BR9913945A - Composição farmacêutica para o tratamento de distúrbios agudos por meio de administração sublingual, e, processo para o tratamento de distúrbios agudos - Google Patents

Composição farmacêutica para o tratamento de distúrbios agudos por meio de administração sublingual, e, processo para o tratamento de distúrbios agudos

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Publication number
BR9913945A
BR9913945A BR9913945-6A BR9913945A BR9913945A BR 9913945 A BR9913945 A BR 9913945A BR 9913945 A BR9913945 A BR 9913945A BR 9913945 A BR9913945 A BR 9913945A
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BR
Brazil
Prior art keywords
treatment
acute disorders
pharmaceutical composition
sublingual administration
composition
Prior art date
Application number
BR9913945-6A
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English (en)
Other versions
BR9913945B1 (pt
BRPI9913945B8 (pt
Inventor
Anders Pettersson
Nyrstr M Christer
Original Assignee
Diabact Ab
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20412702&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9913945(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Diabact Ab filed Critical Diabact Ab
Publication of BR9913945A publication Critical patent/BR9913945A/pt
Publication of BR9913945B1 publication Critical patent/BR9913945B1/pt
Publication of BRPI9913945B8 publication Critical patent/BRPI9913945B8/pt

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/136—Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
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    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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Abstract

"COMPOSIçãO FARMACêUTICA PARA O TRATAMENTO DE DISTúRBIOS AGUDOS POR MEIO DE ADMINISTRAçãO SUBLINGUAL, E, PROCESSO PARA O TRATAMENTO DE DISTúRBIOS AGUDOS". é descrita uma composição farmacêutica para o tratamento de distúrbios agudos. A composição compreende uma mistura ordenada, essencialmente livre de água, de pelo menos um agente farmaceuticamente ativo na forma de micropartículas que são aderidas nas superfícies de partículas portadoras que são substancialmente maiores do que as partículas do agente ativo ou dos agentes ativos, e estão essencialmente livres de água, em combinação com o agente de promotor de mucoadesão e/ou bioadesão. A invenção também refere-se a um processo para a preparação da composição e ao uso da composição para o tratamento de distúrbios agudos.
BRPI9913945A 1998-09-24 1999-09-24 Composição farmacêutica rapidamente atuante para a administração sublingual de um agente farmacêutico para o tratamento de distúrbios agudos BRPI9913945B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9803240A SE9803240D0 (sv) 1998-09-24 1998-09-24 A pharmaceutical composition having a rapid action
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NO20011473L (no) 2001-05-23
LU92636I2 (fr) 2015-03-20
US20140030336A1 (en) 2014-01-30
CA2345121C (en) 2008-06-10
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CY1107711T1 (el) 2013-04-18
RU2193879C1 (ru) 2002-12-10
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HK1148457A1 (en) 2011-09-09
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EP1652518A1 (en) 2006-05-03
DK1115383T3 (da) 2007-07-30
RU2001111025A (ru) 2004-02-20
JP2002526439A (ja) 2002-08-20
AU764346B2 (en) 2003-08-14
KR20010075315A (ko) 2001-08-09
PT2805716T (pt) 2017-12-21
KR100760536B1 (ko) 2007-10-04
CZ20011029A3 (cs) 2001-08-15
CY1115685T1 (el) 2017-01-25
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ES2644770T3 (es) 2017-11-30
ATE365540T1 (de) 2007-07-15

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