CL2015001891A1 - Formas de dosis de liberación controlada encerradas resistentes a manipulaciones indebidas; uso para tratar el dolor; y metodo de preparacion. (divisional de la solicitud n°2754-2014). - Google Patents

Formas de dosis de liberación controlada encerradas resistentes a manipulaciones indebidas; uso para tratar el dolor; y metodo de preparacion. (divisional de la solicitud n°2754-2014).

Info

Publication number
CL2015001891A1
CL2015001891A1 CL2015001891A CL2015001891A CL2015001891A1 CL 2015001891 A1 CL2015001891 A1 CL 2015001891A1 CL 2015001891 A CL2015001891 A CL 2015001891A CL 2015001891 A CL2015001891 A CL 2015001891A CL 2015001891 A1 CL2015001891 A1 CL 2015001891A1
Authority
CL
Chile
Prior art keywords
preparation
divisional
tampering
application
dosage forms
Prior art date
Application number
CL2015001891A
Other languages
English (en)
Inventor
Haiyong Hugh Huang
Original Assignee
Purdue Pharma Lp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45563448&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2015001891(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Purdue Pharma Lp filed Critical Purdue Pharma Lp
Publication of CL2015001891A1 publication Critical patent/CL2015001891A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

FORMA DE DOSIS DE LIBERACION CONTROLADA SOLIDA QUE COMPRENDE UN NUCLEO CON UNA PRIMERA PORCION DE UN ANALGESICO OPIOIDE Y UNA CUBIERTA QUE ENCIERRA EL NUCLEO, CON UNA SEGUNDA PORCION DEL ANALGESICO OPIOIDE; METODO DE PREPARACION; Y SU USO PARA EL TRATAMIENTO DEL DOLOR. (DIVISIONAL DE SOLICITUD 2754-2014).
CL2015001891A 2010-12-22 2015-06-30 Formas de dosis de liberación controlada encerradas resistentes a manipulaciones indebidas; uso para tratar el dolor; y metodo de preparacion. (divisional de la solicitud n°2754-2014). CL2015001891A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201061426306P 2010-12-22 2010-12-22

Publications (1)

Publication Number Publication Date
CL2015001891A1 true CL2015001891A1 (es) 2015-10-23

Family

ID=45563448

Family Applications (4)

Application Number Title Priority Date Filing Date
CL2013001781A CL2013001781A1 (es) 2010-12-22 2013-06-18 Forma de dosis de liberacion controlada solida que comprende un nucleo con una primera porcion de un analgesico opioide y una cubierta que encierra el nucleo y que comprende una segunda porcion del analgesico, la cual es resistente a manipulaciones indebidas.
CL2014001450A CL2014001450A1 (es) 2010-12-22 2014-06-02 Forma de dosis de liberacion controlada solida que comprende un analgesico opioide dispersado en un material de matriz; metodo de preparacion; uso en el tratamiento del dolor.
CL2014002754A CL2014002754A1 (es) 2010-12-22 2014-10-14 Forma de dosis de liberación controlada solida que comprende un nucleo con una primera porcion de un analgesico opioide y una cubierta que encierra el nucleo y comprende una segunda porcion del analgesico opioide; metodo de preparacion; uso en el tratamiento del dolor. (divisional de solicitud n°1450-2014).
CL2015001891A CL2015001891A1 (es) 2010-12-22 2015-06-30 Formas de dosis de liberación controlada encerradas resistentes a manipulaciones indebidas; uso para tratar el dolor; y metodo de preparacion. (divisional de la solicitud n°2754-2014).

Family Applications Before (3)

Application Number Title Priority Date Filing Date
CL2013001781A CL2013001781A1 (es) 2010-12-22 2013-06-18 Forma de dosis de liberacion controlada solida que comprende un nucleo con una primera porcion de un analgesico opioide y una cubierta que encierra el nucleo y que comprende una segunda porcion del analgesico, la cual es resistente a manipulaciones indebidas.
CL2014001450A CL2014001450A1 (es) 2010-12-22 2014-06-02 Forma de dosis de liberacion controlada solida que comprende un analgesico opioide dispersado en un material de matriz; metodo de preparacion; uso en el tratamiento del dolor.
CL2014002754A CL2014002754A1 (es) 2010-12-22 2014-10-14 Forma de dosis de liberación controlada solida que comprende un nucleo con una primera porcion de un analgesico opioide y una cubierta que encierra el nucleo y comprende una segunda porcion del analgesico opioide; metodo de preparacion; uso en el tratamiento del dolor. (divisional de solicitud n°1450-2014).

Country Status (41)

Country Link
US (12) US8808740B2 (es)
EP (4) EP2826467B1 (es)
JP (2) JP5911509B2 (es)
KR (2) KR101647267B1 (es)
CN (2) CN104873455B (es)
AP (2) AP3815A (es)
AR (1) AR084575A1 (es)
AU (3) AU2011346757B2 (es)
CA (3) CA2822790C (es)
CL (4) CL2013001781A1 (es)
CO (1) CO6731103A2 (es)
CR (1) CR20130544A (es)
CY (1) CY1119312T1 (es)
DK (1) DK2826467T3 (es)
DO (2) DOP2013000140A (es)
EA (1) EA032906B1 (es)
EC (1) ECSP13012760A (es)
ES (1) ES2643291T3 (es)
GT (1) GT201300166A (es)
HK (3) HK1204561A1 (es)
HR (1) HRP20171366T1 (es)
HU (1) HUE034955T2 (es)
IL (1) IL226811B (es)
LT (1) LT2826467T (es)
ME (1) ME02874B (es)
MX (1) MX367010B (es)
MY (1) MY166034A (es)
NI (1) NI201300054A (es)
NZ (2) NZ708728A (es)
PE (2) PE20181177A1 (es)
PH (2) PH12015501411A1 (es)
PL (1) PL2826467T3 (es)
PT (1) PT2826467T (es)
RS (1) RS56344B1 (es)
SA (2) SA111330106B1 (es)
SG (2) SG191288A1 (es)
SI (1) SI2826467T1 (es)
TN (1) TN2013000264A1 (es)
TW (2) TWI538699B (es)
UA (1) UA114887C2 (es)
WO (1) WO2012085656A2 (es)

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