CL2008001104A1 - Compuestos derivados de [1,2,3]triazolo[4,5-b]piridin-carboxamidas y [1,2,3]triazolo[4,5-d]pirimidin-carboxamidas, inhibidores de mgl y faah; procedimiento de preparacion; composicion farmaceutica; y su uso en el tratamiento de delolores agudos o cronicos, vertigos, vomitos, nauseas, sindrome metaloico, dispipidemia, entre otros. - Google Patents

Compuestos derivados de [1,2,3]triazolo[4,5-b]piridin-carboxamidas y [1,2,3]triazolo[4,5-d]pirimidin-carboxamidas, inhibidores de mgl y faah; procedimiento de preparacion; composicion farmaceutica; y su uso en el tratamiento de delolores agudos o cronicos, vertigos, vomitos, nauseas, sindrome metaloico, dispipidemia, entre otros.

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Publication number
CL2008001104A1
CL2008001104A1 CL2008001104A CL2008001104A CL2008001104A1 CL 2008001104 A1 CL2008001104 A1 CL 2008001104A1 CL 2008001104 A CL2008001104 A CL 2008001104A CL 2008001104 A CL2008001104 A CL 2008001104A CL 2008001104 A1 CL2008001104 A1 CL 2008001104A1
Authority
CL
Chile
Prior art keywords
carboxamides
triazolo
nausea
vomiting
acute
Prior art date
Application number
CL2008001104A
Other languages
English (en)
Inventor
Luc Hoornaert Christian Even
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of CL2008001104A1 publication Critical patent/CL2008001104A1/es

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract

Compuestos derivados de triazolopiridin-carboxamidas y triazolopirimidin-carboxamidas; procedimiento de preparación; composición farmacéutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de dolores agudos o crónicos, vértigos, vómitos, nauseas, síndrome metabólico, dislipidemia, epilepsia, cáncer, enfermedad infecciosa y viral.
CL2008001104A 2007-04-18 2008-04-17 Compuestos derivados de [1,2,3]triazolo[4,5-b]piridin-carboxamidas y [1,2,3]triazolo[4,5-d]pirimidin-carboxamidas, inhibidores de mgl y faah; procedimiento de preparacion; composicion farmaceutica; y su uso en el tratamiento de delolores agudos o cronicos, vertigos, vomitos, nauseas, sindrome metaloico, dispipidemia, entre otros. CL2008001104A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0702809A FR2915199B1 (fr) 2007-04-18 2007-04-18 Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.

Publications (1)

Publication Number Publication Date
CL2008001104A1 true CL2008001104A1 (es) 2009-01-16

Family

ID=38776272

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2008001104A CL2008001104A1 (es) 2007-04-18 2008-04-17 Compuestos derivados de [1,2,3]triazolo[4,5-b]piridin-carboxamidas y [1,2,3]triazolo[4,5-d]pirimidin-carboxamidas, inhibidores de mgl y faah; procedimiento de preparacion; composicion farmaceutica; y su uso en el tratamiento de delolores agudos o cronicos, vertigos, vomitos, nauseas, sindrome metaloico, dispipidemia, entre otros.

Country Status (17)

Country Link
US (1) US8080547B2 (es)
EP (1) EP2146990A1 (es)
JP (1) JP2010524904A (es)
KR (1) KR20090130057A (es)
CN (1) CN101668758A (es)
AR (1) AR066107A1 (es)
AU (1) AU2008257320A1 (es)
BR (1) BRPI0810440A2 (es)
CA (1) CA2683929A1 (es)
CL (1) CL2008001104A1 (es)
FR (1) FR2915199B1 (es)
IL (1) IL201450A0 (es)
MX (1) MX2009011212A (es)
RU (1) RU2009142431A (es)
TW (1) TW200901993A (es)
UY (1) UY31032A1 (es)
WO (1) WO2008145839A1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2915198B1 (fr) * 2007-04-18 2009-12-18 Sanofi Aventis Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique.
CN102333568B (zh) 2008-12-24 2016-01-20 比亚尔-珀特拉和Ca股份公司 药物化合物
AU2010238745A1 (en) * 2009-04-22 2011-11-10 Janssen Pharmaceutica Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitor
US8435977B2 (en) 2009-04-22 2013-05-07 Janssen Pharmaceutica, Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
KR20120005517A (ko) * 2009-04-22 2012-01-16 얀센 파마슈티카 엔.브이. 모노아실글리세롤 리파제 억제제로서의 헤테로방향족 및 방향족 피페라지닐 아제티디닐 아미드
EP2421848A1 (en) * 2009-04-22 2012-02-29 Janssen Pharmaceutica N.V. Azetidinyl diamides as monoacylglycerol lipase inhibitors
JP5738766B2 (ja) * 2009-09-09 2015-06-24 大日本住友製薬株式会社 ８−オキソジヒドロプリン誘導体
US20130150346A1 (en) 2010-01-08 2013-06-13 Quest Ventures Ltd. Use of FAAH Inhibitors for Treating Parkinson's Disease and Restless Legs Syndrome
WO2011101644A1 (en) 2010-02-18 2011-08-25 Centro Nacional De Investigaciones Oncologicas (Cnio) Triazolo [4, 5 - b] pyridin derivatives
US20130224151A1 (en) 2010-03-31 2013-08-29 United States Of America Use of FAAH Inhibitors for Treating Abdominal, Visceral and Pelvic Pain
NZ703111A (en) 2010-05-17 2016-07-29 Incozen Therapeutics Pvt Ltd Novel 3,5-disubstitued-3h-imidazo[4,5-b]pyridine and 3,5- disubstitued -3h-[1,2,3]triazolo[4,5-b] pyridine compounds as modulators of protein kinases
JP2013536852A (ja) 2010-09-03 2013-09-26 ヤンセン ファーマシューティカ エヌ．ベー． モノアシルグリセロールリパーゼ阻害剤としてのジ−アゼチジニルジアミド
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