CA1051420A - ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDS - Google Patents
ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDSInfo
- Publication number
- CA1051420A CA1051420A CA165,831A CA165831A CA1051420A CA 1051420 A CA1051420 A CA 1051420A CA 165831 A CA165831 A CA 165831A CA 1051420 A CA1051420 A CA 1051420A
- Authority
- CA
- Canada
- Prior art keywords
- formula
- compound
- process according
- penicillanate
- ethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB1168972A GB1427139A (en) | 1972-03-13 | 1972-03-13 | Penicillins |
Publications (1)
Publication Number | Publication Date |
---|---|
CA1051420A true CA1051420A (en) | 1979-03-27 |
Family
ID=9990894
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA165,831A Expired CA1051420A (en) | 1972-03-13 | 1973-03-12 | ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDS |
Country Status (10)
Country | Link |
---|---|
JP (3) | JPS5526147B2 (de) |
AT (1) | AT331391B (de) |
CA (1) | CA1051420A (de) |
CH (2) | CH582707A5 (de) |
DE (1) | DE2311131C3 (de) |
DK (1) | DK145699C (de) |
FR (1) | FR2181811B1 (de) |
GB (1) | GB1427139A (de) |
NL (1) | NL176943C (de) |
SE (2) | SE416811B (de) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1427139A (en) * | 1972-03-13 | 1976-03-10 | Astra Laekemedel Ab | Penicillins |
SU566843A1 (ru) * | 1975-01-06 | 1977-07-30 | Ордена Трудового Красного Знамени Институт Органической Синтеза Ан Латвийской Сср | Способ получени производных 6- -амидинопенициллановой кислоты |
GB1529448A (en) * | 1975-10-29 | 1978-10-18 | Leo Pharm Prod Ltd | 6-amidinopenicillanic acid derivatives |
GB1579931A (en) * | 1976-04-15 | 1980-11-26 | Leo Pharm Prod Ltd | Bis-penicillanoyl-oxy-alkanes |
GB1585165A (en) * | 1976-06-29 | 1981-02-25 | Leo Pharm Prod Ltd | Derivatives of 6-amidino penicillanic acid |
US4345071A (en) | 1976-06-29 | 1982-08-17 | Leo Pharmaceutical Products, Ltd. A/S | Derivatives of penicillanic acid |
LU77362A1 (de) * | 1977-05-17 | 1979-01-19 | ||
IL54859A (en) * | 1977-06-21 | 1982-01-31 | Rech Applications Therap | Derivatives of amidinopenicillanic acid,their production and pharmaceutical compositions containing them |
JPS57156495A (en) * | 1981-03-23 | 1982-09-27 | Kyoto Yakuhin Kogyo Kk | Cephalosporin derivative and remedy for microbism used in oral administration |
JPS5865474U (ja) * | 1981-10-28 | 1983-05-04 | 松下電器産業株式会社 | 電動弁 |
IT1190897B (it) * | 1982-06-29 | 1988-02-24 | Opos Biochimica Srl | Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico |
US4606865A (en) * | 1982-09-20 | 1986-08-19 | Astra Lakemedel Aktiebolag | Methods for the preparation of α-bromodiethylcarbonate |
JPH0495170U (de) * | 1990-12-27 | 1992-08-18 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1003479A (en) * | 1963-05-30 | 1965-09-02 | Wyeth John & Brother Ltd | Acetoxymethyl benzylpenicillinate |
DE1795423C3 (de) * | 1967-09-29 | 1974-02-28 | Loevens Kemiske Fabrik Produktionsaktieselskab, Ballerup (Daenemark) | Pivaloyloxymethyl-alpha-aminobenzylpenicillinat |
BE758782A (fr) * | 1969-11-11 | 1971-05-10 | Leo Pharm Prod Ltd | Nouveaux derives d'acide 6-amidino penicillanique leur procede de preparation et leurs applications comme antibiotiques |
JPS4828904A (de) * | 1971-08-19 | 1973-04-17 | ||
GB1427139A (en) * | 1972-03-13 | 1976-03-10 | Astra Laekemedel Ab | Penicillins |
-
1972
- 1972-03-13 GB GB1168972A patent/GB1427139A/en not_active Expired
- 1972-03-15 SE SE7203298A patent/SE416811B/xx unknown
- 1972-03-15 DK DK119772A patent/DK145699C/da active
-
1973
- 1973-03-07 DE DE2311131A patent/DE2311131C3/de not_active Expired
- 1973-03-12 JP JP2890473A patent/JPS5526147B2/ja not_active Expired
- 1973-03-12 AT AT213973A patent/AT331391B/de not_active IP Right Cessation
- 1973-03-12 NL NLAANVRAGE7303434,A patent/NL176943C/xx not_active IP Right Cessation
- 1973-03-12 FR FR7308757A patent/FR2181811B1/fr not_active Expired
- 1973-03-12 CA CA165,831A patent/CA1051420A/en not_active Expired
- 1973-03-13 CH CH366873A patent/CH582707A5/xx not_active IP Right Cessation
- 1973-03-13 CH CH461576A patent/CH582708A5/xx not_active IP Right Cessation
-
1977
- 1977-12-29 JP JP15850177A patent/JPS53101394A/ja active Pending
-
1978
- 1978-05-24 SE SE7805910A patent/SE7805910L/xx unknown
-
1980
- 1980-02-01 JP JP1194780A patent/JPS55105688A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
ATA213973A (de) | 1975-11-15 |
DE2311131C3 (de) | 1982-06-09 |
DK145699B (da) | 1983-01-31 |
JPS49287A (de) | 1974-01-05 |
NL176943C (nl) | 1985-07-01 |
JPS55105688A (en) | 1980-08-13 |
CH582708A5 (de) | 1976-12-15 |
DE2311131B2 (de) | 1979-02-22 |
FR2181811A1 (de) | 1973-12-07 |
FR2181811B1 (de) | 1976-07-02 |
AT331391B (de) | 1976-08-25 |
CH582707A5 (de) | 1976-12-15 |
SE7805910L (sv) | 1978-05-24 |
JPS5526147B2 (de) | 1980-07-11 |
NL7303434A (de) | 1973-09-17 |
SE416811B (sv) | 1981-02-09 |
DE2311131A1 (de) | 1973-10-18 |
AU5321273A (en) | 1974-09-12 |
GB1427139A (en) | 1976-03-10 |
NL176943B (nl) | 1985-02-01 |
JPS53101394A (en) | 1978-09-04 |
DK145699C (da) | 1983-07-25 |
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