CO6470821A2 - Pirazinilpirazoles - Google Patents

Pirazinilpirazoles

Info

Publication number
CO6470821A2
CO6470821A2 CO11161605A CO11161605A CO6470821A2 CO 6470821 A2 CO6470821 A2 CO 6470821A2 CO 11161605 A CO11161605 A CO 11161605A CO 11161605 A CO11161605 A CO 11161605A CO 6470821 A2 CO6470821 A2 CO 6470821A2
Authority
CO
Colombia
Prior art keywords
pirazinilpirazoles
ylpyrazoles
pyrazinylpyrazoles
parasiticides
pyrazin
Prior art date
Application number
CO11161605A
Other languages
English (en)
Inventor
Hans-Georg Schwarz
Jens Frackenpohl
Achim Hense
Simon Maechling
Stefan Schnatterer
Robert Velten
Stefan Werner
Angela Becker
Olga Malsam
Eva-Maria Franken
Arnd Voerste
Ulrich Gorgens
Peter Lummen
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of CO6470821A2 publication Critical patent/CO6470821A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

Procedimiento para la preparación de Pirazinilpirazoles de fórmula general (I) y composiciones que comprenden dichos pirazin-2-ilpirazoles. Proporcionar insecticidas y/o parasiticidas alternativos que muestren una acción mejorada o un espectro más amplio de actividad en comparación con los ingredientes activos conocidos de la técnica anterior.
CO11161605A 2009-05-29 2011-11-24 Pirazinilpirazoles CO6470821A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09161568A EP2266973A1 (de) 2009-05-29 2009-05-29 Pyrazinylpyrazole

Publications (1)

Publication Number Publication Date
CO6470821A2 true CO6470821A2 (es) 2012-06-29

Family

ID=40897591

Family Applications (1)

Application Number Title Priority Date Filing Date
CO11161605A CO6470821A2 (es) 2009-05-29 2011-11-24 Pirazinilpirazoles

Country Status (21)

Country Link
US (2) US20120190687A1 (es)
EP (2) EP2266973A1 (es)
KR (1) KR101758935B1 (es)
CN (1) CN102459235B (es)
AR (1) AR076798A1 (es)
AU (1) AU2010252346B2 (es)
BR (1) BRPI1012771A2 (es)
CA (1) CA2763498A1 (es)
CO (1) CO6470821A2 (es)
DO (1) DOP2011000366A (es)
EC (1) ECSP11011487A (es)
ES (1) ES2409891T3 (es)
IL (1) IL216337A (es)
MX (1) MX2011012504A (es)
NI (1) NI201100208A (es)
NZ (1) NZ596681A (es)
PE (1) PE20120320A1 (es)
TW (1) TW201107310A (es)
UY (1) UY32659A (es)
WO (1) WO2010136145A1 (es)
ZA (1) ZA201108637B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102574833B (zh) * 2009-10-12 2014-08-20 拜尔农作物科学股份公司 用作杀虫剂的酰胺和硫代酰胺
WO2011045224A1 (de) 2009-10-12 2011-04-21 Bayer Cropscience Ag 1- (pyrid-3-yl) -pyrazole und 1- (pyrimid-5-yl) -pyrazole als schädlingsbekämpfungsmittel
WO2011057984A1 (de) 2009-11-11 2011-05-19 Bayer Cropscience Ag Neue diazinyl-pyrazolylverbindungen
AU2011273694A1 (en) 2010-06-28 2013-02-07 Bayer Intellectual Property Gmbh Heteroaryl-substituted pyridine compounds for use as pesticides
DE102010063691A1 (de) 2010-12-21 2012-06-21 Bayer Animal Health Gmbh Ektoparasitizide Wirkstoffkombinationen
BR112014012243A2 (pt) 2011-11-21 2017-05-30 Basf Se processo de preparação de compostos
MX2014013430A (es) 2012-05-04 2015-04-14 Basf Se Compuestos que contienen pirazol sustituido y su uso como plaguicidas.
CA2886895C (en) * 2012-10-02 2021-10-19 Bayer Cropscience Ag Heterocyclic compounds as pesticides
BR112015009751A2 (pt) * 2012-10-31 2017-07-11 Bayer Cropscience Ag novos compostos heterocíclicos como pesticidas
WO2016174049A1 (en) 2015-04-30 2016-11-03 Bayer Animal Health Gmbh Anti-parasitic combinations including halogen-substituted compounds
EP3312162B1 (en) 2015-06-18 2021-01-06 Nippon Soda Co., Ltd. 1-(2-(ethylsulfonyl)-phenyl)-4-(phenyl)-1h-pyrazole derivatives and related compounds as pesticides
BR112018011124A2 (pt) 2015-11-30 2018-11-21 Hokko Chemical Industry Co., Ltd. derivado de 1,2,3-triazol e inseticida e acaricida contendo o dito derivado como ingrediente ativo
KR102352912B1 (ko) 2015-12-16 2022-01-18 닛뽕소다 가부시키가이샤 아릴아졸 화합물 및 유해 생물 방제제
BR112019010341B1 (pt) 2016-12-19 2022-12-06 Nippon Soda Co., Ltd Composto, e, formulação para controle de organismos nocivos, formulação inseticida ou formulação acaricida, formulação para controle de ectoparasitas, e, formulação para controle de endoparasitas ou para expulsão de endoparasitas
CN110305115A (zh) * 2019-08-19 2019-10-08 南通大学 一种含1-(6-氯吡嗪-2-基)-3-甲氧基吡唑单元的吡唑肟衍生物的制备和应用
CN115943143A (zh) * 2020-04-29 2023-04-07 拜耳公司 1-吡嗪基吡唑基-3-氧基烷基酸和其衍生物及其用于控制不需要的植物生长的用途

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU38903A1 (es) 1959-07-03
FR2326421A1 (fr) 1975-09-30 1977-04-29 Ugine Kuhlmann Nouveaux trifluoromethyl-3-aryl-4 amino-5 pyrazoles et leur application comme bases diazotables pour la synthese de matieres colorantes
US4101540A (en) * 1975-09-30 1978-07-18 Produits Chimiques Ugine Kuhlmann 3-Trifluoromethyl-4-phenyl-pyrazolium azo dyestuffs
JPH08208620A (ja) 1995-02-03 1996-08-13 Takeda Chem Ind Ltd アミノピラゾール誘導体、その製造法および用途
DE19544799A1 (de) * 1995-12-01 1997-06-05 Bayer Ag Substituierte 5-Aminopyrazole
US6169086B1 (en) * 1997-01-27 2001-01-02 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives
EA002101B1 (ru) 1997-01-27 2001-12-24 Дайити Фармасьютикал Ко., Лтд. Производные пиразола
EP1064286A1 (en) 1998-06-10 2001-01-03 Boulder Scientific Company Synthesis of aryl boronic acids
WO2001007413A1 (en) * 1999-07-22 2001-02-01 3-Dimensional Pharmaceuticals, Inc. 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
US7514464B2 (en) 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
CA2620425A1 (en) 2005-08-31 2007-03-08 Bayer Healthcare Llc Anilinopyrazole derivatives useful for the treatment of diabetes
WO2007048733A1 (de) 2005-10-28 2007-05-03 Basf Se Verwendung von 5-amino-pyrazolen zur bekämpfung pflanzenpathogener schadpilze, neue 5-amino-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel
DE102007003036A1 (de) 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
WO2009156090A2 (de) * 2008-06-26 2009-12-30 Bayer Cropscience Aktiengesellschaft Insektizide schwefel-derivatisierte 1-azinylpyrazole
WO2011057984A1 (de) * 2009-11-11 2011-05-19 Bayer Cropscience Ag Neue diazinyl-pyrazolylverbindungen

Also Published As

Publication number Publication date
NZ596681A (en) 2015-09-25
MX2011012504A (es) 2011-12-12
EP2266973A1 (de) 2010-12-29
US20110021539A1 (en) 2011-01-27
IL216337A (en) 2015-09-24
IL216337A0 (en) 2012-01-31
UY32659A (es) 2010-12-31
NI201100208A (es) 2012-08-17
AU2010252346A1 (en) 2011-12-22
EP2435420B1 (de) 2013-04-03
US8513260B2 (en) 2013-08-20
TW201107310A (en) 2011-03-01
CN102459235B (zh) 2015-03-11
AR076798A1 (es) 2011-07-06
ES2409891T3 (es) 2013-06-28
WO2010136145A1 (de) 2010-12-02
ECSP11011487A (es) 2011-12-30
PE20120320A1 (es) 2012-03-30
CN102459235A (zh) 2012-05-16
US20120190687A1 (en) 2012-07-26
KR20120061779A (ko) 2012-06-13
BRPI1012771A2 (pt) 2016-03-29
DOP2011000366A (es) 2011-12-15
EP2435420A1 (de) 2012-04-04
ZA201108637B (en) 2013-01-30
CA2763498A1 (en) 2010-12-02
AU2010252346B2 (en) 2015-11-19
KR101758935B1 (ko) 2017-07-17

Similar Documents

Publication Publication Date Title
CO6470821A2 (es) Pirazinilpirazoles
CL2015001973A1 (es) (divisional de la sol. 1567-2013) combinaciones de principios activos que comprenden piridiletilbenzamidas y otros principios activos.
CO6460772A2 (es) Inhibidores de la replicación del virus de la inmunodeficiencia humana
CR20110458A (es) Compuestos de 3-arilquinazolin-4-ona para combatir plagas de invertebrados
UY31747A (es) Nuevas formulaciones, comprimidos que comprenden tales formulaciones, su uso y procedimiento para su preparacion
PA8660301A1 (es) Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricacion y utilizacion
CL2013000304A1 (es) Compuestos derivados de 2-arilamino-bencimidazoles inhibidores de prostaglandina e2 (mpges-1); composicion farmaceutica que los comprende; compuestos intermediarios; uso en el tratamiento de enfermedades inflamatorias y/o afecciones asociadas, en particular el dolor.
ECSP10010355A (es) Arilpirrolinas insecticidas
CL2012003573A1 (es) Combinaciones que comprenden un derivado de antranilamida y otro principio activo con propiedades insecticidas y acaricidas; composiciones agroquimicas que contienen; uso de dicha combinacion; procedimiento para combatir parasitos animales; y procedimiento para la preparacion de dicha composicion agroquimica.
UY31952A (es) 5-metilideno-1,3-tiazolidina-2,4-dionas sustituidas como inhibidores de quinasa pim
CL2008001302A1 (es) Compuestos derivados de tetramatos sustituidos con 3-(2-alcoxifenilo); su proceso de preparacion de los mismos; agente para combatir plagas animales y/o vegetacion indeseada; procedimiento para su preparacion; uso de dichos compuestos; composicion que comprende a dichos compuestos; y procedimiento para combatir vegetacion indeseada.
CO6341618A2 (es) 4-fenil-1h-pirazoles insecticidas
GT201000023A (es) Nuevos derivados de 6-trialzolopiridacina-sulfanil benzotiazol y bencimidazol, su procedimiento de preparacion, su aplicacion como medicamentos, composiciones farmaceuticas y nueva utilizacion principalmente como inhibidores de met.
HN2008001393A (es) Derivados de 1,2,4,5- tetrahidro -3h- benzazepinas, su procedimiento de preparacion y las composiciones farmaceuticas que las contienen
CO6710916A2 (es) Inhibidores de notum pectinacetilesterasa y métodos de su uso
CL2011000583A1 (es) Composicion plaguicida que comprende un derivado del ácido alfa-alcoxifenil-acetico y un compuesto neonicotenoide.
UY31788A (es) Formulación farmacéutica sólida con liberación retardada
CR10050A (es) Combinacion fungicida de productos activos
UY29980A1 (es) Nuevas combinaciones de productos activos, comprendiendo un derivado de oximéter y un bis-tiocarbamato, procedimientos de preparación y aplicaciones.
EA200602049A1 (ru) Пролекарства стероидов с андрогенным действием
MX2019012375A (es) Formulaciones del inhibidor del antigeno-1 asociado a la funcion de linfocitos (lfa-1).
AR066936A1 (es) 3 - (2r - tetrahidrofuril - metil) - 2 - tioxantina. composiciones farmaceuticas.
UY29640A1 (es) Amidas sustituidas con heteroarilo que comprenden un grupo enlazador saturado, y su uso como agentes farmacéuticos.
ECSP10010292A (es) Nuevos derivados de ácido 2-mercaptociclopentanocarboxílico, su procedimiento de preparación y las composiciones farmacéuticas que los contienen
CR20120286A (es) Nuevos derivados de azabiciclo[3.1.0]hex-2-ilo, su procedimiento de preparación y las composiciones farmacéuticas que los contienen

Legal Events

Date Code Title Description
FC Application refused