BRPI0414471A - nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona - Google Patents

nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona

Info

Publication number
BRPI0414471A
BRPI0414471A BRPI0414471-6A BRPI0414471A BRPI0414471A BR PI0414471 A BRPI0414471 A BR PI0414471A BR PI0414471 A BRPI0414471 A BR PI0414471A BR PI0414471 A BRPI0414471 A BR PI0414471A
Authority
BR
Brazil
Prior art keywords
formulation containing
pharmaceutical formulation
new pharmaceutical
thiazolidinedione derivative
containing biguanide
Prior art date
Application number
BRPI0414471-6A
Other languages
English (en)
Inventor
Unchalee Kositprapa
Robert I Goldfarb
John Cardinal
Avinash Nangia
Original Assignee
Andrx Labs Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34520446&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0414471(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Andrx Labs Llc filed Critical Andrx Labs Llc
Publication of BRPI0414471A publication Critical patent/BRPI0414471A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

"NOVA FORMULAçãO FARMACêUTICA CONTENDO BIGUANIDA E UM DERIVADO DE TIAZOLIDINADIONA". Uma forma de dosagem farmacêutica compreendendo um componente de liberação controlada compreendendo uma droga antihiperglicêmica em combinação com um segundo componente compreendendo um derivado de tiazolidinadiona é aqui divulgada e descrita.
BRPI0414471-6A 2003-09-19 2004-02-12 nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona BRPI0414471A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/664,803 US7785627B2 (en) 2002-09-20 2003-09-19 Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
PCT/US2004/004112 WO2005039540A1 (en) 2003-09-19 2004-02-12 Novel pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative

Publications (1)

Publication Number Publication Date
BRPI0414471A true BRPI0414471A (pt) 2006-11-14

Family

ID=34520446

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0414471-6A BRPI0414471A (pt) 2003-09-19 2004-02-12 nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona

Country Status (11)

Country Link
US (2) US7785627B2 (pt)
EP (1) EP1663170B1 (pt)
JP (3) JP4718465B2 (pt)
KR (2) KR20060076299A (pt)
CN (2) CN1852703A (pt)
AU (2) AU2004283059B2 (pt)
BR (1) BRPI0414471A (pt)
CA (1) CA2537665C (pt)
ES (1) ES2541124T3 (pt)
NZ (2) NZ580804A (pt)
WO (1) WO2005039540A1 (pt)

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US9060941B2 (en) * 2002-09-20 2015-06-23 Actavis, Inc. Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
US7976853B2 (en) 2003-01-29 2011-07-12 Takeda Pharmaceutical Company Limited Process for producing coated preparation
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NZ580804A (en) 2011-02-25
CA2537665A1 (en) 2005-05-06
EP1663170B1 (en) 2015-06-24
JP2014196314A (ja) 2014-10-16
JP4718465B2 (ja) 2011-07-06
CN101675929A (zh) 2010-03-24
JP2007505903A (ja) 2007-03-15
JP2011148819A (ja) 2011-08-04
EP1663170A1 (en) 2006-06-07
AU2011202162A1 (en) 2011-06-02
WO2005039540A1 (en) 2005-05-06
KR20110126761A (ko) 2011-11-23
CA2537665C (en) 2012-08-14
US7785627B2 (en) 2010-08-31
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AU2004283059B2 (en) 2011-02-10
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EP1663170A4 (en) 2012-01-25
ES2541124T3 (es) 2015-07-16
JP5881962B2 (ja) 2016-03-09
US8309125B2 (en) 2012-11-13
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US20100316708A1 (en) 2010-12-16
US20040106660A1 (en) 2004-06-03

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