CO7071139A2 - Tratamiento contra el cáncer cerebral - Google Patents

Tratamiento contra el cáncer cerebral

Info

Publication number
CO7071139A2
CO7071139A2 CO14208829A CO14208829A CO7071139A2 CO 7071139 A2 CO7071139 A2 CO 7071139A2 CO 14208829 A CO14208829 A CO 14208829A CO 14208829 A CO14208829 A CO 14208829A CO 7071139 A2 CO7071139 A2 CO 7071139A2
Authority
CO
Colombia
Prior art keywords
brain cancer
cancer treatment
compounds
treatment against
against brain
Prior art date
Application number
CO14208829A
Other languages
English (en)
Inventor
Patrice A Lee
Shannon L Winski
Kevin Koch
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48048296&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO7071139(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of CO7071139A2 publication Critical patent/CO7071139A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K39/395Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Abstract

Se proporcionan en la presente compuestos para el tratamiento contra el cáncer cerebral. Además, se proporcionan en la presente composiciones farmacéuticas que integran esos compuestos para el tratamiento contra el cáncer cerebral.
CO14208829A 2012-03-23 2014-09-19 Tratamiento contra el cáncer cerebral CO7071139A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261615082P 2012-03-23 2012-03-23

Publications (1)

Publication Number Publication Date
CO7071139A2 true CO7071139A2 (es) 2014-09-30

Family

ID=48048296

Family Applications (1)

Application Number Title Priority Date Filing Date
CO14208829A CO7071139A2 (es) 2012-03-23 2014-09-19 Tratamiento contra el cáncer cerebral

Country Status (30)

Country Link
US (3) US20150110780A1 (es)
EP (4) EP3400943B1 (es)
JP (6) JP2015514075A (es)
KR (3) KR102317166B1 (es)
CN (2) CN104203279B (es)
AU (4) AU2013234921A1 (es)
CA (1) CA2867723C (es)
CL (1) CL2014002497A1 (es)
CO (1) CO7071139A2 (es)
CY (2) CY1120204T1 (es)
DK (2) DK2827900T3 (es)
ES (2) ES2855142T3 (es)
HK (1) HK1206276A1 (es)
HR (1) HRP20180659T1 (es)
HU (2) HUE053156T2 (es)
IL (3) IL234627B (es)
LT (1) LT2827900T (es)
MX (1) MX354024B (es)
MY (2) MY174883A (es)
NZ (4) NZ756264A (es)
PH (1) PH12014502032A1 (es)
PL (2) PL3400943T3 (es)
PT (2) PT3400943T (es)
RS (1) RS57140B1 (es)
RU (2) RU2672575C2 (es)
SG (1) SG11201405954YA (es)
SI (2) SI2827900T1 (es)
TR (1) TR201808450T4 (es)
UA (1) UA122044C2 (es)
WO (1) WO2013142875A1 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE035247T2 (hu) 2011-10-14 2018-05-02 Array Biopharma Inc Szilárd diszperzió
EP2766363A1 (en) 2011-10-14 2014-08-20 Array Biopharma, Inc. Polymorphs of arry-380, a selective herb2 inhibitor and pharmaceutical compositions containing them
ES2855142T3 (es) 2012-03-23 2021-09-23 Array Biopharma Inc Compuestos para la utilización en el tratamiento de las metástasis cerebrales en un paciente con cáncer de mama ErbB2+
CA3055957A1 (en) * 2017-03-09 2018-09-13 The Board Of Trustees Of The Leland Stanford Junior University Treatment of pediatric brain tumors with targeting of cd47 pathway
EP3615067A1 (en) 2017-04-28 2020-03-04 Seattle Genetics, Inc. Treatment of her2 positive cancers
WO2019197973A1 (en) * 2018-04-09 2019-10-17 Moshe Giladi Treating tumors with ttfields and an aurora kinase inhibitor
CN109942576B (zh) * 2019-03-07 2020-09-11 上海工程技术大学 Irbinitinib及中间体的制备方法
CN111825604A (zh) * 2019-04-16 2020-10-27 宁波药腾医药科技有限公司 一种图卡替尼及其中间产物的合成方法
MX2022001863A (es) 2019-08-12 2022-05-30 Deciphera Pharmaceuticals Llc Metodos para tratar los tumores del estroma gastrointestinal.
AU2020417282B2 (en) 2019-12-30 2023-08-31 Deciphera Pharmaceuticals, Llc Compositions of 1-(4-bromo-5-(1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl)-2-fluorophenyl)-3-phenylurea
PL4084778T3 (pl) 2019-12-30 2024-03-04 Deciphera Pharmaceuticals, Llc Formulacje amorficznych inhibitorów kinazy i sposoby ich zastosowania

Family Cites Families (14)

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Publication number Priority date Publication date Assignee Title
CH690163A5 (fr) * 1995-07-28 2000-05-31 Symphar Sa Dérivés gem-diphosphonates substitués utiles en tant qu'agents anti-cancers.
US6350786B1 (en) * 1998-09-22 2002-02-26 Hoffmann-La Roche Inc. Stable complexes of poorly soluble compounds in ionic polymers
RU2255765C2 (ru) * 2000-01-21 2005-07-10 Чилдренз Хоспитал Лос-Анджелес Способ ингибирования роста опухолей головного мозга с помощью отобранных антагонистов интегринов
US20020137731A1 (en) 2000-05-30 2002-09-26 Gewirtz David A. Combination of radiation and vitamin D3 analogs for the treatment of cancer
CN103772373B (zh) 2003-08-14 2017-06-09 阿雷生物药品公司 作为受体酪氨酸激酶抑制剂的喹唑啉类似物
BRPI0511754A (pt) 2004-06-03 2008-01-02 Smithkline Beechman Cork Ltd uso de um composto ou sais ou solvatos do mesmo
CN1989112A (zh) * 2004-06-03 2007-06-27 史密丝克莱恩比彻姆(科克)有限公司 癌症治疗方法
BR122018075851B1 (pt) 2005-11-15 2022-01-11 Array Biopharma Inc Compostos relacionados ao tratamento de doença hiperproliferativa e processos para preparar compostos
JP5068270B2 (ja) 2006-01-31 2012-11-07 ノバルティス アーゲー 癌を処置するためのil−17アンタゴニスト抗体
JP2010540460A (ja) * 2007-09-24 2010-12-24 トラガラ ファーマシューティカルズ,インク. COX‐2阻害薬と抗HER2[ErbB2]抗体の混合物又はCOX‐2阻害薬とHER2[ErbB2]受容体チロシンキナーゼ阻害薬の混合物を用いた癌の治療
EP3692988A3 (en) 2008-03-18 2020-10-14 Genentech, Inc. Combinations of an anti-her2 antibody-drug conjugate and 5-fu, anti-vegf antibody, carboplatin or abt-869 and methods of use
EP2766363A1 (en) 2011-10-14 2014-08-20 Array Biopharma, Inc. Polymorphs of arry-380, a selective herb2 inhibitor and pharmaceutical compositions containing them
HUE035247T2 (hu) 2011-10-14 2018-05-02 Array Biopharma Inc Szilárd diszperzió
ES2855142T3 (es) 2012-03-23 2021-09-23 Array Biopharma Inc Compuestos para la utilización en el tratamiento de las metástasis cerebrales en un paciente con cáncer de mama ErbB2+

Also Published As

Publication number Publication date
ES2673165T3 (es) 2018-06-20
DK2827900T3 (en) 2018-05-07
IL261659A (en) 2018-10-31
KR102490961B1 (ko) 2023-01-19
MY174883A (en) 2020-05-20
HK1206276A1 (en) 2016-01-08
PT2827900T (pt) 2018-06-14
PL2827900T3 (pl) 2018-08-31
NZ630843A (en) 2017-01-27
NZ756264A (en) 2022-09-30
JP2017141302A (ja) 2017-08-17
DK3400943T3 (da) 2021-02-08
WO2013142875A1 (en) 2013-09-26
IL269205B (en) 2020-06-30
HUE053156T2 (hu) 2021-06-28
CA2867723C (en) 2022-11-08
EP4252855A3 (en) 2023-11-15
KR20140139009A (ko) 2014-12-04
EP2827900A1 (en) 2015-01-28
JP2015514075A (ja) 2015-05-18
JP2024019526A (ja) 2024-02-09
IL234627B (en) 2018-10-31
TR201808450T4 (tr) 2018-07-23
PT3400943T (pt) 2021-02-02
JP2019081792A (ja) 2019-05-30
PH12014502032A1 (en) 2014-11-24
HUE037966T2 (hu) 2018-09-28
JP2022190126A (ja) 2022-12-22
KR102317166B1 (ko) 2021-10-26
JP2021178820A (ja) 2021-11-18
KR20210131426A (ko) 2021-11-02
RU2014142700A (ru) 2016-05-20
EP4252855A2 (en) 2023-10-04
AU2021261849A1 (en) 2021-12-02
SI3400943T1 (sl) 2021-03-31
JP7404485B2 (ja) 2023-12-25
CY1120204T1 (el) 2018-12-12
RU2018138976A3 (es) 2022-04-08
LT2827900T (lt) 2018-05-10
PL3400943T3 (pl) 2021-06-14
CA2867723A1 (en) 2013-09-26
EP3400943A1 (en) 2018-11-14
SG11201405954YA (en) 2014-10-30
CN104203279A (zh) 2014-12-10
MX354024B (es) 2018-02-08
CN109223791A (zh) 2019-01-18
CL2014002497A1 (es) 2014-11-14
AU2017272232A1 (en) 2018-01-04
US20230190749A1 (en) 2023-06-22
KR20200115656A (ko) 2020-10-07
KR102160462B1 (ko) 2020-09-28
UA122044C2 (uk) 2020-09-10
NZ741615A (en) 2019-10-25
US20150110780A1 (en) 2015-04-23
CY1123837T1 (el) 2022-05-27
MY202114A (en) 2024-04-04
AU2013234921A1 (en) 2014-10-02
RU2018138976A (ru) 2018-12-06
ES2855142T3 (es) 2021-09-23
AU2017272232C1 (en) 2019-08-15
EP3842044A1 (en) 2021-06-30
US20190255051A1 (en) 2019-08-22
HRP20180659T1 (hr) 2018-06-01
AU2017272232B2 (en) 2019-02-28
US11504370B2 (en) 2022-11-22
EP3400943B1 (en) 2020-12-02
AU2019203618B2 (en) 2021-08-05
RS57140B1 (sr) 2018-07-31
MX2014011437A (es) 2014-11-10
NZ724544A (en) 2018-05-25
AU2019203618A1 (en) 2019-06-13
EP2827900B1 (en) 2018-03-21
JP6898960B2 (ja) 2021-07-07
CN104203279B (zh) 2018-10-30
IL269205A (en) 2019-11-28
RU2672575C2 (ru) 2018-11-16
SI2827900T1 (en) 2018-06-29

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