BRPI1010024A2 - derivados de aminopirrolidinona e uso dos mesmos - Google Patents
derivados de aminopirrolidinona e uso dos mesmosInfo
- Publication number
- BRPI1010024A2 BRPI1010024A2 BRPI1010024A BRPI1010024A BRPI1010024A2 BR PI1010024 A2 BRPI1010024 A2 BR PI1010024A2 BR PI1010024 A BRPI1010024 A BR PI1010024A BR PI1010024 A BRPI1010024 A BR PI1010024A BR PI1010024 A2 BRPI1010024 A2 BR PI1010024A2
- Authority
- BR
- Brazil
- Prior art keywords
- aminopyrrolidinone
- derivatives
- aminopyrrolidinone derivatives
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18438609P | 2009-06-05 | 2009-06-05 | |
| US29502310P | 2010-01-14 | 2010-01-14 | |
| PCT/US2010/037582 WO2010141932A1 (en) | 2009-06-05 | 2010-06-07 | Aminopyrrolidinone derivatives and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI1010024A2 true BRPI1010024A2 (pt) | 2019-09-24 |
Family
ID=42635266
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI1010024A BRPI1010024A2 (pt) | 2009-06-05 | 2010-06-07 | derivados de aminopirrolidinona e uso dos mesmos |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8252829B2 (pt) |
| EP (1) | EP2438059A1 (pt) |
| JP (1) | JP2012529432A (pt) |
| CN (1) | CN102548986A (pt) |
| AU (1) | AU2010256360A1 (pt) |
| BR (1) | BRPI1010024A2 (pt) |
| CA (1) | CA2764387A1 (pt) |
| IL (1) | IL216768A0 (pt) |
| MX (1) | MX2011013016A (pt) |
| SG (1) | SG176628A1 (pt) |
| WO (1) | WO2010141932A1 (pt) |
| ZA (1) | ZA201109034B (pt) |
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| RU2011150248A (ru) * | 2009-05-11 | 2013-06-20 | Энвиво Фармасьютикалз, Инк. | Лечение когнитивных расстройств с определенными рецепторами альфа-7 никотиновой кислоты в комбинации с ингибиторами ацетилхолинэстеразы |
| US8834874B2 (en) | 2009-10-09 | 2014-09-16 | Armagen Technologies, Inc. | Methods and compositions for increasing iduronate 2-sulfatase activity in the CNS |
| PT3029039T (pt) | 2010-05-17 | 2017-11-28 | Forum Pharmaceuticals Inc | Formulações farmacêuticas que compreendem formas cristalinas de cloridrato de (r)-7-cloro-n-(quinuclidin-3-il)benzo(b)tiofeno-2-carboxamida mono-hidratado |
| KR20150013476A (ko) * | 2012-04-04 | 2015-02-05 | 아이백스 인터내셔널 게엠베하 | 조합요법용 약학적 조성물 |
| CA2872005A1 (en) | 2012-05-08 | 2013-11-14 | Forum Pharmaceuticals, Inc. | Methods of maintaining, treating or improving cognitive function |
| EP2861263B1 (en) * | 2012-06-19 | 2017-12-06 | University of Florida Research Foundation, Inc. | Compositions and methods for treating diabetes |
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| JP6958860B2 (ja) * | 2017-11-07 | 2021-11-02 | 学校法人自治医科大学 | ミトコンドリアの機能障害の改善剤、及びミトコンドリアの機能障害に起因する疾患又は症状の予防又は治療薬、並びにそれらの用途 |
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| CN112945913A (zh) * | 2019-12-10 | 2021-06-11 | 中国科学院大连化学物理研究所 | 一种萘酰亚胺类荧光探针在脂滴成像领域中的应用 |
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| US8907095B2 (en) | 2007-10-22 | 2014-12-09 | Merck Sharp & Dohme Corp. | Bicyclic heterocycle derivatives and their use as modulators of the activity of GPR119 |
| JP5544296B2 (ja) | 2007-11-16 | 2014-07-09 | ライジェル ファーマシューティカルズ， インコーポレイテッド | 代謝障害のためのカルボキサミド、スルホンアミド、およびアミン化合物 |
| US20100298372A1 (en) | 2007-12-11 | 2010-11-25 | Schering Corporation | Gamma secretase modulators |
| TWI447099B (zh) | 2008-01-29 | 2014-08-01 | Nissan Chemical Ind Ltd | Aryl sulfonic acid compounds and the use of electron acceptables |
| KR101331032B1 (ko) | 2008-07-30 | 2013-11-19 | 삼성전자주식회사 | 가상화 환경과 결합된 어플리케이션 실행 방법 |
| EP2237405B1 (en) | 2009-03-31 | 2013-02-20 | STMicroelectronics Srl | Control device for the change of the driving modality of an electromagnetic load |
| US8473905B1 (en) | 2009-09-30 | 2013-06-25 | Emc Corporation | Managing user interface characteristics in displaying data storage systems information |
| JP5646195B2 (ja) | 2010-03-30 | 2014-12-24 | 富士フイルム株式会社 | インクジェット記録装置及び断熱処理方法 |
| TWI437908B (zh) | 2011-05-17 | 2014-05-11 | Leadtrend Tech Corp | 具電流平衡功能的驅動電路 |
-
2010
- 2010-06-07 US US12/795,065 patent/US8252829B2/en not_active Expired - Fee Related
- 2010-06-07 AU AU2010256360A patent/AU2010256360A1/en not_active Abandoned
- 2010-06-07 CN CN2010800350077A patent/CN102548986A/zh active Pending
- 2010-06-07 BR BRPI1010024A patent/BRPI1010024A2/pt not_active IP Right Cessation
- 2010-06-07 CA CA2764387A patent/CA2764387A1/en not_active Abandoned
- 2010-06-07 WO PCT/US2010/037582 patent/WO2010141932A1/en active Application Filing
- 2010-06-07 SG SG2011089018A patent/SG176628A1/en unknown
- 2010-06-07 JP JP2012514220A patent/JP2012529432A/ja not_active Withdrawn
- 2010-06-07 MX MX2011013016A patent/MX2011013016A/es not_active Application Discontinuation
- 2010-06-07 EP EP10724958A patent/EP2438059A1/en not_active Withdrawn
-
2011
- 2011-12-04 IL IL216768A patent/IL216768A0/en unknown
- 2011-12-08 ZA ZA2011/09034A patent/ZA201109034B/en unknown
-
2012
- 2012-07-13 US US13/548,363 patent/US20130289086A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20130289086A1 (en) | 2013-10-31 |
| MX2011013016A (es) | 2012-04-20 |
| WO2010141932A1 (en) | 2010-12-09 |
| EP2438059A1 (en) | 2012-04-11 |
| AU2010256360A1 (en) | 2012-01-12 |
| ZA201109034B (en) | 2013-02-27 |
| US8252829B2 (en) | 2012-08-28 |
| JP2012529432A (ja) | 2012-11-22 |
| CN102548986A (zh) | 2012-07-04 |
| SG176628A1 (en) | 2012-01-30 |
| IL216768A0 (en) | 2012-02-29 |
| US20110021590A1 (en) | 2011-01-27 |
| CA2764387A1 (en) | 2010-12-09 |
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| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |