CS268156B2 - Process for preparing 1,1-dioxydes of 6-aminoalkylpenicillanic acids - Google Patents
Process for preparing 1,1-dioxydes of 6-aminoalkylpenicillanic acids Download PDFInfo
- Publication number
- CS268156B2 CS268156B2 CS83122A CS12283A CS268156B2 CS 268156 B2 CS268156 B2 CS 268156B2 CS 83122 A CS83122 A CS 83122A CS 12283 A CS12283 A CS 12283A CS 268156 B2 CS268156 B2 CS 268156B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- group
- hydrogen
- compounds
- benzyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US33879782A | 1982-01-11 | 1982-01-11 | |
US38832482A | 1982-06-14 | 1982-06-14 | |
US06/434,371 US4452796A (en) | 1982-06-14 | 1982-10-21 | 6-Aminoalkylpenicillanic acid 1,1-dioxides as beta-lactamase inhibitors |
Publications (2)
Publication Number | Publication Date |
---|---|
CS12283A2 CS12283A2 (en) | 1988-08-16 |
CS268156B2 true CS268156B2 (en) | 1990-03-14 |
Family
ID=27407295
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS83122A CS268156B2 (en) | 1982-01-11 | 1983-01-07 | Process for preparing 1,1-dioxydes of 6-aminoalkylpenicillanic acids |
Country Status (3)
Country | Link |
---|---|
KR (1) | KR860001278B1 (ko) |
CS (1) | CS268156B2 (ko) |
SU (1) | SU1170972A3 (ko) |
-
1983
- 1983-01-07 CS CS83122A patent/CS268156B2/cs unknown
- 1983-01-10 KR KR1019830000068A patent/KR860001278B1/ko not_active IP Right Cessation
- 1983-01-10 SU SU833534105A patent/SU1170972A3/ru active
Also Published As
Publication number | Publication date |
---|---|
KR860001278B1 (ko) | 1986-09-05 |
KR840003256A (ko) | 1984-08-20 |
CS12283A2 (en) | 1988-08-16 |
SU1170972A3 (ru) | 1985-07-30 |
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