CL2008003584A1 - Uso de la 10-[(3r)-1-azabiciclo]oct-3-ilmetil]-10-h-fenotiazina, o una de sus sales farmaceuticamente aceptables para la preparación de un medicamento util para prevenir o tratar la bronconeumopatia obstructiva. - Google Patents

Uso de la 10-[(3r)-1-azabiciclo]oct-3-ilmetil]-10-h-fenotiazina, o una de sus sales farmaceuticamente aceptables para la preparación de un medicamento util para prevenir o tratar la bronconeumopatia obstructiva.

Info

Publication number
CL2008003584A1
CL2008003584A1 CL2008003584A CL2008003584A CL2008003584A1 CL 2008003584 A1 CL2008003584 A1 CL 2008003584A1 CL 2008003584 A CL2008003584 A CL 2008003584A CL 2008003584 A CL2008003584 A CL 2008003584A CL 2008003584 A1 CL2008003584 A1 CL 2008003584A1
Authority
CL
Chile
Prior art keywords
azabicyclo
phenothiazine
ylmethyl
oct
preparation
Prior art date
Application number
CL2008003584A
Other languages
English (en)
Inventor
Thierry Clerc
Jacky Tisne-Versailles
Christophe Przybylski
Didier Cussac
Original Assignee
Pf Medicament
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pf Medicament filed Critical Pf Medicament
Publication of CL2008003584A1 publication Critical patent/CL2008003584A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

Uso de la 10-[(3R)-1-azabiciclo]oct-3-ilmetil]-10-H-fenotiazina, o una de sus sales farmacéuticamente aceptables, que sirve para la preparación de un medicamento útil para prevenir o tratar la bronconeumopatía obstructiva, donde el medicamento se presenta en forma de tableta, en forma de disolución para pulverización oral, o de un polvo para la inhalación.
CL2008003584A 2007-12-04 2008-12-01 Uso de la 10-[(3r)-1-azabiciclo]oct-3-ilmetil]-10-h-fenotiazina, o una de sus sales farmaceuticamente aceptables para la preparación de un medicamento util para prevenir o tratar la bronconeumopatia obstructiva. CL2008003584A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0759538A FR2924344B1 (fr) 2007-12-04 2007-12-04 Utilisation de la mequitazine sous la forme de racemate ou d'enantiomeres pour la preparation d'un medicament destine au traitement ou a la prevention de pathologies impliquant les recepteurs histaminiques h4.
FR0854144A FR2924345B1 (fr) 2007-12-04 2008-06-23 Utilisation de la mequitazine sous la forme de racemate ou d'enantiomeres pour la preparation d'un medicament destine au traitement ou a la prevention de pathologies impliquant les recepteurs histaminiques h4.

Publications (1)

Publication Number Publication Date
CL2008003584A1 true CL2008003584A1 (es) 2009-05-22

Family

ID=39522380

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2008003584A CL2008003584A1 (es) 2007-12-04 2008-12-01 Uso de la 10-[(3r)-1-azabiciclo]oct-3-ilmetil]-10-h-fenotiazina, o una de sus sales farmaceuticamente aceptables para la preparación de un medicamento util para prevenir o tratar la bronconeumopatia obstructiva.

Country Status (22)

Country Link
US (1) US20100273752A1 (es)
EP (2) EP2227235B1 (es)
JP (2) JP2011505411A (es)
KR (1) KR20100108347A (es)
CN (1) CN101883566B (es)
AR (1) AR070673A1 (es)
AU (1) AU2008333220B2 (es)
BR (1) BRPI0820652A2 (es)
CA (1) CA2706898A1 (es)
CL (1) CL2008003584A1 (es)
FR (2) FR2924344B1 (es)
HK (1) HK1148667A1 (es)
IL (1) IL206073A0 (es)
MA (1) MA31930B1 (es)
MX (1) MX2010006139A (es)
NZ (1) NZ586212A (es)
PA (1) PA8805501A1 (es)
RU (1) RU2510273C2 (es)
TN (1) TN2010000241A1 (es)
TW (1) TW200932242A (es)
WO (1) WO2009071625A1 (es)
ZA (2) ZA201004312B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2201982A1 (en) 2008-12-24 2010-06-30 INSERM (Institut National de la Santé et de la Recherche Médicale) Histamine H4 receptor antagonists for the treatment of vestibular disorders
HUE039713T2 (hu) 2012-06-08 2019-02-28 Sensorion H4 receptor inhibitorok tinnitus kezelésére

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2440371A1 (fr) * 1978-10-31 1980-05-30 Fisons Ltd Nouveaux composes azotes heterocycliques, des compositions pharmaceutiques en contenant et des procedes pour les preparer
FR2522660A1 (fr) * 1982-03-05 1983-09-09 Pharmuka Lab Isomere levogyre de la mequitazine, son procede de preparation et medicaments le contenant
JPS6330420A (ja) * 1986-07-25 1988-02-09 Sekisui Chem Co Ltd 持続性抗アレルギ−固形塗布剤
JP2735122B2 (ja) * 1988-06-13 1998-04-02 旭化成工業株式会社 メキタジンの液状シロップ製剤
IT1251161B (it) * 1991-08-07 1995-05-04 Derivati ammonio quaternari di (-) e (+)-3-(10 h-fenotiazin-10-ilmetil)-l-azabiciclo (2.2.2.)ottano e composizioni farmaceutiche che li contengono
DE19653969A1 (de) * 1996-12-20 1998-06-25 Boehringer Ingelheim Kg Neue wässrige Arzneimittelzubereitung zur Erzeugung treibgasfreier Aerosole
FR2822709B1 (fr) * 2001-03-30 2007-01-19 Antialis Composition pharmaceutique anti-allergique comprenant au moins un allergene et au moins un compose antihistaminique
DE10158036B4 (de) * 2001-11-27 2007-05-03 Kosmas Kg Antiallergisches Mittel und dessen Verwendung
US20050090527A1 (en) * 2003-01-28 2005-04-28 Schering Corporation Combination of H1, H3 and H4 receptor antagonists for treatment of allergic and non-allergic pulmonary inflammation, congestion and allergic rhinitis
JP2005060233A (ja) * 2003-08-08 2005-03-10 Rohto Pharmaceut Co Ltd 皮膚外用剤
EP1526135A1 (en) * 2003-10-24 2005-04-27 Warner-Lambert Company LLC Azabenzodiazepines as pde4 inhibitors
WO2005063253A1 (ja) * 2003-12-26 2005-07-14 Taiho Pharmaceutical Co., Ltd. アレルギー症状治療用医薬組成物
FR2896690B1 (fr) * 2006-01-30 2008-05-02 Pierre Fabre Medicament Sa Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique

Also Published As

Publication number Publication date
EP2227235A1 (en) 2010-09-15
TN2010000241A1 (en) 2011-11-11
NZ586212A (en) 2012-09-28
CN101883566A (zh) 2010-11-10
FR2924344B1 (fr) 2010-04-16
WO2009071625A1 (en) 2009-06-11
RU2510273C2 (ru) 2014-03-27
BRPI0820652A2 (pt) 2019-09-10
IL206073A0 (en) 2010-11-30
EP2227235B1 (en) 2014-11-12
PA8805501A1 (es) 2009-12-16
FR2924345A1 (fr) 2009-06-05
EP2255811A1 (en) 2010-12-01
FR2924345B1 (fr) 2010-06-04
HK1148667A1 (en) 2011-09-16
TW200932242A (en) 2009-08-01
KR20100108347A (ko) 2010-10-06
FR2924344A1 (fr) 2009-06-05
JP2014065726A (ja) 2014-04-17
ZA201007626B (en) 2011-08-31
AR070673A1 (es) 2010-04-28
CN101883566B (zh) 2013-03-06
AU2008333220A1 (en) 2009-06-11
US20100273752A1 (en) 2010-10-28
ZA201004312B (en) 2011-02-23
AU2008333220B2 (en) 2014-04-24
MA31930B1 (fr) 2010-12-01
CA2706898A1 (en) 2009-06-11
RU2010125711A (ru) 2012-01-10
MX2010006139A (es) 2010-10-15
JP2011505411A (ja) 2011-02-24

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