CN1331576A - 用于缓解疼痛的方法和经皮组合物 - Google Patents
用于缓解疼痛的方法和经皮组合物 Download PDFInfo
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- CN1331576A CN1331576A CN99810055A CN99810055A CN1331576A CN 1331576 A CN1331576 A CN 1331576A CN 99810055 A CN99810055 A CN 99810055A CN 99810055 A CN99810055 A CN 99810055A CN 1331576 A CN1331576 A CN 1331576A
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- A61K31/33—Heterocyclic compounds
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Biophysics (AREA)
- Molecular Biology (AREA)
- Neurosurgery (AREA)
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- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| US09/106,684 | 1998-06-29 | ||
| US09/106,684 US6290986B1 (en) | 1996-10-24 | 1998-06-29 | Method and composition for transdermal administration of pharmacologic agents |
| US12290399P | 1999-03-05 | 1999-03-05 | |
| US60/122,903 | 1999-03-05 |
Publications (1)
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| CN1331576A true CN1331576A (zh) | 2002-01-16 |
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| CN99810055A Pending CN1331576A (zh) | 1998-06-29 | 1999-06-29 | 用于缓解疼痛的方法和经皮组合物 |
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| JP (1) | JP2002519310A (es) |
| KR (1) | KR20010078754A (es) |
| CN (1) | CN1331576A (es) |
| AU (1) | AU4841599A (es) |
| BG (1) | BG105175A (es) |
| BR (1) | BR9912508A (es) |
| CA (1) | CA2335837A1 (es) |
| HR (1) | HRP20000905A2 (es) |
| HU (1) | HUP0102728A3 (es) |
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| IL (1) | IL140420A0 (es) |
| MX (1) | MXPA00012767A (es) |
| NO (1) | NO20006604L (es) |
| PL (1) | PL345216A1 (es) |
| SK (1) | SK20012000A3 (es) |
| TR (1) | TR200003801T2 (es) |
| WO (1) | WO2000000120A1 (es) |
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| US6572880B2 (en) * | 1996-10-24 | 2003-06-03 | Pharmaceutical Applications Associates Llc | Methods and transdermal compositions for pain relief |
| ATE289295T1 (de) | 1997-04-22 | 2005-03-15 | Euro Celtique Sa | Die verwendung von durch carbozyklische und heterozyklische reste substituierte semicarbazonen und thiosemicarbazonen als natriumkanalblocker |
| PT1459751E (pt) | 1999-07-01 | 2005-11-30 | Pharmacia & Upjohn Co Llc | (s,s)-reboxetina para tratar as enxaquecas |
| DK1459751T3 (da) * | 1999-07-01 | 2005-12-19 | Pharmacia & Upjohn Co Llc | (S,S)reboxetin til behandling af migrænehovedpine |
| AU1261501A (en) * | 1999-12-06 | 2001-06-18 | Stanley L. Gore | Compositions and methods for intranasal delivery of active agents to the brain |
| IN191512B (es) * | 2000-01-21 | 2003-12-06 | Panacea Biotech | |
| DE10032132A1 (de) * | 2000-07-01 | 2002-01-17 | Lohmann Therapie Syst Lts | Dermales Therapeutisches System enthaltend nichtsteroidale Antiphlogistika mit selektiver COX-2-Hemmung |
| DE10042412B4 (de) * | 2000-08-30 | 2005-12-22 | Lts Lohmann Therapie-Systeme Ag | Transdermales therapeutisches System zur Abgabe von Venlafaxin, und seine Verwendung |
| US20040001889A1 (en) | 2002-06-25 | 2004-01-01 | Guohua Chen | Short duration depot formulations |
| EP2959893A1 (en) | 2002-12-13 | 2015-12-30 | DURECT Corporation | Oral drug delivery system comprising high viscosity liquid carrier materials |
| JP2005154368A (ja) * | 2003-11-27 | 2005-06-16 | Teikoku Seiyaku Co Ltd | ジソピラミド含有神経因性疼痛の鎮痛剤 |
| JP4807721B2 (ja) * | 2004-01-29 | 2011-11-02 | 株式会社 メドレックス | 消炎鎮痛外用剤 |
| PL1809329T3 (pl) | 2004-09-17 | 2012-08-31 | Durect Corp | Kompozycja znieczulająca zawierająca saib o przedłużonym uwalnianiu do stosowania miejscowego |
| US20070027105A1 (en) | 2005-07-26 | 2007-02-01 | Alza Corporation | Peroxide removal from drug delivery vehicle |
| JP2007308403A (ja) * | 2006-05-17 | 2007-11-29 | Kenji Yoshida | 皮膚外用剤 |
| KR100880748B1 (ko) * | 2006-08-29 | 2009-02-02 | 정헌택 | 디메톡시커큐민을 함유하는 혈관재협착 방지용 조성물 |
| US8337883B2 (en) | 2006-11-03 | 2012-12-25 | Durect Corporation | Transdermal delivery systems |
| US9511016B2 (en) * | 2007-06-12 | 2016-12-06 | Epicentrx, Inc. | Topical composition for treating pain |
| WO2009088414A2 (en) | 2007-12-06 | 2009-07-16 | Durect Corporation | Oral pharmaceutical dosage forms |
| US20100260844A1 (en) | 2008-11-03 | 2010-10-14 | Scicinski Jan J | Oral pharmaceutical dosage forms |
| EP2428211A4 (en) * | 2009-05-07 | 2013-04-03 | Moon & J Inc | PHARMACEUTICAL COMPOSITION FOR THE PREVENTION OR TREATMENT OF NEURAL DAMAGE AND NEUROLOGICAL DISEASES |
| US8491927B2 (en) | 2009-12-02 | 2013-07-23 | Nimble Epitech, Llc | Pharmaceutical composition containing a hypomethylating agent and a histone deacetylase inhibitor |
| CA2905131A1 (en) | 2013-03-15 | 2014-09-18 | Durect Corporation | Compositions with a rheological modifier to reduce dissolution variability |
| AU2015217309A1 (en) * | 2014-02-11 | 2016-08-25 | Dr. Reddy's Laboratories Ltd. | Parenteral compositions of celecoxib |
| WO2020084548A1 (en) | 2018-10-26 | 2020-04-30 | Viramal Limited | Mucoadhesive gel composition |
| EP3659583B1 (en) | 2018-11-30 | 2023-06-07 | Viramal Limited | A method of preparing a gelling agent, the gelling agent obtained thereby, and the use of said gelling agent |
| KR20220140711A (ko) | 2020-01-13 | 2022-10-18 | 듀렉트 코퍼레이션 | 불순물이 감소된 지속 방출 약물 전달 시스템 및 관련 방법 |
| FR3108841B1 (fr) * | 2020-04-06 | 2023-11-03 | Algotherapeutix | Composition pharmaceutique topique sous forme de gel aqueux comprenant au moins de l’amitriptyline |
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| US4395420A (en) * | 1981-12-09 | 1983-07-26 | Bernstein Joel E | Method and composition for treating pruritis |
| SI9300468A (en) * | 1992-10-14 | 1994-06-30 | Hoffmann La Roche | Injectable composition for the sustained release of biologically active compounds |
| GB9315856D0 (en) * | 1993-07-30 | 1993-09-15 | Wellcome Found | Stabilized pharmaceutical |
| US5654337A (en) * | 1995-03-24 | 1997-08-05 | II William Scott Snyder | Topical formulation for local delivery of a pharmaceutically active agent |
| US5837289A (en) * | 1996-07-23 | 1998-11-17 | Grasela; John C. | Transdermal delivery of medications using a combination of penetration enhancers |
| US5885597A (en) * | 1997-10-01 | 1999-03-23 | Medical Research Industries,Inc. | Topical composition for the relief of pain |
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- 1999-06-29 BR BR9912508-0A patent/BR9912508A/pt not_active Application Discontinuation
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- 1999-06-29 TR TR2000/03801T patent/TR200003801T2/xx unknown
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- 1999-06-29 ID IDW20010231A patent/ID28213A/id unknown
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2000
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- 2000-12-28 HR HR20000905A patent/HRP20000905A2/hr not_active Application Discontinuation
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Also Published As
| Publication number | Publication date |
|---|---|
| HUP0102728A3 (en) | 2002-12-28 |
| SK20012000A3 (sk) | 2001-08-06 |
| NO20006604D0 (no) | 2000-12-22 |
| HUP0102728A2 (hu) | 2002-03-28 |
| HRP20000905A2 (en) | 2001-08-31 |
| NO20006604L (no) | 2001-02-28 |
| EP1093348A1 (en) | 2001-04-25 |
| WO2000000120A9 (en) | 2000-03-30 |
| BR9912508A (pt) | 2001-05-02 |
| TR200003801T2 (tr) | 2001-06-21 |
| WO2000000120A1 (en) | 2000-01-06 |
| EP1093348A4 (en) | 2003-07-16 |
| AU4841599A (en) | 2000-01-17 |
| BG105175A (bg) | 2001-11-30 |
| MXPA00012767A (es) | 2002-08-09 |
| CA2335837A1 (en) | 2000-01-06 |
| IL140420A0 (en) | 2002-02-10 |
| PL345216A1 (en) | 2001-12-03 |
| JP2002519310A (ja) | 2002-07-02 |
| ID28213A (id) | 2001-05-10 |
| KR20010078754A (ko) | 2001-08-21 |
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