DE3680000D1 - Stabilisierte aktive formen von vitamin-d3. - Google Patents

Stabilisierte aktive formen von vitamin-d3.

Info

Publication number
DE3680000D1
DE3680000D1 DE8686101828T DE3680000T DE3680000D1 DE 3680000 D1 DE3680000 D1 DE 3680000D1 DE 8686101828 T DE8686101828 T DE 8686101828T DE 3680000 T DE3680000 T DE 3680000T DE 3680000 D1 DE3680000 D1 DE 3680000D1
Authority
DE
Germany
Prior art keywords
vitamin
active forms
stabilized active
stabilized
forms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE8686101828T
Other languages
English (en)
Inventor
Kaoru Nemoto
Kazuo Igusa
Toshichika Ogasawara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chugai Pharmaceutical Co Ltd
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DE3680000D1 publication Critical patent/DE3680000D1/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/59Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE8686101828T 1985-02-14 1986-02-13 Stabilisierte aktive formen von vitamin-d3. Expired - Fee Related DE3680000D1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2807385 1985-02-14

Publications (1)

Publication Number Publication Date
DE3680000D1 true DE3680000D1 (de) 1991-08-08

Family

ID=12238593

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8686101828T Expired - Fee Related DE3680000D1 (de) 1985-02-14 1986-02-13 Stabilisierte aktive formen von vitamin-d3.

Country Status (4)

Country Link
US (1) US4836957A (de)
EP (1) EP0191489B1 (de)
JP (1) JPS6217A (de)
DE (1) DE3680000D1 (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1272953A (en) * 1984-10-08 1990-08-21 Yuji Makino Pharmaceutical composition for external use containing active-type vitamin d.sub.3
JPH02274A (ja) * 1987-10-14 1990-01-05 Toyo Jozo Co Ltd 新規な25−ヒドロキシビタミンd↓3誘導体およびその製造法およびそれを用いた定量法
US5182274A (en) * 1988-09-26 1993-01-26 Teijin Limited Stabilized aqueous preparation of active form of vitamin d3
JP2525478B2 (ja) * 1989-03-01 1996-08-21 帝人株式会社 安定性の改良された活性型ビタミンd▲下3▼類固型製剤
EP0508756B1 (de) * 1991-04-09 1996-10-23 Takeda Chemical Industries, Ltd. Stabilisiertes Vitamin D Arzneimittel
CN1062877C (zh) * 1995-07-27 2001-03-07 中国科学院长春应用化学研究所 全溶性不同分子量聚苯胺及其衍生物的制备
US6432422B1 (en) * 1997-12-09 2002-08-13 Chugai Seiyaku Kabushiki Kaisha Creams containing vitamin D3 derivatives
US6491936B1 (en) 1997-12-09 2002-12-10 Chugai Seiyaku Kabushiki Kaisha Creams containing vitamin D3 derivatives
DK1044017T3 (da) * 1998-01-05 2008-12-08 Univ Johns Hopkins Kosttilskud til dialysepatienter
JP2002500869A (ja) * 1998-01-22 2002-01-15 アボット・ラボラトリーズ 加水分解したタンパク質を含む栄養食品中のビタミンdの安定性を改善する方法および該方法により得られる食品
US7141544B2 (en) * 2003-10-10 2006-11-28 Baxter International, Inc. Stabilization of pharmaceutical protein formulations with small peptides
WO2007000884A1 (ja) * 2005-06-29 2007-01-04 National University Corporation Kanazawa University 骨・関節疾患の予防・治療剤およびそのスクリーニング方法
AU2007296924A1 (en) * 2006-09-14 2008-03-20 Dsm Ip Assets B.V. Food supplementation composition containing one or more vitamin D3 compounds and one or more magnesium salts
JP5652723B2 (ja) * 2012-08-17 2015-01-14 フォーモサ・ラボラトリーズ・インコーポレーテッド マキサカルシトールの新しい結晶形態
JPWO2015119183A1 (ja) * 2014-02-05 2017-03-23 協和発酵キリン株式会社 活性型ビタミンd3またはその誘導体を含有する液剤
JP6905538B2 (ja) * 2016-12-28 2021-07-21 中外製薬株式会社 Ed−71の固体分散体および油分分散体を含む医薬組成物
JP6952468B2 (ja) * 2017-01-31 2021-10-20 中外製薬株式会社 ビタミンd化合物を含有する水性医薬組成物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH304182A (de) * 1951-10-26 1954-12-31 C M Kuehn & Co Verfahren zum Stabilisieren von oxydationsempfindlichen organischen Stoffen.
GB799068A (en) * 1955-12-29 1958-07-30 Hoffmann La Roche A stabilized vitamin-d composition and a process for the production thereof
JPS51128417A (en) * 1975-04-28 1976-11-09 Teijin Ltd A method for stabilizing active vitamin d3 derivatives
JPS603045B2 (ja) * 1976-04-19 1985-01-25 中外製薬株式会社 1α―ヒドロキシビタミンD類軟カプセルの製造方法
JPS53136512A (en) * 1977-04-28 1978-11-29 Chugai Pharmaceut Co Ltd Stable oily preparation containing 1alpha-hydroxyvitamin d
JPS5569562A (en) * 1978-11-21 1980-05-26 Teijin Ltd Stabilization of active vitamin d3 derivative
DE2921852A1 (de) * 1979-05-29 1980-12-11 Fresenius Chem Pharm Ind Lipide senkendes mittel
JPS59193814A (ja) * 1983-04-20 1984-11-02 Ajinomoto Co Inc アミノ酸含有脂肪乳剤
JPS6025918A (ja) * 1983-07-25 1985-02-08 Ajinomoto Co Inc 脂溶性薬物含有水性液

Also Published As

Publication number Publication date
EP0191489B1 (de) 1991-07-03
EP0191489A2 (de) 1986-08-20
US4836957A (en) 1989-06-06
EP0191489A3 (en) 1987-08-26
JPS6217A (ja) 1987-01-06

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee