DE60218493D1 - Substituierte 7-aza-ä2.2.1übicycloheptane für die behandlung von krankheiten - Google Patents

Substituierte 7-aza-ä2.2.1übicycloheptane für die behandlung von krankheiten

Info

Publication number
DE60218493D1
DE60218493D1 DE60218493T DE60218493T DE60218493D1 DE 60218493 D1 DE60218493 D1 DE 60218493D1 DE 60218493 T DE60218493 T DE 60218493T DE 60218493 T DE60218493 T DE 60218493T DE 60218493 D1 DE60218493 D1 DE 60218493D1
Authority
DE
Germany
Prior art keywords
aza
diseases
substituted
treatment
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60218493T
Other languages
English (en)
Inventor
Donn G Wishka
Daniel Patrick Walker
Jeffrey W Corbett
Steven Charles Reitz
Mark R Rauckhorst
Vincent E Groppi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co LLC
Original Assignee
Pharmacia and Upjohn Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn Co LLC filed Critical Pharmacia and Upjohn Co LLC
Application granted granted Critical
Publication of DE60218493D1 publication Critical patent/DE60218493D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE60218493T 2001-09-12 2002-09-04 Substituierte 7-aza-ä2.2.1übicycloheptane für die behandlung von krankheiten Expired - Lifetime DE60218493D1 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US32234601P 2001-09-12 2001-09-12
US32210001P 2001-09-12 2001-09-12
US32233301P 2001-09-12 2001-09-12
US39953002P 2002-07-30 2002-07-30
PCT/US2002/025959 WO2003022856A1 (en) 2001-09-12 2002-09-04 Substituted 7-aza[2.2.1] bicycloheptanes for the treatment of diseases

Publications (1)

Publication Number Publication Date
DE60218493D1 true DE60218493D1 (de) 2007-04-12

Family

ID=27502238

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60218493T Expired - Lifetime DE60218493D1 (de) 2001-09-12 2002-09-04 Substituierte 7-aza-ä2.2.1übicycloheptane für die behandlung von krankheiten

Country Status (10)

Country Link
US (1) US20030105089A1 (de)
EP (1) EP1425286B1 (de)
JP (1) JP2005527472A (de)
AR (1) AR036779A1 (de)
AT (1) ATE355293T1 (de)
BR (1) BR0212477A (de)
CA (1) CA2460075A1 (de)
DE (1) DE60218493D1 (de)
MX (1) MXPA04002377A (de)
WO (1) WO2003022856A1 (de)

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Also Published As

Publication number Publication date
BR0212477A (pt) 2004-08-24
US20030105089A1 (en) 2003-06-05
JP2005527472A (ja) 2005-09-15
EP1425286B1 (de) 2007-02-28
CA2460075A1 (en) 2003-03-20
WO2003022856A1 (en) 2003-03-20
EP1425286A1 (de) 2004-06-09
MXPA04002377A (es) 2004-11-22
ATE355293T1 (de) 2006-03-15
AR036779A1 (es) 2004-10-06

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