CN109071407A - 一种沙库必曲的中间体及其制备方法 - Google Patents

一种沙库必曲的中间体及其制备方法 Download PDF

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CN109071407A
CN109071407A CN201780013500.0A CN201780013500A CN109071407A CN 109071407 A CN109071407 A CN 109071407A CN 201780013500 A CN201780013500 A CN 201780013500A CN 109071407 A CN109071407 A CN 109071407A
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acid ester
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陈磊
孙国栋
韩小东
李顺
曾洁滨
王仲清
罗忠华
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Sunshine Lake Pharma Co Ltd
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Abstract

本发明涉及一种沙库必曲中间体及其制备方法,本发明所述的沙库必曲中间体,其可以通过一种化合物经过脱保护反应制备获得;另外,可采用所述中间体作为物料进一步地合成沙库必曲化合物。本发明所述的方法具有原料易得、工艺简洁、经济环保等优点,非常适合工业化生产。

Description

PCT国内申请,说明书已公开。

Claims (35)

  1. PCT国内申请,权利要求书已公开。
CN201780013500.0A 2016-02-29 2017-02-28 一种沙库必曲的中间体及其制备方法 Pending CN109071407A (zh)

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EP3424899A1 (en) 2019-01-09
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