BRPI1011959A2 - compostos de cetolídeo tendo atividade antimicrobiana. - Google Patents

compostos de cetolídeo tendo atividade antimicrobiana.

Info

Publication number
BRPI1011959A2
BRPI1011959A2 BRPI1011959A BRPI1011959A BRPI1011959A2 BR PI1011959 A2 BRPI1011959 A2 BR PI1011959A2 BR PI1011959 A BRPI1011959 A BR PI1011959A BR PI1011959 A BRPI1011959 A BR PI1011959A BR PI1011959 A2 BRPI1011959 A2 BR PI1011959A2
Authority
BR
Brazil
Prior art keywords
antimicrobial activity
ketolide compounds
ketolide
compounds
antimicrobial
Prior art date
Application number
BRPI1011959A
Other languages
English (en)
Inventor
Bharat Kalidas Trivedi
Mahesh Vithalbhai Patel
Original Assignee
Wockhardt Research Center
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wockhardt Research Center filed Critical Wockhardt Research Center
Publication of BRPI1011959A2 publication Critical patent/BRPI1011959A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
BRPI1011959A 2009-05-27 2010-05-26 compostos de cetolídeo tendo atividade antimicrobiana. BRPI1011959A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1307MU2009 2009-05-27
PCT/IB2010/052325 WO2010136971A1 (en) 2009-05-27 2010-05-26 Ketolide compounds having antimicrobial activity

Publications (1)

Publication Number Publication Date
BRPI1011959A2 true BRPI1011959A2 (pt) 2016-04-26

Family

ID=42731985

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1011959A BRPI1011959A2 (pt) 2009-05-27 2010-05-26 compostos de cetolídeo tendo atividade antimicrobiana.

Country Status (14)

Country Link
US (1) US8541420B2 (pt)
EP (1) EP2435460B1 (pt)
JP (1) JP5607149B2 (pt)
KR (1) KR101566053B1 (pt)
CN (1) CN102459296B (pt)
AU (1) AU2010252641B2 (pt)
BR (1) BRPI1011959A2 (pt)
CA (1) CA2763246C (pt)
ES (1) ES2561332T3 (pt)
MX (1) MX2011012614A (pt)
NZ (1) NZ596628A (pt)
RU (1) RU2011153353A (pt)
WO (1) WO2010136971A1 (pt)
ZA (1) ZA201108844B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2673285B1 (en) * 2010-12-09 2017-07-19 Wockhardt Limited Ketolide compounds
CA2830861C (en) * 2011-03-22 2017-01-24 Wockhardt Limited Process for preparation of ketolide compounds
ITMI20130444A1 (it) * 2013-03-22 2014-09-23 S B M Science Of Biology In Medici Ne Srl Composto di inclusione comprendente adjudin [1-(2,4-diclorobenzil) - 1h-indazolo-3-carboidrazide] e ciclodestrina, sua preparazione e utilizzo.
EP3004094B1 (de) 2013-06-04 2017-03-01 Bayer Pharma Aktiengesellschaft 3-aryl-substituierte imidazo[1,2-a]pyridine und ihre verwendung
CN106459090A (zh) 2014-02-19 2017-02-22 拜耳制药股份公司 3‑(嘧啶‑2‑基)咪唑并[1,2‑a]吡啶
US20170027917A1 (en) * 2014-04-18 2017-02-02 Wockhardt Limited Pharmaceutical compositions comprising antibacterial agents
EP3227287B1 (de) 2014-12-02 2019-08-07 Bayer Pharma Aktiengesellschaft Heteroaryl-substituierte imidazo[1,2-a]pyridine und ihre verwendung
CN108778254B (zh) * 2016-01-12 2020-09-04 沃克哈特有限公司 药物组合物
RU2018129198A (ru) * 2016-01-12 2020-02-13 Вокхардт Лимитед Фармацевтические композиции
RU2018129197A (ru) * 2016-01-12 2020-02-13 Вокхардт Лимитед Фармацевтические композиции для лечения бактериальных инфекций
WO2018167675A1 (en) * 2017-03-16 2018-09-20 Wockhardt Limited A process for preparing ketolide compounds

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2719587B1 (fr) 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
WO1998009978A1 (en) 1996-09-04 1998-03-12 Abbott Laboratories 6-o-substituted ketolides having antibacterial activity
CO4990960A1 (es) * 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
ES2199524T3 (es) * 1998-04-24 2004-02-16 Pfizer Products Inc. Derivados 9a,11b-deshidro de 9-oxima-3-ceto-6-o-metileritromicina.
KR100502031B1 (ko) * 2000-08-22 2005-07-25 바실리어 파마슈티카 아게 항균 활성을 갖는 신규한 매크롤라이드
NZ526450A (en) 2000-12-21 2005-04-29 Pliva Istrazivacki Inst D Macrolide antibiotics
GB0031312D0 (en) 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
GB0127349D0 (en) 2001-11-14 2002-01-02 Glaxo Group Ltd Macrolides
US6995143B2 (en) 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
US6727229B2 (en) 2002-08-19 2004-04-27 Enanta Pharmaceuticals, Inc. 11,12-substituted lactone ketolide derivatives having antibacterial activity
US7163924B2 (en) * 2003-04-25 2007-01-16 Chiron Corporation Ketolide derivatives
EP1846430B1 (en) * 2005-02-09 2009-04-01 Basilea Pharmaceutica AG New macrolides
KR20090042971A (ko) 2006-08-24 2009-05-04 욱크하르트 리서치 센터 항미생물 활성을 갖는 신규한 마크로라이드 및 케토라이드

Also Published As

Publication number Publication date
EP2435460A1 (en) 2012-04-04
EP2435460B1 (en) 2015-01-07
JP5607149B2 (ja) 2014-10-15
CA2763246A1 (en) 2010-12-02
MX2011012614A (es) 2012-02-22
KR20120037916A (ko) 2012-04-20
CN102459296A (zh) 2012-05-16
US8541420B2 (en) 2013-09-24
ES2561332T3 (es) 2016-02-25
CA2763246C (en) 2013-10-29
NZ596628A (en) 2013-03-28
RU2011153353A (ru) 2013-07-10
AU2010252641A1 (en) 2011-12-15
CN102459296B (zh) 2014-10-29
US20120142710A1 (en) 2012-06-07
JP2012528142A (ja) 2012-11-12
ZA201108844B (en) 2013-02-27
AU2010252641B2 (en) 2015-09-17
WO2010136971A1 (en) 2010-12-02
KR101566053B1 (ko) 2015-11-04

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07E Notice of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06T Formal requirements before examination [chapter 6.20 patent gazette]
B11E Dismissal acc. art. 34 of ipl - requirements for examination incomplete
B11T Dismissal: dismissal of application maintained