CA1006875A - Indole derivatives - Google Patents

Indole derivatives

Info

Publication number: CA1006875A
Authority: CA; Canada
Prior art keywords: indole derivatives; indole; derivatives
Prior art date: 1971-06-01
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

CA143,820A

Other languages

English (en)

Other versions

CA143820S (en

Inventor

Ivo L. Jirkovsky

Thomas A. Dobson

Leslie G. Humber

Christopher A. Demerson

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Wyeth LLC

Original Assignee

American Home Products Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-06-01

Filing date

1972-05-31

Publication date

1977-03-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22527916&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CA1006875(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1972-05-31 Application filed by American Home Products Corp filed Critical American Home Products Corp

1977-03-15 Application granted granted Critical

1977-03-15 Publication of CA1006875A publication Critical patent/CA1006875A/en

Status Expired legal-status Critical Current

Links

229940054051 antipsychotic indole derivative Drugs 0.000 title 1
150000002475 indoles Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/052—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
- H—ELECTRICITY
- H01—ELECTRIC ELEMENTS
- H01L—SEMICONDUCTOR DEVICES NOT COVERED BY CLASS H10
- H01L29/00—Semiconductor devices specially adapted for rectifying, amplifying, oscillating or switching and having potential barriers; Capacitors or resistors having potential barriers, e.g. a PN-junction depletion layer or carrier concentration layer; Details of semiconductor bodies or of electrodes thereof ; Multistep manufacturing processes therefor
- H01L29/66—Types of semiconductor device ; Multistep manufacturing processes therefor
- H01L29/68—Types of semiconductor device ; Multistep manufacturing processes therefor controllable by only the electric current supplied, or only the electric potential applied, to an electrode which does not carry the current to be rectified, amplified or switched
- H01L29/70—Bipolar devices
- H01L29/72—Transistor-type devices, i.e. able to continuously respond to applied control signals
- H01L29/73—Bipolar junction transistors

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Power Engineering (AREA)
Microelectronics & Electronic Packaging (AREA)
Engineering & Computer Science (AREA)
Condensed Matter Physics & Semiconductors (AREA)
General Physics & Mathematics (AREA)
Physics & Mathematics (AREA)
Computer Hardware Design (AREA)
Ceramic Engineering (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

CA143,820A 1971-06-01 1972-05-31 Indole derivatives Expired CA1006875A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US00148895A US3843681A (en)	1971-06-01	1971-06-01	1-carboxamido pyrano(thiopyrano)(3,4-6)indole derivatives

Publications (1)

Publication Number	Publication Date
CA1006875A true CA1006875A (en)	1977-03-15

Family

ID=22527916

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA143,820A Expired CA1006875A (en)	1971-06-01	1972-05-31	Indole derivatives

Country Status (23)

Country	Link
US (1)	US3843681A (de)
JP (1)	JPS5638594B1 (de)
AR (1)	AR198787A1 (de)
AU (1)	AU463079B2 (de)
BE (1)	BE784284A (de)
CA (1)	CA1006875A (de)
CH (1)	CH580101A5 (de)
CS (1)	CS178409B2 (de)
DE (1)	DE2226340A1 (de)
DK (1)	DK155328C (de)
ES (1)	ES403343A1 (de)
FI (1)	FI54125C (de)
FR (1)	FR2140154B1 (de)
GB (1)	GB1391005A (de)
HK (1)	HK13078A (de)
HU (1)	HU169432B (de)
IL (1)	IL39466A (de)
MY (1)	MY7800237A (de)
NL (1)	NL173405C (de)
PH (2)	PH10625A (de)
SE (1)	SE387122B (de)
SU (1)	SU463262A3 (de)
ZA (1)	ZA723344B (de)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3974179A (en) *	1971-06-01	1976-08-10	American Home Products Corporation	1,3,4,9-Tetrahydropyrano[3,4-b]indole-1-acetamides and derivatives
US4118394A (en) *	1976-10-18	1978-10-03	Ayerst, Mckenna & Harrison Limited	Pyrano- and thiopyranoindole derivatives
US4179503A (en) *	1978-05-08	1979-12-18	American Home Products Corp.	1-Hydroxyalkanamine pyrano[3,4-b]indole derivatives
US4309348A (en) *	1979-05-14	1982-01-05	American Home Products Corporation	Tricyclic indole derivatives
US4235903A (en) *	1979-08-06	1980-11-25	American Home Products Corporation	1-Hydroxyalkanamine tetrahydrocarbazoles and cyclopent[b]indoles, compositions and method of use
US4319029A (en) *	1979-08-06	1982-03-09	American Home Products Corporation	Hydroxyalkanamide tetrahydrocarbazoles
JPS58179164A (ja) *	1982-04-10	1983-10-20	Toshiharu Nakai	金属表面処理等に用いられるｓｃｒ整流器の定格直流電圧選定方法並びに定格直流電圧切替方法
US4775690A (en) *	1987-01-13	1988-10-04	American Home Products Corporation	Substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
US4826994A (en) *	1986-03-11	1989-05-02	American Home Products Corporation	Production of substituted 1,3,4,9-tetrahydropyrano(3,4-B)indole-1-acetic acids
US4670462A (en) *	1986-03-11	1987-06-02	American Home Products Corporation	Substituted 1,3,4,9-tetrahydropyrano(3,4-B)indole-1-acetic acids
US4971960A (en) *	1986-03-11	1990-11-20	American Home Products Corporation	Substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
US4663345A (en) *	1986-04-17	1987-05-05	American Home Products Corporation	Etodolac for treatment of gout
US4686213A (en) *	1986-08-15	1987-08-11	American Home Products Corporation	Substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
US4748252A (en) *	1986-08-15	1988-05-31	American Home Products Corporation	Substituted 1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acids
US4810699A (en) *	1987-02-20	1989-03-07	American Home Products Corporation	Substituted 1,3,4,9-tetrahydropyrano[3,4,-b]indole-1-acetic acids, pharmaceutical compositions containing them, and methods for treating inflammatory conditions and for analgesic purposes using them
US4824961A (en) *	1987-08-27	1989-04-25	American Home Products Corporation	Production of substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
US4897493A (en) *	1987-08-27	1990-01-30	American Home Products Corporation	Production of substituted 1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acids
US4822781A (en) *	1987-10-08	1989-04-18	American Home Products	Substituted-8-alkenyl-1,3,4,9-tetrahydropyrano-[3,4-b]indole-1-acetic acids
US4822893A (en) *	1988-02-08	1989-04-18	American Home Products	Production of substituted 1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acids
US4873257A (en) *	1988-04-21	1989-10-10	American Home Products Corporation	Susbtituted fused tetrahydrocarbazole acetic acid derivatives
CA2131992A1 (en) *	1992-03-13	1993-09-16	James W. Young	Antipyretic and analgesic methods and compositions containing optically pure r-etodolac
IT1288123B1 (it) *	1996-09-04	1998-09-10	Nicox Sa	Uso di nitroderivati per l'incontinenza urinaria
AU742787B2 (en)	1997-07-09	2002-01-10	Androsolutions, Inc.	Improved methods and compositions for treating male erectile dysfunction
US6103765A (en)	1997-07-09	2000-08-15	Androsolutions, Inc.	Methods for treating male erectile dysfunction
PT1104297E (pt) *	1998-07-09	2006-05-31	Cephalon Inc	Composicoes para o tratamento da leucemia linfocitica cronica
US6066741A (en) *	1998-09-08	2000-05-23	A.M.S.A. Anonima Materie Sintetiche & Affini S.P.A.	Process for the preparation of etodolac
IT1308633B1 (it)	1999-03-02	2002-01-09	Nicox Sa	Nitrossiderivati.
US7151100B1 (en)	1999-07-23	2006-12-19	The Regents Of The University Of California	Indole compounds useful for the treatment of cancer
US6545034B1 (en) *	1999-07-23	2003-04-08	The Regents Of The University Of California	Use of etodolac for the treatment of chronic lymphocytic leukemia
US7129262B2 (en) *	1999-07-23	2006-10-31	The Regents Of The University Of California	Indole compounds useful for the treatment of cancer
US7361680B2 (en) *	1999-07-23	2008-04-22	The Regents Of The University Of California	Indole compounds useful for the treatment of cancer
US7105560B1 (en)	1999-07-23	2006-09-12	The Regents Of The University Of California	Use of etodolac in the treatment of multiple myeloma
IT1318673B1 (it) *	2000-08-08	2003-08-27	Nicox Sa	Farmaci per le disfunzioni sessuali.
IT1318674B1 (it) *	2000-08-08	2003-08-27	Nicox Sa	Faramaci per l'incontinenza.
CA2419060A1 (en) *	2000-08-09	2002-02-14	The Regents Of The University Of California	Indole compounds useful for the treatment of cancer
US20040152672A1 (en) *	2000-08-09	2004-08-05	Carson Dennis A.	Indole compounds useful for the treatment of cancer
US6544556B1 (en)	2000-09-11	2003-04-08	Andrx Corporation	Pharmaceutical formulations containing a non-steroidal antiinflammatory drug and a proton pump inhibitor
US7601846B2 (en) *	2001-06-26	2009-10-13	The Regents Of The University Of California	Compounds having activity as inhibitors of apoptosis
US20030232794A1 (en) *	2001-06-26	2003-12-18	Cottam Howard B.	Use of STAT-6 inhibitors as therapeutic agents
JP4625637B2 (ja)	2002-02-22	2011-02-02	シャイアエルエルシー	活性物質送達系及び活性物質を保護し投与する方法
ITMI20020773A1 (it) *	2002-04-11	2003-10-13	Nicox Sa	Farmaci per il trattamento dell'artrite
TW200400818A (en)	2002-05-21	2004-01-16	Wyeth Corp	Method for the use of pyranoindole derivatives to treat infection with hepatitis C virus
TW200400963A (en)	2002-05-21	2004-01-16	Wyeth Corp	R-enantiomers of pyranoindole derivatives and the use thereof for the treatment of hepatitis C virus infection or disease
AU2003295336A1 (en) *	2002-09-19	2004-04-08	Dennis A. Carson	Use of etodoclac to treat hyperplasia
DE10252667A1 (de) *	2002-11-11	2004-05-27	Grünenthal GmbH	Spirocyclische Cyclohexan-Derivate
TW200526668A (en) *	2003-10-02	2005-08-16	Salmedix Inc	Substituted indole derivatives
CA2573508A1 (en) *	2004-09-10	2006-03-23	Wyeth	Process for the scalable synthesis of 1, 3, 4, 9-tetrahydropyrano[3, 4-b]-indole derivatives
EP1683521A1 (de) *	2005-01-21	2006-07-26	Centre National De La Recherche Scientifique (Cnrs)	Peptid-Deformylase-Inhibitoren, deren Verwendung und pharmazeutische Zusammensetzungen, welche sie enthalten
CA2657606A1 (en)	2006-03-08	2007-09-13	Cortria Corporation	Combination therapy with non-selective cox inhibitors to prevent cox-related gastric injuries
KR20210099206A (ko) *	2008-07-23	2021-08-11	아레나 파마슈티칼스, 인크.	자가면역성 및 염증성의 장애의 치료에 유용한 치환된 1,2,3,4-테트라히드로시클로펜타[ｂ]인돌-3-일)아세트산 유도체

1971
- 1971-06-01 US US00148895A patent/US3843681A/en not_active Expired - Lifetime
1972
- 1972-05-16 ZA ZA723344A patent/ZA723344B/xx unknown
- 1972-05-17 IL IL39466A patent/IL39466A/xx unknown
- 1972-05-22 AU AU42554/72A patent/AU463079B2/en not_active Ceased
- 1972-05-24 PH PH13564A patent/PH10625A/en unknown
- 1972-05-30 DE DE2226340A patent/DE2226340A1/de active Granted
- 1972-05-30 FI FI1511/72A patent/FI54125C/fi active
- 1972-05-31 CS CS3759A patent/CS178409B2/cs unknown
- 1972-05-31 SU SU1792255A patent/SU463262A3/ru active
- 1972-05-31 SE SE7207142A patent/SE387122B/xx unknown
- 1972-05-31 DK DK271972A patent/DK155328C/da not_active IP Right Cessation
- 1972-05-31 CA CA143,820A patent/CA1006875A/en not_active Expired
- 1972-05-31 AR AR242297A patent/AR198787A1/es active
- 1972-05-31 ES ES403343A patent/ES403343A1/es not_active Expired
- 1972-06-01 BE BE784284A patent/BE784284A/xx not_active IP Right Cessation
- 1972-06-01 CH CH813372A patent/CH580101A5/xx not_active IP Right Cessation
- 1972-06-01 HU HUAE361A patent/HU169432B/hu unknown
- 1972-06-01 JP JP5474472A patent/JPS5638594B1/ja active Pending
- 1972-06-01 GB GB2560572A patent/GB1391005A/en not_active Expired
- 1972-06-01 NL NLAANVRAGE7207408,A patent/NL173405C/xx not_active IP Right Cessation
- 1972-06-01 FR FR7219699A patent/FR2140154B1/fr not_active Expired
1975
- 1975-03-24 PH PH16956A patent/PH11673A/en unknown
1978
- 1978-03-09 HK HK130/78A patent/HK13078A/xx unknown
- 1978-12-30 MY MY237/78A patent/MY7800237A/xx unknown

Also Published As

Publication number	Publication date
NL173405C (nl)	1984-01-16
ES403343A1 (es)	1975-04-16
AU4255472A (en)	1973-11-29
GB1391005A (en)	1975-04-16
AU463079B2 (en)	1975-07-17
IL39466A (en)	1975-05-22
DK155328B (da)	1989-03-28
DE2226340A1 (de)	1973-03-15
IL39466A0 (en)	1972-07-26
DE2226340C2 (de)	1987-07-16
AR198787A1 (es)	1974-07-24
CS178409B2 (de)	1977-09-15
FR2140154B1 (de)	1976-04-16
US3843681A (en)	1974-10-22
HU169432B (de)	1976-11-28
MY7800237A (en)	1978-12-31
BE784284A (fr)	1972-12-01
FI54125B (fi)	1978-06-30
ZA723344B (en)	1973-12-19
FI54125C (fi)	1978-10-10
SE387122B (sv)	1976-08-30
NL7207408A (de)	1972-12-05
CH580101A5 (de)	1976-09-30
HK13078A (en)	1978-03-17
FR2140154A1 (de)	1973-01-12
SU463262A3 (ru)	1975-03-05
JPS5638594B1 (de)	1981-09-08
DK155328C (da)	1989-09-18
PH10625A (en)	1977-07-21
PH11673A (en)	1978-05-19

Publication	Publication Date	Title
AU463079B2 (en)	1975-07-17	Indole derivatives
CA983932A (en)	1976-02-17	Indole derivatives
AU468250B2 (en)	1976-01-08	3-nitropyrazole derivatives
AU462723B2 (en)	1975-07-03	2-nitro-5-imidazolyaldehyde derivatives
CA1012150A (en)	1977-06-14	Indole derivatives
AU461957B2 (en)	1975-06-12	Lumilysergol derivatives
CA1017335A (en)	1977-09-13	Triazolyl-ethenyl-phenylene derivatives
AU463679B2 (en)	1975-07-31	Dibenzocycloheptadioxolan derivatives
AU472069B2 (en)	1976-05-13	Dibenzoxirenazepine derivatives
AU470552B2 (en)	1976-03-18	Aminocephalosporin derivatives
GB1405800A (en)	1975-09-10	Indole derivatives
CA882140A (en)	1971-09-28	Indole derivatives
CA878514A (en)	1971-08-17	Indole derivatives
CA876724A (en)	1971-07-27	Indole derivatives
CA861515A (en)	1971-01-19	Indole derivatives
AU464145B2 (en)	1975-08-14	Indole derivatives
AU438840B2 (en)	1972-11-23	Indole derivatives
CA973882A (en)	1975-09-02	Indoles
CA866825A (en)	1971-03-23	2-benzoyl-3-(2-tertiaryamino-ethoxy)-indole derivatives
AU2912871A (en)	1972-11-23	Indole derivatives
CA877321A (en)	1971-08-03	Ndole derivatives
CA882717A (en)	1971-10-05	Indole alkaloid derivatives
AU450164B2 (en)	1974-07-04	Thienobenzothiazepine derivatives
AU458249B2 (en)	1972-12-07	Tropan-3-ol derivatives
CA862773A (en)	1971-02-02	N-phenylsuccinimide derivatives