CN101186587B - 一种β-氨基酸的衍生物合成方法及其中间产物 - Google Patents
一种β-氨基酸的衍生物合成方法及其中间产物 Download PDFInfo
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CN2006101294313A CN101186587B (zh) | 2006-11-16 | 2006-11-16 | 一种β-氨基酸的衍生物合成方法及其中间产物 |
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CN101186587A CN101186587A (zh) | 2008-05-28 |
CN101186587B true CN101186587B (zh) | 2010-04-21 |
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Families Citing this family (5)
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CN101279929B (zh) * | 2007-09-04 | 2011-04-20 | 重庆博腾制药科技股份有限公司 | 一种光学活性的3-氨基-n-环丙基-2-羟基己酰胺的制备方法 |
CN101691338B (zh) * | 2009-08-26 | 2013-08-14 | 凯莱英生命科学技术(天津)有限公司 | 一种手性环氧化合物的合成方法及其中间产物与最终产物 |
BR112014030870A2 (pt) * | 2012-06-13 | 2017-06-27 | Janssen Pharmaceutica Nv | método para preparação de 3-amino-n-ciclopropil-2-hidroxil- hexanamida |
CN106191147B (zh) * | 2016-07-08 | 2020-03-27 | 凯莱英医药集团(天津)股份有限公司 | 手性β-氨基酸的制备方法 |
CN108048317B (zh) * | 2017-12-12 | 2023-08-15 | 凯莱英医药集团(天津)股份有限公司 | 一种非天然氨基酸的连续合成***及连续合成方法 |
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Joseph Cacciola.the synthesis of lysine a-ketoamide thrombin inhibitors via anamide ring opening.Tetrahedron Letters38 33.1997,38(33),5741-5744. * |
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Effective date of registration: 20090227 Address after: Zip code six, Dongting Sanjie, Seventh Avenue, Tianjin economic and Technological Development Zone, Tianjin, China: 300457 Applicant after: Chinese medicine and Chemistry (Tianjin) Co., Ltd. Co-applicant after: Asymchem Life Science and Technology (Tianjin) Co., Ltd. Co-applicant after: Fu Xin Address before: Six, Dongting street, Seventh Street, TEDA Development Zone, Tianjin, Tianjin, China: 300457 Applicant before: Kailaiying Medical Chemical (Tianjin) Co., Ltd. |
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Owner name: ASYMCHEM LABORATORIES UXIN ) TECHNOLOGY CO., LTD. Free format text: FORMER OWNER: GLORIAIN MEDICINE CHEMICAL ( TIANJIN ) CO., LTD. Effective date: 20091002 |
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Effective date of registration: 20091002 Address after: E 42, road, Fuxin economic and Technological Development Zone, Liaoning 123000, China Applicant after: Asymchem Medicinal and Pharmaceutical Chemistry (Fuxin) Co., Ltd. Address before: Zip code six, Dongting Sanjie, Seventh Avenue, Tianjin economic and Technological Development Zone, Tianjin, China: 300457 Applicant before: Chinese medicine and Chemistry (Tianjin) Co., Ltd. Co-applicant before: Asymchem Life Science and Technology (Tianjin) Co., Ltd. Co-applicant before: Asymchem Medicinal and Pharmaceutical Chemistry (Fuxin) Co., Ltd. Co-applicant before: Jilin Asymchem Medicinal and Pharmaceutical Chemistry Co., Ltd. |
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