CO6900144A2 - Compuestos de triazolopiridina como inhibidores de la ped10a - Google Patents

Compuestos de triazolopiridina como inhibidores de la ped10a

Info

Publication number: CO6900144A2
Authority: CO; Colombia
Prior art keywords: ped10a; inhibitors; triazolopyridine compounds; triazolopyridine; compounds
Prior art date: 2011-09-19

Application number

CO14047250A

Other languages

English (en)

Inventor

Alexander Flohr

Zbinden Katrin Groebke

Matthias Koerner

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-09-19

Filing date

2014-03-05

Publication date

2014-03-20

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46851999&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6900144(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2014-03-05 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2014-03-20 Publication of CO6900144A2 publication Critical patent/CO6900144A2/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

CO14047250A 2011-09-19 2014-03-05 Compuestos de triazolopiridina como inhibidores de la ped10a CO6900144A2 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP11181752		2011-09-19

Publications (1)

Publication Number	Publication Date
CO6900144A2 true CO6900144A2 (es)	2014-03-20

Family

ID=46851999

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CO14047250A CO6900144A2 (es)	2011-09-19	2014-03-05	Compuestos de triazolopiridina como inhibidores de la ped10a

Country Status (18)

Country	Link
US (2)	US8946427B2 (es)
EP (1)	EP2758396B1 (es)
JP (1)	JP2014526533A (es)
KR (1)	KR101584925B1 (es)
CN (1)	CN103827114B (es)
AU (1)	AU2012311713A1 (es)
BR (1)	BR112014006248A2 (es)
CA (1)	CA2846758C (es)
CL (1)	CL2014000641A1 (es)
CO (1)	CO6900144A2 (es)
EA (1)	EA201490599A1 (es)
ES (1)	ES2626801T3 (es)
IL (1)	IL231403A0 (es)
MX (1)	MX2014003025A (es)
PE (1)	PE20141553A1 (es)
SG (1)	SG11201400759RA (es)
UA (1)	UA108711C2 (es)
WO (1)	WO2013041472A1 (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2013043518A1 (en)	2011-09-22	2013-03-28	Merck Sharp & Dohme Corp.	Imidazopyridyl compounds as aldosterone synthase inhibitors
WO2013043520A1 (en)	2011-09-22	2013-03-28	Merck Sharp & Dohme Corp.	Triazolopyridyl compounds as aldosterone synthase inhibitors
DK2991984T3 (en) *	2013-04-30	2017-05-08	Hoffmann La Roche	PALLADIUM-CATALYST COUPLING OF PYRAZOLAMIDES
TWI652014B (zh)	2013-09-13	2019-03-01	美商艾佛艾姆希公司	雜環取代之雙環唑殺蟲劑
KR20170032329A (ko) *	2014-07-30	2017-03-22	모찌다 세이야쿠 가부시끼가이샤	피라졸 유도체의 제조 방법
KR20170032328A (ko) *	2014-07-30	2017-03-22	모찌다 세이야쿠 가부시끼가이샤	피라졸 유도체의 제조 방법
CN112608300B (zh)	2015-03-11	2024-04-26	Fmc公司	杂环取代的二环唑杀有害生物剂
KR102536024B1 (ko)	2015-03-12	2023-05-24	에프엠씨 코포레이션	헤테로환-치환 이환 아졸 살충제
WO2017062729A1 (en)	2015-10-08	2017-04-13	E. I. Du Pont De Nemours And Company	Heterocycle-substituted bicyclic azole pesticides
ES2932627T3 (es) *	2017-08-22	2023-01-23	Bayer Ag	Derivados heterocíclicos como pesticidas
BR112021023409A2 (pt)	2019-05-27	2022-01-04	Nihon Nohyaku Co Ltd	Composto heterocíclico condensado tendo um átomo de nitrogênio em cabeça de ponte ou sal do mesmo, inseticida agrícola ou hortícola compreendendo o composto e método para usar o inseticida
AR119140A1 (es)	2019-06-13	2021-11-24	Pi Industries Ltd	Compuestos heterocíclicos fusionados y su uso como agentes de control de plagas
CN110396157B (zh) *	2019-08-07	2021-07-30	广州市建筑科学研究院有限公司	缓释型聚羧酸纳米减水剂及其制备方法和应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6355653B1 (en) *	1999-09-06	2002-03-12	Hoffmann-La Roche Inc.	Amino-triazolopyridine derivatives
CA2534432A1 (en)	2003-07-31	2005-02-10	Bayer Pharmaceuticals Corporation	Methods for treating diabetes and related disorders using pde10a inhibitors
NL2000397C2 (nl) *	2006-01-05	2007-10-30	Pfizer Prod Inc	Bicyclische heteroarylverbindingen als PDE10 inhibitoren.
JPWO2010035745A1 (ja) *	2008-09-25	2012-02-23	杏林製薬株式会社	ヘテロ環ビアリール誘導体及びそれらを有効成分とするｐｄｅ阻害剤
WO2010059836A1 (en) *	2008-11-20	2010-05-27	Decode Genetics Ehf	Substituted aza-bridged bicyclics for cardiovascular and cns disease
US8685967B2 (en) *	2009-04-07	2014-04-01	Merck Sharp & Dohme Corp.	Substituted triazolopyridines and analogs thereof
JP5629322B2 (ja) *	2009-09-24	2014-11-19	エフ．ホフマン−ラロシュアーゲーＦ．Ｈｏｆｆｍａｎｎ−ＬａＲｏｃｈｅＡｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ	ホスホジエステラーゼ１０ａ阻害剤としてのイミダゾピリジンまたはイミダゾピリミジン誘導体
RU2542586C2 (ru)	2009-11-24	2015-02-20	Нокиа Корпорейшн	Устройство для обработки звуковых сигналов
TW201200516A (en) *	2009-12-17	2012-01-01	Lundbeck & Co As H	Phenylimidazole derivatives comprising an ethynylene linker as PDE10A enzyme inhibitors
TWI487705B (zh) *	2009-12-17	2015-06-11	Lundbeck & Co As H	作為ｐｄｅ１０ａ酵素抑制劑之雜芳香族芳基***衍生物
TWI485151B (zh) *	2009-12-17	2015-05-21	Lundbeck & Co As H	作為ｐｄｅ１０ａ酵素抑制劑之雜芳香族苯基咪唑衍生物

2012
- 2012-09-17 AU AU2012311713A patent/AU2012311713A1/en not_active Abandoned
- 2012-09-17 EA EA201490599A patent/EA201490599A1/ru unknown
- 2012-09-17 EP EP12759445.5A patent/EP2758396B1/en not_active Not-in-force
- 2012-09-17 ES ES12759445.5T patent/ES2626801T3/es active Active
- 2012-09-17 SG SG11201400759RA patent/SG11201400759RA/en unknown
- 2012-09-17 JP JP2014531187A patent/JP2014526533A/ja active Pending
- 2012-09-17 WO PCT/EP2012/068203 patent/WO2013041472A1/en active Application Filing
- 2012-09-17 CA CA2846758A patent/CA2846758C/en not_active Expired - Fee Related
- 2012-09-17 UA UAA201404029A patent/UA108711C2/uk unknown
- 2012-09-17 BR BR112014006248A patent/BR112014006248A2/pt not_active IP Right Cessation
- 2012-09-17 PE PE2014000366A patent/PE20141553A1/es not_active Application Discontinuation
- 2012-09-17 MX MX2014003025A patent/MX2014003025A/es active IP Right Grant
- 2012-09-17 KR KR1020147009588A patent/KR101584925B1/ko not_active IP Right Cessation
- 2012-09-17 CN CN201280045398.XA patent/CN103827114B/zh not_active Expired - Fee Related
2014
- 2014-03-05 CO CO14047250A patent/CO6900144A2/es unknown
- 2014-03-06 IL IL231403A patent/IL231403A0/en unknown
- 2014-03-17 CL CL2014000641A patent/CL2014000641A1/es unknown
- 2014-03-18 US US14/218,275 patent/US8946427B2/en not_active Expired - Fee Related
- 2014-12-16 US US14/572,312 patent/US9227970B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
CN103827114A (zh)	2014-05-28
EP2758396A1 (en)	2014-07-30
US8946427B2 (en)	2015-02-03
JP2014526533A (ja)	2014-10-06
US20140303141A1 (en)	2014-10-09
UA108711C2 (uk)	2015-05-25
ES2626801T3 (es)	2017-07-26
KR20140075716A (ko)	2014-06-19
CA2846758A1 (en)	2013-03-28
AU2012311713A1 (en)	2014-03-13
CA2846758C (en)	2017-09-12
CL2014000641A1 (es)	2014-11-14
NZ621597A (en)	2015-04-24
SG11201400759RA (en)	2014-07-30
US9227970B2 (en)	2016-01-05
PE20141553A1 (es)	2014-10-30
EA201490599A1 (ru)	2014-07-30
MX2014003025A (es)	2014-05-28
BR112014006248A2 (pt)	2017-04-11
IL231403A0 (en)	2014-04-30
KR101584925B1 (ko)	2016-01-12
CN103827114B (zh)	2016-08-24
EP2758396B1 (en)	2017-03-29
US20150099735A1 (en)	2015-04-09
WO2013041472A1 (en)	2013-03-28

Publication	Publication Date	Title
CO6920291A2 (es)	2014-04-10	3-pirmidin-4-il-oxazolidin-2-onas como inhibidores de la idhmutante
CO6801747A2 (es)	2013-11-29	Derivados de pirrolotriazinona como inhibidores de pi3k
CO6900145A2 (es)	2014-03-20	Compuesto de ciclopropanoamina
CO6930358A2 (es)	2014-04-28	Compuestos inhibidores de metaloenzimas
CO6910199A2 (es)	2014-03-31	Heterociclilaminas como inhibidores de pi3k
CO6900144A2 (es)	2014-03-20	Compuestos de triazolopiridina como inhibidores de la ped10a
CO6920292A2 (es)	2014-04-10	Compuesto de quinolona
CO6980657A2 (es)	2014-06-27	Triazolopiridinas sustituidas
CO6880068A2 (es)	2014-02-28	Aminoquinazolinas como inhibidores de quinasa
CO6880065A2 (es)	2014-02-28	Nuevos compuestos de 4-piperidinilo para uso como inhibidores de la tankirasa
BR112013022102A2 (pt)	2018-06-26	composição
BR112013015449A2 (pt)	2016-09-20	compostos de bi-heteroarila como inibidores de vps23
BR112014012016A2 (pt)	2017-05-16	compostos
BR112013029474A2 (pt)	2017-01-17	ferramenta multi-abrasiva
SMT201600328B (it)	2016-11-10	Nuovi composti come inibitori di diacilglicerolo aciltransferasi
DK2678329T3 (da)	2016-02-22	Triazolopyridinforbindelser som pim-kinase-hæmmere
CU24164B1 (es)	2016-03-31	Inhibidores sustituidos de acetil-coa carboxilasa
BR112014011686A2 (pt)	2017-07-11	ferramenta de tração
CO6801751A2 (es)	2013-11-29	Triazolopiridinas
CO6910197A2 (es)	2014-03-31	Compuestos novedosos
CO6862145A2 (es)	2014-02-10	Imidazopiridazinas como inhibidores de quinasa akt
BR112013013912A2 (pt)	2016-09-13	compostos de triazolopiridina
BR112013028029A2 (pt)	2017-08-08	composto
CO6960557A2 (es)	2014-05-30	Derivados de 2-yodo-imidazol
CO7020914A2 (es)	2014-08-11	Nievos derivados de morofolinilo útiles como inhibidores de mogat-2