CH512475A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH512475A
CH512475A CH952368A CH952368A CH512475A CH 512475 A CH512475 A CH 512475A CH 952368 A CH952368 A CH 952368A CH 952368 A CH952368 A CH 952368A CH 512475 A CH512475 A CH 512475A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH952368A
Other languages
English (en)
Inventor
Ian Fryer Rodney
Henryk Sternbach Leo
Valentine Earley James
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH512475A publication Critical patent/CH512475A/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CH952368A 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH512475A (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65065267A 1967-07-03 1967-07-03
US65065167A 1967-07-03 1967-07-03

Publications (1)

Publication Number Publication Date
CH512475A true CH512475A (de) 1971-09-15

Family

ID=27095915

Family Applications (3)

Application Number Title Priority Date Filing Date
CH892371A CH526558A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH892271A CH524621A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH952368A CH512475A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CH892371A CH526558A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH892271A CH524621A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (11)

Country Link
US (1) US3523939A (de)
BE (1) BE717478A (de)
CA (1) CA952106A (de)
CH (3) CH526558A (de)
DE (1) DE1770778A1 (de)
FR (2) FR8488M (de)
GB (2) GB1205995A (de)
IE (1) IE32217B1 (de)
IL (2) IL30282A (de)
NL (1) NL6809403A (de)
SE (1) SE358167B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4837280B1 (de) * 1969-03-08 1973-11-09
US3723414A (en) * 1970-02-13 1973-03-27 Schering Corp 1-polyfluoroalkyl benzodiazepines
AT333284B (de) * 1971-12-09 1976-11-10 Degussa Verfahren zur herstellung von neuen 6-aza-3h-1,4-benzodiazepinen, deren optischen isomeren und deren salzen
US4089953A (en) * 1973-06-20 1978-05-16 Ddsa Pharmaceuticals 1,5-Benzodiazocines
US4056525A (en) * 1975-06-02 1977-11-01 American Home Products Corporation 2,3-dialkoxy-3h-1,4-benzodiazepines
WO2008141081A1 (en) * 2007-05-10 2008-11-20 Amr Technology, Inc. Aryl- and heteroaryl-substituted tetrahydrobenzo-1,4-diazepines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
US9249161B2 (en) 2010-12-02 2016-02-02 Constellation Pharmaceuticals, Inc. Bromodomain inhibitors and uses thereof
AR084070A1 (es) 2010-12-02 2013-04-17 Constellation Pharmaceuticals Inc Inhibidores del bromodominio y usos de los mismos
US9422292B2 (en) 2011-05-04 2016-08-23 Constellation Pharmaceuticals, Inc. Bromodomain inhibitors and uses thereof
EP2721031B1 (de) 2011-06-17 2016-01-20 Constellation Pharmaceuticals, Inc. Bromodomainhemmer und ihre verwendungen
EP2864336B1 (de) 2012-06-06 2016-11-23 Constellation Pharmaceuticals, Inc. Benzo[b]isoxazolazepinbromdomänenhemmer und verwendungen davon
TWI602820B (zh) 2012-06-06 2017-10-21 星宿藥物公司 溴域抑制劑及其用途
EP3157928B1 (de) 2014-06-20 2019-02-13 Constellation Pharmaceuticals, Inc. Kristalline formen von 2-((4s)-6-(4-chlorophenyl)-1-methyl-4h-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamid

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2893992A (en) * 1959-07-07 I ii i i
US3109843A (en) * 1963-11-05 Process for preparing
US3371085A (en) * 1959-12-10 1968-02-27 Hoffmann La Roche 5-aryl-3h-1,4-benzodiazepin-2(1h)-ones
GB1051795A (de) * 1964-02-11

Also Published As

Publication number Publication date
SE358167B (de) 1973-07-23
US3523939A (en) 1970-08-11
CH524621A (de) 1972-06-30
DE1770778A1 (de) 1972-02-17
IE32217B1 (en) 1973-05-16
FR8488M (de) 1973-07-27
CA952106A (en) 1974-07-30
GB1205995A (en) 1970-09-23
IE32217L (en) 1969-01-03
CH526558A (de) 1972-08-15
IL30282A0 (en) 1968-09-26
IL30282A (en) 1972-11-28
FR1586872A (de) 1970-03-06
GB1205996A (en) 1970-09-23
NL6809403A (de) 1969-01-07
IL38208A (en) 1973-04-30
BE717478A (de) 1969-01-02

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Legal Events

Date Code Title Description
PL Patent ceased