CY1109186T1 - COMPOSITION OF DIOXYBYTYNYL HEXAMETHYL-DOTA - Google Patents

COMPOSITION OF DIOXYBYTYNYL HEXAMETHYL-DOTA

Info

Publication number
CY1109186T1
CY1109186T1 CY20091100674T CY091100674T CY1109186T1 CY 1109186 T1 CY1109186 T1 CY 1109186T1 CY 20091100674 T CY20091100674 T CY 20091100674T CY 091100674 T CY091100674 T CY 091100674T CY 1109186 T1 CY1109186 T1 CY 1109186T1
Authority
CY
Cyprus
Prior art keywords
dota
dioxybytynyl
hexamethyl
composition
oxytripyrrolidinophosphium
Prior art date
Application number
CY20091100674T
Other languages
Greek (el)
Inventor
Mauro Marzi
Marzo Maria Di
Original Assignee
Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP06763428A external-priority patent/EP1899354B1/en
Application filed by Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. filed Critical Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.
Publication of CY1109186T1 publication Critical patent/CY1109186T1/en

Links

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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Περιγράφεται μια διαδιακασία για την σύνθεση της δεοξυβιοτυνίλης εξαμεθυλενοδιαμίνης-DOTA. Η εν λόγω διαδικασία περιλαμβάνει την αντίδραση της δεοξυβιοτυνίλης εξαμεθυλενοφιαμίνης με το τρι-τερτ-βουτυλ-DOTA στην παρουσία του benzotriazol-1-yl-oxytripyrrolidinophosphium hexafluorophosphate, ως παράγοντας συμπύκνωσης, και της τριαιθυλαμίνης ως βάση.A procedure for the synthesis of deoxybiotynil hexamethylenediamine-DOTA is described. This process involves the reaction of deoxybutynyl hexamethylenephiamine with tert-butyl-DOTA in the presence of benzotriazol-1-yl-oxytripyrrolidinophosphium hexafluorophosphate, as a condensing agent, and triethylamine.

CY20091100674T 2005-06-30 2009-06-29 COMPOSITION OF DIOXYBYTYNYL HEXAMETHYL-DOTA CY1109186T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMU20050345 2005-06-30
EP06763428A EP1899354B1 (en) 2005-06-30 2006-05-31 Synthesis of deoxybiotinyl hexamethylenediamine-dota

Publications (1)

Publication Number Publication Date
CY1109186T1 true CY1109186T1 (en) 2014-07-02

Family

ID=41694430

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20091100674T CY1109186T1 (en) 2005-06-30 2009-06-29 COMPOSITION OF DIOXYBYTYNYL HEXAMETHYL-DOTA

Country Status (3)

Country Link
CY (1) CY1109186T1 (en)
PT (1) PT1899354E (en)
RS (1) RS50816B (en)

Also Published As

Publication number Publication date
RS50816B (en) 2010-08-31
PT1899354E (en) 2009-06-04

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