CS233746B2 - Processing of amidazolin derivatives - Google Patents

Processing of amidazolin derivatives Download PDF

Info

Publication number
CS233746B2
CS233746B2 CS832172A CS217283A CS233746B2 CS 233746 B2 CS233746 B2 CS 233746B2 CS 832172 A CS832172 A CS 832172A CS 217283 A CS217283 A CS 217283A CS 233746 B2 CS233746 B2 CS 233746B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
compound
sub
alcohol
adrenoreceptor
Prior art date
Application number
CS832172A
Other languages
Czech (cs)
English (en)
Inventor
Michael R Stillings
Original Assignee
Reckitt & Colmann Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reckitt & Colmann Prod Ltd filed Critical Reckitt & Colmann Prod Ltd
Publication of CS233746B2 publication Critical patent/CS233746B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, ***e
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/12—1,4-Dioxanes; Hydrogenated 1,4-dioxanes not condensed with other rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Lock And Its Accessories (AREA)
  • Vehicle Interior And Exterior Ornaments, Soundproofing, And Insulation (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Paper (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Photoreceptors In Electrophotography (AREA)
CS832172A 1982-04-17 1983-03-29 Processing of amidazolin derivatives CS233746B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8211205 1982-04-17

Publications (1)

Publication Number Publication Date
CS233746B2 true CS233746B2 (en) 1985-03-14

Family

ID=10529762

Family Applications (1)

Application Number Title Priority Date Filing Date
CS832172A CS233746B2 (en) 1982-04-17 1983-03-29 Processing of amidazolin derivatives

Country Status (24)

Country Link
US (1) US4446148A (fi)
EP (1) EP0092328B1 (fi)
JP (1) JPS58192882A (fi)
AT (1) ATE27275T1 (fi)
AU (1) AU552397B2 (fi)
CA (1) CA1190932A (fi)
CS (1) CS233746B2 (fi)
DD (1) DD209628A5 (fi)
DE (1) DE3371631D1 (fi)
DK (1) DK160093C (fi)
ES (1) ES8405394A1 (fi)
FI (1) FI73676C (fi)
GB (1) GB2118548B (fi)
GR (1) GR78528B (fi)
HU (1) HU190894B (fi)
IE (1) IE54922B1 (fi)
IL (1) IL68318A (fi)
NO (1) NO158019C (fi)
NZ (1) NZ203680A (fi)
PL (1) PL143658B1 (fi)
PT (1) PT76558B (fi)
SU (1) SU1217257A3 (fi)
ZA (1) ZA832278B (fi)
ZW (1) ZW8783A1 (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4882343A (en) * 1987-08-28 1989-11-21 G. D. Searle & Co. Biarylalkylimidazole derivatives as anti-depressants
AU6307690A (en) * 1989-09-27 1991-04-11 Rhone-Poulenc Sante Imidazoles
FR2698789B1 (fr) * 1992-12-07 1995-03-03 Pf Medicament Utilisation de l'idazoxan et ses dérivés pour la préparation d'un médicament destiné au traitement de la maladie de Parkinson et de son évolution.
FR2700113B1 (fr) * 1993-01-07 1995-03-24 Pf Medicament Utilisation de l'Idazoxan et ses dérivés pour la fabrication de médicaments destinés au traitement des maladies neurodégénératives et en particulier l'évolution de la maladie d'Alzheimer.
US6162455A (en) * 1997-01-22 2000-12-19 American Cyanamid Company Method for increasing lean meat, improving the lean meat to fat ratio and improving amino acid utilization in warm-blooded animals
FR2766824B1 (fr) * 1997-07-30 1999-09-10 Adir Nouveaux composes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2795727B1 (fr) * 1999-06-29 2001-09-21 Pf Medicament Nouveaux derives benzodioxanne imidazolines fluores, leur preparation et leurs applications en therapeutique

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2979511A (en) * 1959-03-25 1961-04-11 Olin Mathieson Certain 1, 4-benzodioxanyl imidazolines and corresponding pyrimidines and process
PH16249A (en) * 1980-02-04 1983-08-16 Reckitt & Colmann Prod Ltd Imidazoline derivatives,its pharmaceutical composition and method of use
NZ199469A (en) * 1981-01-30 1984-03-16 Reckitt & Colmann Prod Ltd Benzodioxanyl-2-imidazoline derivatives and pharmaceutical compositions

Also Published As

Publication number Publication date
FI73676C (fi) 1987-11-09
NO158019B (no) 1988-03-21
GR78528B (fi) 1984-09-27
ZW8783A1 (en) 1983-07-06
ES521440A0 (es) 1984-06-01
NZ203680A (en) 1985-08-16
DE3371631D1 (de) 1987-06-25
IL68318A (en) 1986-07-31
US4446148A (en) 1984-05-01
DK160093B (da) 1991-01-28
EP0092328A2 (en) 1983-10-26
EP0092328A3 (en) 1985-05-08
AU552397B2 (en) 1986-05-29
FI73676B (fi) 1987-07-31
NO158019C (no) 1988-06-29
PL241515A1 (en) 1984-07-30
ZA832278B (en) 1983-12-28
GB2118548B (en) 1985-07-31
IE830858L (en) 1983-10-17
FI831199L (fi) 1983-10-18
EP0092328B1 (en) 1987-05-20
DD209628A5 (de) 1984-05-16
IE54922B1 (en) 1990-03-28
JPS58192882A (ja) 1983-11-10
DK160093C (da) 1991-06-24
DK163783D0 (da) 1983-04-14
HU190894B (en) 1986-12-28
CA1190932A (en) 1985-07-23
IL68318A0 (en) 1983-07-31
NO831318L (no) 1983-10-18
SU1217257A3 (ru) 1986-03-07
JPH0427984B2 (fi) 1992-05-13
PT76558A (en) 1983-05-01
PT76558B (en) 1986-01-21
PL143658B1 (en) 1988-03-31
ES8405394A1 (es) 1984-06-01
AU1329883A (en) 1983-10-20
GB2118548A (en) 1983-11-02
FI831199A0 (fi) 1983-04-11
DK163783A (da) 1983-10-18
ATE27275T1 (de) 1987-06-15

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