CY1121313T1 - Φαρμακευτικη διεργασια και ενδιαμεσα - Google Patents

Φαρμακευτικη διεργασια και ενδιαμεσα

Info

Publication number
CY1121313T1
CY1121313T1 CY20181101287T CY181101287T CY1121313T1 CY 1121313 T1 CY1121313 T1 CY 1121313T1 CY 20181101287 T CY20181101287 T CY 20181101287T CY 181101287 T CY181101287 T CY 181101287T CY 1121313 T1 CY1121313 T1 CY 1121313T1
Authority
CY
Cyprus
Prior art keywords
pharmaceutical process
pharmaceutical
hydrates
intermediates
compound
Prior art date
Application number
CY20181101287T
Other languages
English (en)
Inventor
Benedict MCKEEVER
Louis Joseph Diorazio
Martin Francis Jones
Leigh FERRIS
Sophie Laure Marie JANBON
Pawel Stanislaw SIEDLECKI
Gwydion Huw Churchill
Peter Alan CRAFTS
Original Assignee
Rigel Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rigel Pharmaceuticals, Inc. filed Critical Rigel Pharmaceuticals, Inc.
Publication of CY1121313T1 publication Critical patent/CY1121313T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Η παρούσα αποκάλυψη παρέχει διεργασίες και ενδιάμεσα στην ευρείας κλίμακας παρασκευή της ένωσης του τύπου (I) ή υδριτών αυτής.
CY20181101287T 2013-12-20 2018-12-04 Φαρμακευτικη διεργασια και ενδιαμεσα CY1121313T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361919671P 2013-12-20 2013-12-20
PCT/US2014/071613 WO2015095765A1 (en) 2013-12-20 2014-12-19 Pharmaceutical process and intermediates

Publications (1)

Publication Number Publication Date
CY1121313T1 true CY1121313T1 (el) 2020-05-29

Family

ID=52358996

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20181101287T CY1121313T1 (el) 2013-12-20 2018-12-04 Φαρμακευτικη διεργασια και ενδιαμεσα

Country Status (16)

Country Link
US (2) US9388203B2 (el)
EP (1) EP3083648B1 (el)
JP (1) JP6522005B2 (el)
CN (1) CN105849115B (el)
CA (2) CA2934535C (el)
CY (1) CY1121313T1 (el)
DK (1) DK3083648T3 (el)
ES (1) ES2701088T3 (el)
HR (1) HRP20181933T1 (el)
HU (1) HUE042204T2 (el)
LT (1) LT3083648T (el)
PL (1) PL3083648T3 (el)
PT (1) PT3083648T (el)
RS (1) RS58084B1 (el)
SI (1) SI3083648T1 (el)
WO (1) WO2015095765A1 (el)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109912622A (zh) * 2019-03-20 2019-06-21 中国药科大学 一种福他替尼关键中间体的制备方法及其中间体和利用中间体制备福他替尼的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20120062863A (ko) 2003-07-30 2012-06-14 리겔 파마슈티칼스, 인크. 자가면역 질환의 치료 또는 예방에 사용하기 위한 2,4-피리미딘디아민 화합물
EP2161275A1 (en) * 2005-01-19 2010-03-10 Rigel Pharmaceuticals, Inc. Prodrugs of 2,4-pyrimidinediamine compounds and their uses
EP2078026B1 (en) * 2006-11-21 2012-01-04 Rigel Pharmaceuticals, Inc. Prodrug salts of 2, 4-pyrimidinediamine compounds and their uses
UA108077C2 (xx) * 2009-07-02 2015-03-25 Синтез динатрієвої солі n4-(2,2-диметил-4-$(дигідрофосфонокси)метил]-3-оксо-5-піридо$1,4]оксазин-6-іл)-5-фтор-n2-(3,4,5-триметоксифеніл)-2,4-піримідиндіаміну
CA2780777C (en) * 2009-11-20 2017-12-05 Rigel Pharmaceuticals, Inc. 2,4-pyrimidinediamine compounds and prodrugs thereof and their uses

Also Published As

Publication number Publication date
CN105849115A (zh) 2016-08-10
WO2015095765A1 (en) 2015-06-25
LT3083648T (lt) 2019-01-25
CA2934535C (en) 2023-03-28
PT3083648T (pt) 2018-12-14
US20160355531A1 (en) 2016-12-08
PL3083648T3 (pl) 2019-05-31
ES2701088T3 (es) 2019-02-20
EP3083648A1 (en) 2016-10-26
CA3186267A1 (en) 2015-06-25
US9388203B2 (en) 2016-07-12
CN105849115B (zh) 2019-06-11
JP2017503018A (ja) 2017-01-26
CA2934535A1 (en) 2015-06-25
SI3083648T1 (sl) 2019-02-28
HUE042204T2 (hu) 2019-06-28
RS58084B1 (sr) 2019-02-28
US20150175639A1 (en) 2015-06-25
EP3083648B1 (en) 2018-09-12
JP6522005B2 (ja) 2019-05-29
DK3083648T3 (en) 2019-01-07
US9695204B2 (en) 2017-07-04
HRP20181933T1 (hr) 2019-01-11

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