TR200102133T2 - Antibakteriyal olarak 3,6-di-ikame edilmiş penam sülfon türevleri. - Google Patents

Antibakteriyal olarak 3,6-di-ikame edilmiş penam sülfon türevleri.

Info

Publication number
TR200102133T2
TR200102133T2 TR2001/02133T TR200102133T TR200102133T2 TR 200102133 T2 TR200102133 T2 TR 200102133T2 TR 2001/02133 T TR2001/02133 T TR 2001/02133T TR 200102133 T TR200102133 T TR 200102133T TR 200102133 T2 TR200102133 T2 TR 200102133T2
Authority
TR
Turkey
Prior art keywords
antibacterial
substituted
sulfone derivatives
carbamoyl
cyano
Prior art date
Application number
TR2001/02133T
Other languages
English (en)
Inventor
Lin Yang-I
Bitha Panayota
Li Zhong
Delacruz Francisco Gerardo
Original Assignee
American Cyanamid Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Company filed Critical American Cyanamid Company
Publication of TR200102133T2 publication Critical patent/TR200102133T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

sFormül (I) ve formül (II)'nin bilesimleri sunulmaktadir; öyle ki bu formüllerde n, 0 veya 1'dir ve n=1 oldugunda R, 5 veya 6 üyeli olan bir heterosiklik halka, hidroksi, halojen, okso, karbamoil, alkoksi veya di-ikame edilmis aminodur; n=0 oldugunda R bir ester, siyano veya amid gubudur; X, CH ya da NH'dir; R3 siyano, metoksi veya asetamidodur; R1 hidrojen, alkil, bir negatif yük, sodyum, potasyum, tetraalkilamonyum ve asiloksialkil veya alkoksikarboniloksialkil içeren bir gruptan seçilmis bir katyondur ve R2 hidrojen, asil, tri-ikameli silil karbamoil veya bir amino asit artigidir, veya bunun farmasötik olarak kabul edilebilir tuzlari sunulur.
TR2001/02133T 1999-01-26 2000-01-26 Antibakteriyal olarak 3,6-di-ikame edilmiş penam sülfon türevleri. TR200102133T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23772699A 1999-01-26 1999-01-26

Publications (1)

Publication Number Publication Date
TR200102133T2 true TR200102133T2 (tr) 2001-12-21

Family

ID=22894903

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/02133T TR200102133T2 (tr) 1999-01-26 2000-01-26 Antibakteriyal olarak 3,6-di-ikame edilmiş penam sülfon türevleri.

Country Status (20)

Country Link
EP (1) EP1144418A1 (tr)
JP (1) JP2002535335A (tr)
KR (1) KR20010101649A (tr)
CN (1) CN1188417C (tr)
AU (1) AU2624600A (tr)
BG (1) BG105737A (tr)
BR (1) BR0007729A (tr)
CA (1) CA2355738A1 (tr)
CZ (1) CZ20012691A3 (tr)
EA (1) EA200100813A1 (tr)
HK (1) HK1038747A1 (tr)
HU (1) HUP0200013A3 (tr)
ID (1) ID29400A (tr)
IL (1) IL144116A0 (tr)
NO (1) NO20013640L (tr)
PL (1) PL349874A1 (tr)
SK (1) SK10142001A3 (tr)
TR (1) TR200102133T2 (tr)
WO (1) WO2000043399A1 (tr)
ZA (1) ZA200104323B (tr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5705751B2 (ja) * 2009-03-10 2015-04-22 レール・リキード−ソシエテ・アノニム・プール・レテュード・エ・レクスプロワタシオン・デ・プロセデ・ジョルジュ・クロード ｌｏｗ−ｋシリル化用の環式アミノ化合物
CN109422765B (zh) * 2017-09-05 2020-08-28 香港理工大学深圳研究院 C类β-内酰胺酶抑制剂及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2076812A (en) * 1980-05-22 1981-12-09 Ciba Geigy Ag Penam-dioxide compounds, processes for their manufacture, and their use
EP0083977A1 (en) * 1982-01-11 1983-07-20 Pfizer Inc. 6-Alpha-hydroxymethylpenicillanic acid sulfone as a beta-lactamase inhibitor
US4562073A (en) * 1982-12-24 1985-12-31 Taiho Pharmaceutical Company Limited Penicillin derivatives
US4503040A (en) * 1984-02-27 1985-03-05 Pfizer Inc. 6-(Aminoacyloxymethyl)penicillanic acid 1,1-dioxides as beta-lactamase inhibitors
US4591459A (en) * 1984-12-03 1986-05-27 Pfizer Inc. Intermediates for 6-(aminoacyloxymethyl) penicillanic acid 1,1-dioxides
TW383308B (en) * 1993-08-24 2000-03-01 Hoffmann La Roche 2-beta-alkenyl penam sulfones as beta-lactamase inhibitors

Also Published As

Publication number Publication date
ID29400A (id) 2001-08-30
CZ20012691A3 (cs) 2002-06-12
CN1188417C (zh) 2005-02-09
HUP0200013A2 (hu) 2002-05-29
PL349874A1 (en) 2002-09-23
BG105737A (en) 2002-05-31
HUP0200013A3 (en) 2002-10-28
NO20013640D0 (no) 2001-07-24
JP2002535335A (ja) 2002-10-22
CN1337965A (zh) 2002-02-27
EP1144418A1 (en) 2001-10-17
IL144116A0 (en) 2002-05-23
ZA200104323B (en) 2002-08-26
AU2624600A (en) 2000-08-07
NO20013640L (no) 2001-07-24
EA200100813A1 (ru) 2003-02-27
WO2000043399A1 (en) 2000-07-27
CA2355738A1 (en) 2000-07-27
SK10142001A3 (sk) 2002-07-02
BR0007729A (pt) 2001-10-30
HK1038747A1 (zh) 2002-03-28
KR20010101649A (ko) 2001-11-14

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