DE2824065A1 - Acylderivate - Google Patents

Acylderivate

Info

Publication number
DE2824065A1
DE2824065A1 DE19782824065 DE2824065A DE2824065A1 DE 2824065 A1 DE2824065 A1 DE 2824065A1 DE 19782824065 DE19782824065 DE 19782824065 DE 2824065 A DE2824065 A DE 2824065A DE 2824065 A1 DE2824065 A1 DE 2824065A1
Authority
DE
Germany
Prior art keywords
salts
methyl
formula
compounds
hydrates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE19782824065
Other languages
German (de)
English (en)
Inventor
Marc Dr Montavon
Roland Dr Reiner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of DE2824065A1 publication Critical patent/DE2824065A1/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DE19782824065 1977-06-03 1978-06-01 Acylderivate Withdrawn DE2824065A1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU77485 1977-06-03
CH314278 1978-03-22

Publications (1)

Publication Number Publication Date
DE2824065A1 true DE2824065A1 (de) 1978-12-14

Family

ID=25692293

Family Applications (2)

Application Number Title Priority Date Filing Date
DE19782824065 Withdrawn DE2824065A1 (de) 1977-06-03 1978-06-01 Acylderivate
DE7878100078T Expired DE2860248D1 (en) 1977-06-03 1978-06-01 New cephalosporin derivatives, their preparations and their pharmaceutical compositions

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE7878100078T Expired DE2860248D1 (en) 1977-06-03 1978-06-01 New cephalosporin derivatives, their preparations and their pharmaceutical compositions

Country Status (26)

Country Link
EP (1) EP0000005B1 (fr)
JP (1) JPS5412394A (fr)
AR (1) AR225134A1 (fr)
AT (2) AT362501B (fr)
AU (1) AU518648B2 (fr)
BR (1) BR7803565A (fr)
CA (1) CA1114808A (fr)
CU (1) CU21118A (fr)
DE (2) DE2824065A1 (fr)
DK (1) DK246878A (fr)
ES (2) ES470442A1 (fr)
FI (1) FI781754A (fr)
FR (1) FR2393000A1 (fr)
GB (1) GB1599232A (fr)
GR (1) GR73554B (fr)
HU (1) HU182498B (fr)
IE (1) IE46903B1 (fr)
IL (1) IL54803A (fr)
IT (1) IT1098306B (fr)
MC (1) MC1195A1 (fr)
NL (1) NL7805715A (fr)
NO (1) NO781934L (fr)
NZ (1) NZ187392A (fr)
PH (1) PH14653A (fr)
PT (1) PT68134A (fr)
SE (1) SE7806465L (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0008372A1 (fr) * 1978-07-19 1980-03-05 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Esters et éthers de céphalosporines facilement hydrolysables, leur préparation et compositions les contenant

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4200745A (en) * 1977-12-20 1980-04-29 Eli Lilly And Company 7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins
FR2432521A1 (fr) * 1978-03-31 1980-02-29 Roussel Uclaf Nouvelles oximes o-substituees derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
MC1259A1 (fr) * 1978-05-30 1980-01-14 Hoffmann La Roche Derives acyles
US4472574A (en) * 1981-05-22 1984-09-18 Hoffman-La Roche Inc. Process for the manufacture of a cephem carboxylic acid derivative
US4698338A (en) * 1986-02-19 1987-10-06 Eli Lilly And Company 7[2-(2-aminothiazol-4-yl)-2-benzyloximino]acetamido-3[4-alkyl-5-oxo-6-hydroxy-3,4-dihydro-1,2,4-triazin-3-yl]thiomethyl cephalosporins

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1399086A (en) * 1971-05-14 1975-06-25 Glaxo Lab Ltd Cephalosporin compounds
CH609989A5 (en) * 1974-06-21 1979-03-30 Hoffmann La Roche Process for the preparation of acyl derivatives
CA1100129A (fr) * 1974-08-02 1981-04-28 William H.W. Lunn Traduction non-disponible
GB1555471A (en) * 1975-06-19 1979-11-14 Glaxo Lab Ltd 7 carbamoylalkoxyimino acetamido 3 em 4 carboxylic acidsand derivatives thereof
GB1576625A (en) * 1976-04-12 1980-10-08 Fujisawa Pharmaceutical Co Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof
GB1596278A (en) * 1976-11-30 1981-08-26 Glaxo Operations Ltd 7-(-oxyimino-acetamino)cephalosporin derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0008372A1 (fr) * 1978-07-19 1980-03-05 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Esters et éthers de céphalosporines facilement hydrolysables, leur préparation et compositions les contenant

Also Published As

Publication number Publication date
AU3658878A (en) 1979-12-06
IE46903B1 (en) 1983-11-02
SE7806465L (sv) 1978-12-04
BR7803565A (pt) 1979-02-20
NL7805715A (nl) 1978-12-05
IL54803A (en) 1982-01-31
EP0000005A1 (fr) 1978-12-20
PH14653A (en) 1981-10-14
ES470442A1 (es) 1979-10-01
ATA345980A (de) 1981-05-15
HU182498B (en) 1984-01-30
CA1114808A (fr) 1981-12-22
AT365197B (de) 1981-12-28
CU21118A (es) 1983-04-06
FR2393000B1 (fr) 1982-10-29
IE781056L (en) 1978-12-03
NZ187392A (en) 1984-05-31
NO781934L (no) 1978-12-05
ES478115A1 (es) 1979-06-01
AR225134A1 (es) 1982-02-26
DK246878A (da) 1978-12-04
FI781754A (fi) 1978-12-04
GB1599232A (en) 1981-09-30
GR73554B (fr) 1984-03-14
MC1195A1 (fr) 1979-02-23
PT68134A (en) 1978-07-01
IT7824165A0 (it) 1978-06-02
FR2393000A1 (fr) 1978-12-29
IL54803A0 (en) 1978-07-31
ATA403578A (de) 1980-10-15
IT1098306B (it) 1985-09-07
AT362501B (de) 1981-05-25
JPS5412394A (en) 1979-01-30
AU518648B2 (en) 1981-10-15
DE2860248D1 (en) 1981-01-29
EP0000005B1 (fr) 1980-10-29

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Legal Events

Date Code Title Description
8139 Disposal/non-payment of the annual fee