 가부시기가이샤 | 퀴놀론카르복실산 유도체의 제조방법 |
US6875784B2 (en) | 2002-10-09 | 2005-04-05 | Pharmacia & Upjohn Company | Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives |
WO2004108680A1 (ja) * | 2003-06-06 | 2004-12-16 | Daiichi Pharmaceutical Co., Ltd. | 光学活性なキノロンカルボン酸誘導体の製造中間体およびその製造法 |
EP1634879A4 (en) * | 2003-06-19 | 2007-09-05 | Daiichi Seiyaku Co | METHOD FOR THE SELECTIVE INTRODUCTION OF AN AMINO SUBSTITUENT |
WO2005030752A1 (ja) * | 2003-09-29 | 2005-04-07 | Daiichi Pharmaceutical Co., Ltd. | 8−シアノキノロンカルボン酸誘導体 |
HUE025625T2 (en) | 2003-12-12 | 2016-04-28 | Daiichi Sankyo Co Ltd | Intermediates for the preparation of optically active cyclopropylamine derivatives and a process for the preparation of intermediates |
MX2008012328A (es) | 2006-03-28 | 2008-10-09 | Procter & Gamble | Sales de malato, y polimorfos de acido (3s,5s)-7-[3-amino-5-metil- piperidinil]-1-ciclopropil-1,4-dihidro-8-metoxi-4-oxo-3-quinolinc arboxilico. |
JP2009531418A (ja) | 2006-03-28 | 2009-09-03 | ザ プロクター アンド ギャンブル カンパニー | キノロン中間体調製のためのカップリング方法 |
PL2097400T3 (pl) | 2007-01-05 | 2013-11-29 | Daiichi Sankyo Co Ltd | Skondensowane podstawione pochodne aminopirolidyny |
US8278313B2 (en) | 2008-03-11 | 2012-10-02 | Abbott Laboratories | Macrocyclic spiro pyrimidine derivatives |
US8436005B2 (en) | 2008-04-03 | 2013-05-07 | Abbott Laboratories | Macrocyclic pyrimidine derivatives |
US10300155B2 (en) | 2015-12-31 | 2019-05-28 | Washington University | Alpha-synuclein ligands |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5772981A (en) * | 1980-10-22 | 1982-05-07 | Dainippon Pharmaceut Co Ltd | 1,8-naphthyridine derivative and its salt |
CS274601B2 (en) * | 1983-07-27 | 1991-09-15 | Dainippon Pharmaceutical Co | Method of 1,8-naphthyridine derivative production |
JPS60260577A (ja) * | 1984-06-06 | 1985-12-23 | Dainippon Pharmaceut Co Ltd | 1,8−ナフチリジン誘導体 |
IL79189A (en) * | 1985-06-26 | 1990-07-12 | Daiichi Seiyaku Co | Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them |
JPH0676400B2 (ja) * | 1987-08-25 | 1994-09-28 | 大日本製薬株式会社 | 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩 |
IL90062A (en) * | 1988-04-27 | 1994-10-07 | Daiichi Seiyaku Co | History of pyridonecarboxylic acid, their preparation and pharmaceutical preparations containing them |
JP2844079B2 (ja) * | 1988-05-23 | 1999-01-06 | 塩野義製薬株式会社 | ピリドンカルボン酸系抗菌剤 |
HU219403B (hu) * | 1989-08-16 | 2001-04-28 | Pfizer Inc. | Azabiciklo-csoporttal helyettesített kinolon- és naftiridon-karbonsavak és eljárás ezek előállítására |
RU2100351C1 (ru) * | 1991-05-28 | 1997-12-27 | Дайити Фармасьютикал Ко., Лтд. | Производные пиридонкарбоновой кислоты и композиция на их основе |
KR960011370B1 (ko) * | 1991-12-31 | 1996-08-22 | 재단법인 한국화학연구소 | 스피로알킬아민 유도체와 그의 제조방법 |
EP0550016A1 (en) * | 1991-12-31 | 1993-07-07 | Korea Research Institute Of Chemical Technology | Novel quinolone carboxylic acid derivatives and processes for preparing same |
US5990106A (en) * | 1994-02-04 | 1999-11-23 | Dainippon Pharmaceutical Co., Ltd. | Bicyclic amino group-substituted pyridonecarboxylic acid derivatives, esters thereof and salts thereof, and bicyclic amines useful as intermediates thereof |
EA003321B1 (ru) * | 1995-11-22 | 2003-04-24 | Дайити Фармасьютикал Ко., Лтд. | Производные аминоциклоалкилпирролидона и антибактериальное лекарственное средство на их основе |
-
1996
- 1996-02-01 CA CA002212007A patent/CA2212007C/en not_active Expired - Fee Related
- 1996-02-01 PT PT96901518T patent/PT807630E/pt unknown
- 1996-02-01 WO PCT/JP1996/000208 patent/WO1996023782A1/ja active IP Right Grant
- 1996-02-01 DE DE69637717T patent/DE69637717D1/de not_active Expired - Lifetime
- 1996-02-01 TW TW85101378A patent/TW487701B/zh active
- 1996-02-01 US US08/875,678 patent/US5849757A/en not_active Expired - Fee Related
- 1996-02-01 KR KR1019970705257A patent/KR100389773B1/ko not_active IP Right Cessation
- 1996-02-01 AT AT96901518T patent/ATE239720T1/de not_active IP Right Cessation
- 1996-02-01 AT AT03000883T patent/ATE411309T1/de not_active IP Right Cessation
- 1996-02-01 EP EP96901518A patent/EP0807630B1/en not_active Expired - Lifetime
- 1996-02-01 EP EP03000883A patent/EP1304329B1/en not_active Expired - Lifetime
- 1996-02-01 ES ES03000883T patent/ES2315432T3/es not_active Expired - Lifetime
- 1996-02-01 DE DE69627985T patent/DE69627985T2/de not_active Expired - Fee Related
- 1996-02-01 ES ES96901518T patent/ES2198474T3/es not_active Expired - Lifetime
- 1996-02-01 DK DK96901518T patent/DK0807630T3/da active
-
1997
- 1997-07-31 NO NO19973530A patent/NO314546B1/no not_active IP Right Cessation
- 1997-08-01 FI FI973207A patent/FI973207A/fi unknown
Also Published As
Publication number | Publication date |
---|---|
ATE239720T1 (de) | 2003-05-15 |
ATE411309T1 (de) | 2008-10-15 |
EP1304329A2 (en) | 2003-04-23 |
DE69627985T2 (de) | 2004-02-19 |
CA2212007C (en) | 2004-09-14 |
FI973207A (fi) | 1997-10-01 |
WO1996023782A1 (fr) | 1996-08-08 |
DE69637717D1 (de) | 2008-11-27 |
EP0807630A1 (en) | 1997-11-19 |
US5849757A (en) | 1998-12-15 |
CA2212007A1 (en) | 1996-08-08 |
EP1304329B1 (en) | 2008-10-15 |
NO973530L (no) | 1997-10-02 |
KR19980701860A (ko) | 1998-06-25 |
ES2315432T3 (es) | 2009-04-01 |
KR100389773B1 (ko) | 2003-10-23 |
NO314546B1 (no) | 2003-04-07 |
EP0807630A4 (en) | 1998-05-13 |
EP1304329A3 (en) | 2004-09-15 |
TW487701B (en) | 2002-05-21 |
FI973207A0 (fi) | 1997-08-01 |
EP0807630B1 (en) | 2003-05-07 |
NO973530D0 (no) | 1997-07-31 |
ES2198474T3 (es) | 2004-02-01 |
PT807630E (pt) | 2003-08-29 |
DE69627985D1 (de) | 2003-06-12 |
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