CN1919846A - 伏立康唑及其药用盐、中间体的一种新定向合成制备方法 - Google Patents
伏立康唑及其药用盐、中间体的一种新定向合成制备方法 Download PDFInfo
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- CN1919846A CN1919846A CNA2006101131068A CN200610113106A CN1919846A CN 1919846 A CN1919846 A CN 1919846A CN A2006101131068 A CNA2006101131068 A CN A2006101131068A CN 200610113106 A CN200610113106 A CN 200610113106A CN 1919846 A CN1919846 A CN 1919846A
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- voriconazole
- pyrimidine
- triazole
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Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
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CN 200610113106 CN1919846B (zh) | 2006-09-14 | 2006-09-14 | 伏立康唑及其药用盐、中间体的一种新定向合成制备方法 |
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CN 200610113106 CN1919846B (zh) | 2006-09-14 | 2006-09-14 | 伏立康唑及其药用盐、中间体的一种新定向合成制备方法 |
Publications (2)
Publication Number | Publication Date |
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CN1919846A true CN1919846A (zh) | 2007-02-28 |
CN1919846B CN1919846B (zh) | 2013-01-02 |
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CN 200610113106 Expired - Fee Related CN1919846B (zh) | 2006-09-14 | 2006-09-14 | 伏立康唑及其药用盐、中间体的一种新定向合成制备方法 |
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Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2452049A (en) * | 2007-08-21 | 2009-02-25 | Alpharma Aps | Process for the preparation of voriconazole |
WO2011110198A1 (en) | 2010-03-10 | 2011-09-15 | Synthron B.V. | A process for making voriconazole |
CN102898419A (zh) * | 2012-11-15 | 2013-01-30 | 南京海陵中药制药工艺技术研究有限公司 | 一种制备伏立康唑中间体ⅰ的方法 |
CN103788073A (zh) * | 2013-12-18 | 2014-05-14 | 北京华禧联合科技发展有限公司 | 一种制备伏立康唑关键中间体的新方法 |
WO2020169025A1 (zh) | 2019-02-19 | 2020-08-27 | 浙江华海立诚药业有限公司 | 伏立康唑及其中间体的制备方法 |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1026788C (zh) * | 1990-02-02 | 1994-11-30 | 美国辉瑞有限公司 | ***类抗真菌剂的制备方法 |
CN1195346A (zh) * | 1995-08-05 | 1998-10-07 | 辉瑞研究开发公司 | 通过有机金属化合物对酮及其中间体的加成合成***化合物 |
CN1261287A (zh) * | 1997-06-21 | 2000-07-26 | 辉瑞大药厂 | 含有伏利康唑的药物制剂 |
-
2006
- 2006-09-14 CN CN 200610113106 patent/CN1919846B/zh not_active Expired - Fee Related
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1026788C (zh) * | 1990-02-02 | 1994-11-30 | 美国辉瑞有限公司 | ***类抗真菌剂的制备方法 |
CN1195346A (zh) * | 1995-08-05 | 1998-10-07 | 辉瑞研究开发公司 | 通过有机金属化合物对酮及其中间体的加成合成***化合物 |
CN1261287A (zh) * | 1997-06-21 | 2000-07-26 | 辉瑞大药厂 | 含有伏利康唑的药物制剂 |
Non-Patent Citations (2)
Title |
---|
FU-YAO ZHANG ET. AL.: "Enantioselective addition of diethylzinc to aromatic aldehydes catalyzed by titanium-5,5",6,6",7,7",8,8"-octahydro-l,l"–bi-2-naphthol complex", 《TETRAHEDRON:ASYMMETRY》 * |
MAKI MORI ET. AL.: "Asymmetric Catalytic Alkylation of Aldehydes with Diethylzinc Using a Chiral Binaphthol-Titanium Complex", 《TETRAHEDRON LETTERS》 * |
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2452049A (en) * | 2007-08-21 | 2009-02-25 | Alpharma Aps | Process for the preparation of voriconazole |
WO2011110198A1 (en) | 2010-03-10 | 2011-09-15 | Synthron B.V. | A process for making voriconazole |
CN102898419A (zh) * | 2012-11-15 | 2013-01-30 | 南京海陵中药制药工艺技术研究有限公司 | 一种制备伏立康唑中间体ⅰ的方法 |
CN103788073A (zh) * | 2013-12-18 | 2014-05-14 | 北京华禧联合科技发展有限公司 | 一种制备伏立康唑关键中间体的新方法 |
CN103788073B (zh) * | 2013-12-18 | 2017-11-03 | 北京华禧联合科技发展有限公司 | 一种制备伏立康唑关键中间体的新方法 |
WO2020169025A1 (zh) | 2019-02-19 | 2020-08-27 | 浙江华海立诚药业有限公司 | 伏立康唑及其中间体的制备方法 |
Also Published As
Publication number | Publication date |
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CN1919846B (zh) | 2013-01-02 |
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C41 | Transfer of patent application or patent right or utility model | ||
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Effective date of registration: 20071109 Address after: Room B, building 20C1, building 1, science and Technology Exhibition Center, North Third Ring Road West, Haidian District, Beijing Applicant after: Dadao Longda (Beijing) Medical Technology Development Co.Ltd Address before: Room B, building 20C1, building 1, science and Technology Exhibition Center, North Third Ring Road West, Haidian District, Beijing Applicant before: Boerda Biotech Development Co., Ltd., Beijing |
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Effective date of registration: 20080125 Address after: No. 1 Jiangnan Road, Taizhou, Jiangsu Applicant after: Yangtze River Pharmaceutical Co., Ltd. Address before: Room B, building 20C1, building 1, science and Technology Exhibition Center, North Third Ring Road West, Haidian District, Beijing Applicant before: Dadao Longda (Beijing) Medical Technology Development Co.Ltd |
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Owner name: DDLD (BEIJING) PHARMACEUTICAL TECHNOLOGY CO., LTD. Free format text: FORMER OWNER: YANGTZE RIVER PHARMACEUTICAL CO., LTD. Effective date: 20101125 |
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Free format text: CORRECT: ADDRESS; FROM: 225321 NO.1, YANGTZE RIVER SOUTH ROAD, TAIZHOU CITY, JIANGSU PROVINCE TO: 100086 ROOM 20C1, TOWER B, BUILDING 1, BEIJING SCIENCE AND TECHNOLOGY EXHIBITION CENTER, NO.48, N. 3RD RING ROAD WEST, HAIDIAN DISTRICT, BEIJING |
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Effective date of registration: 20101125 Address after: 100086, 20C1, room 48, building B, building 1, Beijing science and Technology Exhibition Center, No. West Third Ring Road, Beijing, China Applicant after: DDLD (Beijing) Pharmaceutical Technology Co.,Ltd. Address before: 225321 Taizhou Jiangnan Road, No. 1, Jiangsu, China Applicant before: Yangtze River Pharmaceutical Co., Ltd. |
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