CA2355738A1 - 3,6-disubstituted penam sulfone derivatives as antibacterials - Google Patents

3,6-disubstituted penam sulfone derivatives as antibacterials Download PDF

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Publication number
CA2355738A1
CA2355738A1 CA002355738A CA2355738A CA2355738A1 CA 2355738 A1 CA2355738 A1 CA 2355738A1 CA 002355738 A CA002355738 A CA 002355738A CA 2355738 A CA2355738 A CA 2355738A CA 2355738 A1 CA2355738 A1 CA 2355738A1
Authority
CA
Canada
Prior art keywords
compound
hydrogen
methyl
pharmaceutically acceptable
carbamoyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002355738A
Other languages
English (en)
French (fr)
Inventor
Yang-I Lin
Panayota Bitha
Zhong Li
Gerardo Delacruz Francisco
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Holdings LLC
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2355738A1 publication Critical patent/CA2355738A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
CA002355738A 1999-01-26 2000-01-26 3,6-disubstituted penam sulfone derivatives as antibacterials Abandoned CA2355738A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23772699A 1999-01-26 1999-01-26
US09/237,726 1999-01-26
PCT/US2000/001630 WO2000043399A1 (en) 1999-01-26 2000-01-26 3,6-disubstituted penam sulfone derivatives as antibacterials

Publications (1)

Publication Number Publication Date
CA2355738A1 true CA2355738A1 (en) 2000-07-27

Family

ID=22894903

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002355738A Abandoned CA2355738A1 (en) 1999-01-26 2000-01-26 3,6-disubstituted penam sulfone derivatives as antibacterials

Country Status (20)

Country Link
EP (1) EP1144418A1 (de)
JP (1) JP2002535335A (de)
KR (1) KR20010101649A (de)
CN (1) CN1188417C (de)
AU (1) AU2624600A (de)
BG (1) BG105737A (de)
BR (1) BR0007729A (de)
CA (1) CA2355738A1 (de)
CZ (1) CZ20012691A3 (de)
EA (1) EA200100813A1 (de)
HK (1) HK1038747A1 (de)
HU (1) HUP0200013A3 (de)
ID (1) ID29400A (de)
IL (1) IL144116A0 (de)
NO (1) NO20013640L (de)
PL (1) PL349874A1 (de)
SK (1) SK10142001A3 (de)
TR (1) TR200102133T2 (de)
WO (1) WO2000043399A1 (de)
ZA (1) ZA200104323B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5705751B2 (ja) * 2009-03-10 2015-04-22 レール・リキード−ソシエテ・アノニム・プール・レテュード・エ・レクスプロワタシオン・デ・プロセデ・ジョルジュ・クロード ｌｏｗ−ｋシリル化用の環式アミノ化合物
CN109422765B (zh) * 2017-09-05 2020-08-28 香港理工大学深圳研究院 C类β-内酰胺酶抑制剂及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2076812A (en) * 1980-05-22 1981-12-09 Ciba Geigy Ag Penam-dioxide compounds, processes for their manufacture, and their use
EP0083977A1 (de) * 1982-01-11 1983-07-20 Pfizer Inc. 6-Alpha-Hydroxymethyl-Penicillansäure-Sulfon als Beta-Lactamase-Inhibitor
US4562073A (en) * 1982-12-24 1985-12-31 Taiho Pharmaceutical Company Limited Penicillin derivatives
US4503040A (en) * 1984-02-27 1985-03-05 Pfizer Inc. 6-(Aminoacyloxymethyl)penicillanic acid 1,1-dioxides as beta-lactamase inhibitors
US4591459A (en) * 1984-12-03 1986-05-27 Pfizer Inc. Intermediates for 6-(aminoacyloxymethyl) penicillanic acid 1,1-dioxides
TW383308B (en) * 1993-08-24 2000-03-01 Hoffmann La Roche 2-beta-alkenyl penam sulfones as beta-lactamase inhibitors

Also Published As

Publication number Publication date
ID29400A (id) 2001-08-30
CZ20012691A3 (cs) 2002-06-12
CN1188417C (zh) 2005-02-09
HUP0200013A2 (hu) 2002-05-29
PL349874A1 (en) 2002-09-23
BG105737A (en) 2002-05-31
HUP0200013A3 (en) 2002-10-28
NO20013640D0 (no) 2001-07-24
JP2002535335A (ja) 2002-10-22
CN1337965A (zh) 2002-02-27
EP1144418A1 (de) 2001-10-17
IL144116A0 (en) 2002-05-23
ZA200104323B (en) 2002-08-26
AU2624600A (en) 2000-08-07
TR200102133T2 (tr) 2001-12-21
NO20013640L (no) 2001-07-24
EA200100813A1 (ru) 2003-02-27
WO2000043399A1 (en) 2000-07-27
SK10142001A3 (sk) 2002-07-02
BR0007729A (pt) 2001-10-30
HK1038747A1 (zh) 2002-03-28
KR20010101649A (ko) 2001-11-14

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued