BRPI0415525A - derivados de imidazola e seu uso como agentes farmacêuticos - Google Patents
derivados de imidazola e seu uso como agentes farmacêuticosInfo
- Publication number
- BRPI0415525A BRPI0415525A BRPI0415525-4A BRPI0415525A BRPI0415525A BR PI0415525 A BRPI0415525 A BR PI0415525A BR PI0415525 A BRPI0415525 A BR PI0415525A BR PI0415525 A BRPI0415525 A BR PI0415525A
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical agents
- imidazole derivatives
- cancer
- compounds
- treatment
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Abstract
"DERIVADOS DE IMIDAZOLA E SEU USO COMO AGENTES FARMACêUTICOS". Compostos da fórmula geral (I): são produtos terapêuticos valiosos para o tratamento de câncer e doenças relacionadas ao câncer.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP03023677 | 2003-10-17 | ||
PCT/EP2004/011598 WO2005040154A1 (en) | 2003-10-17 | 2004-10-15 | Novel imidazole derivatives and their use as pharmaceutical agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0415525A true BRPI0415525A (pt) | 2006-12-26 |
Family
ID=34486074
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0415525-4A BRPI0415525A (pt) | 2003-10-17 | 2004-10-15 | derivados de imidazola e seu uso como agentes farmacêuticos |
Country Status (16)
Country | Link |
---|---|
US (1) | US7169781B2 (pt) |
EP (1) | EP1678163B1 (pt) |
JP (1) | JP2007508344A (pt) |
KR (1) | KR100796971B1 (pt) |
CN (1) | CN1867563A (pt) |
AR (1) | AR046286A1 (pt) |
AT (1) | ATE420084T1 (pt) |
AU (1) | AU2004283845A1 (pt) |
BR (1) | BRPI0415525A (pt) |
CA (1) | CA2538134A1 (pt) |
DE (1) | DE602004018962D1 (pt) |
ES (1) | ES2317030T3 (pt) |
MX (1) | MXPA06003698A (pt) |
RU (1) | RU2006116628A (pt) |
TW (1) | TW200528447A (pt) |
WO (1) | WO2005040154A1 (pt) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT1889836E (pt) | 2005-08-24 | 2013-08-28 | Eisai R&D Man Co Ltd | Novo derivado de piridina e derivado de pirimidina (3) |
ATE453635T1 (de) * | 2006-03-22 | 2010-01-15 | Vertex Pharma | C-met-proteinkinasehemmer zur behandlung proliferativer erkrankungen |
AU2007261440A1 (en) * | 2006-06-22 | 2007-12-27 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
WO2008021781A1 (en) | 2006-08-07 | 2008-02-21 | Incyte Corporation | Triazolotriazines as kinase inhibitors |
ES2375284T3 (es) | 2006-08-23 | 2012-02-28 | Eisai R&D Management Co., Ltd. | Sal de un derivado de fenoxipiridina, o cristal de la misma, y procedimiento de producción de la misma. |
US7790885B2 (en) | 2006-08-31 | 2010-09-07 | Eisai R&D Management Co., Ltd. | Process for preparing phenoxypyridine derivatives |
US8148391B2 (en) | 2006-10-23 | 2012-04-03 | Cephalon, Inc. | Fused bicyclic derivatives of 2,4-diaminopyrimidine as ALK and c-Met inhibitors |
ES2689444T3 (es) | 2006-11-22 | 2018-11-14 | Incyte Holdings Corporation | Imidazotriazinas e imidazopirimidinas como inhibidores de la quinasa |
MX2009011810A (es) * | 2007-05-02 | 2010-01-14 | Vertex Pharma | Tiazoles y pirazoles utiles como inhibidores de cinasa. |
MX2009012719A (es) * | 2007-05-24 | 2010-02-04 | Vertex Pharma | Tiazoles y pirazoles utiles como inhibidores de cinasa. |
MX2010003563A (es) * | 2007-10-03 | 2010-06-02 | Vertex Pharma | Inhibidores de proteina cinasa de c-met. |
JP2009132660A (ja) | 2007-11-30 | 2009-06-18 | Eisai R & D Management Co Ltd | 食道癌治療用組成物 |
CN102007124B (zh) | 2008-02-15 | 2014-06-18 | 里格尔制药公司 | 嘧啶-2-胺化合物及其作为jak激酶抑制剂的用途 |
SI2300455T1 (sl) | 2008-05-21 | 2017-12-29 | Incyte Holdings Corporation | Soli 2-fluoro-n-metil-4-(7-(kinolin-6-il-metil)-imidazo(1,2-b)1,2,4) triazin-2-il)benzamid in postopki v zvezi z njihovo pripravo |
BR112012019302B1 (pt) | 2010-02-03 | 2022-06-21 | Incyte Holdings Corporation | Imidazo[1,2-b] [1,2,4]triazinas como inibidores de c-met, composição que as compreende e métodos in vitro de inibir a atividade de c-met cinase, de inibir a via de sinalização da hgf/c-met cinase em uma célula e de inibir a atividade proliferativa de uma célula |
AU2013280644B2 (en) | 2012-06-26 | 2018-08-02 | Jeffrey A. BACHA | Methods for treating tyrosine-kinase-inhibitor-resistant malignancies in patients with genetic polymorphisms or AHI1 dysregulations or mutations employing dianhydrogalactitol, diacetyldianhydrogalactitol, dibromodulcitol, or analogs or derivatives thereof |
CA2892045C (en) | 2012-11-21 | 2022-05-31 | Ptc Therapeutics, Inc. | Substituted reverse pyrimidine bmi-1 inhibitors |
NZ748260A (en) | 2013-08-30 | 2020-01-31 | Ptc Therapeutics Inc | Substituted pyrimidine bmi-1 inhibitors |
US10584115B2 (en) | 2013-11-21 | 2020-03-10 | Ptc Therapeutics, Inc. | Substituted pyridine and pyrazine BMI-1 inhibitors |
KR102030886B1 (ko) * | 2016-09-23 | 2019-10-10 | 재단법인 대구경북첨단의료산업진흥재단 | 신규한 이미다졸일 피리미딘 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 암의 예방 또는 치료용 약학적 조성물 |
US11066404B2 (en) | 2018-10-11 | 2021-07-20 | Incyte Corporation | Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors |
WO2020168197A1 (en) | 2019-02-15 | 2020-08-20 | Incyte Corporation | Pyrrolo[2,3-d]pyrimidinone compounds as cdk2 inhibitors |
TW202100520A (zh) | 2019-03-05 | 2021-01-01 | 美商英塞特公司 | 作為cdk2 抑制劑之吡唑基嘧啶基胺化合物 |
US11919904B2 (en) | 2019-03-29 | 2024-03-05 | Incyte Corporation | Sulfonylamide compounds as CDK2 inhibitors |
US11447494B2 (en) | 2019-05-01 | 2022-09-20 | Incyte Corporation | Tricyclic amine compounds as CDK2 inhibitors |
US11440914B2 (en) | 2019-05-01 | 2022-09-13 | Incyte Corporation | Tricyclic amine compounds as CDK2 inhibitors |
MX2022001940A (es) | 2019-08-14 | 2022-05-10 | Incyte Corp | Compuestos de imidazolil pirimidinilamina como inhibidores de cdk2. |
PE20221905A1 (es) | 2019-10-11 | 2022-12-23 | Incyte Corp | Aminas biciclicas como inhibidoras de la cdk2 |
US11976073B2 (en) | 2021-12-10 | 2024-05-07 | Incyte Corporation | Bicyclic amines as CDK2 inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5656644A (en) | 1994-07-20 | 1997-08-12 | Smithkline Beecham Corporation | Pyridyl imidazoles |
WO1996018626A1 (en) | 1994-12-13 | 1996-06-20 | F. Hoffmann-La Roche Ag | Imidazole derivatives as protein kinase inhibitors in particular egf-r tyrosine kinase |
EP0994870A4 (en) | 1997-06-19 | 2002-10-23 | Smithkline Beecham | NEW IMIDAZOLE COMPOUNDS SUBSTITUTED BY AN ARYLOXYREST |
US6790852B2 (en) | 2002-04-18 | 2004-09-14 | Hoffmann-La Roche Inc. | 2-(2,6-dichlorophenyl)-diarylimidazoles |
-
2004
- 2004-10-12 US US10/961,907 patent/US7169781B2/en not_active Expired - Fee Related
- 2004-10-14 AR ARP040103728A patent/AR046286A1/es unknown
- 2004-10-14 TW TW093131229A patent/TW200528447A/zh unknown
- 2004-10-15 CA CA002538134A patent/CA2538134A1/en not_active Abandoned
- 2004-10-15 JP JP2006534696A patent/JP2007508344A/ja active Pending
- 2004-10-15 WO PCT/EP2004/011598 patent/WO2005040154A1/en active Application Filing
- 2004-10-15 AT AT04765966T patent/ATE420084T1/de not_active IP Right Cessation
- 2004-10-15 CN CNA2004800305837A patent/CN1867563A/zh active Pending
- 2004-10-15 MX MXPA06003698A patent/MXPA06003698A/es active IP Right Grant
- 2004-10-15 BR BRPI0415525-4A patent/BRPI0415525A/pt not_active IP Right Cessation
- 2004-10-15 KR KR1020067007335A patent/KR100796971B1/ko not_active IP Right Cessation
- 2004-10-15 ES ES04765966T patent/ES2317030T3/es active Active
- 2004-10-15 DE DE602004018962T patent/DE602004018962D1/de active Active
- 2004-10-15 AU AU2004283845A patent/AU2004283845A1/en not_active Abandoned
- 2004-10-15 EP EP04765966A patent/EP1678163B1/en not_active Not-in-force
- 2004-10-15 RU RU2006116628/04A patent/RU2006116628A/ru not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
ES2317030T3 (es) | 2009-04-16 |
TW200528447A (en) | 2005-09-01 |
ATE420084T1 (de) | 2009-01-15 |
KR20060063985A (ko) | 2006-06-12 |
AR046286A1 (es) | 2005-11-30 |
MXPA06003698A (es) | 2006-06-05 |
WO2005040154A1 (en) | 2005-05-06 |
JP2007508344A (ja) | 2007-04-05 |
CN1867563A (zh) | 2006-11-22 |
KR100796971B1 (ko) | 2008-01-22 |
US20050113342A1 (en) | 2005-05-26 |
EP1678163A1 (en) | 2006-07-12 |
CA2538134A1 (en) | 2005-05-06 |
RU2006116628A (ru) | 2007-11-27 |
DE602004018962D1 (de) | 2009-02-26 |
AU2004283845A1 (en) | 2005-05-06 |
EP1678163B1 (en) | 2009-01-07 |
US7169781B2 (en) | 2007-01-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012. |