BR9904429A - Heterociclos - Google Patents
HeterociclosInfo
- Publication number
- BR9904429A BR9904429A BR9904429-3A BR9904429A BR9904429A BR 9904429 A BR9904429 A BR 9904429A BR 9904429 A BR9904429 A BR 9904429A BR 9904429 A BR9904429 A BR 9904429A
- Authority
- BR
- Brazil
- Prior art keywords
- nso
- alkyl
- preparation
- heterocycles
- halo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
- C07D211/96—Sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Patente de Invenção: <B>"HETEROCICLOS"<D>. A presente invenção refere-se um composto de fórmula ou um seu sal de adição de ácido farmaceuticamente aceitável, em que Ar é fenila substituída por 1 ou 2 substituinte(s) cada qual independentemente escolhido a partir de flúor e cloro; X é NSO~ 2~(C~ 1~-C~ 4~ alquila), NSO~ 2~(halo(C~ 1~-C~ 4~ alquila)) ou O; m é 0 ou 1; n é 1 ou 2; p é 1 ou 2; q é 1 ou 2; e r é 1 ou 2, em conjunto com processos para a preparação de, intermediários usados na preparação de, composições contendo e utilizações de, tais derivados. Os compostos têm atividade antagonista do receptor taquiquinina.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9821898.5A GB9821898D0 (en) | 1998-10-08 | 1998-10-08 | Heterocycles |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9904429A true BR9904429A (pt) | 2000-08-08 |
Family
ID=10840166
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9904429-3A BR9904429A (pt) | 1998-10-08 | 1999-10-08 | Heterociclos |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0992493A1 (pt) |
JP (1) | JP3091844B2 (pt) |
BR (1) | BR9904429A (pt) |
CA (1) | CA2285120A1 (pt) |
GB (1) | GB9821898D0 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9600235D0 (en) * | 1996-01-05 | 1996-03-06 | Pfizer Ltd | Therapeutic agents |
CN102317291B (zh) | 2009-02-13 | 2015-02-11 | 拜耳知识产权有限责任公司 | 稠合嘧啶 |
KR101063877B1 (ko) * | 2009-05-28 | 2011-09-09 | (주)이오알지 | 발차기 운동기구 |
WO2012101013A1 (en) | 2011-01-28 | 2012-08-02 | Boehringer Ingelheim International Gmbh | Substituted pyridinyl-pyrimidines and their use as medicaments |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2676055B1 (fr) * | 1991-05-03 | 1993-09-03 | Sanofi Elf | Composes polycycliques amines et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant. |
ATE177095T1 (de) * | 1994-08-25 | 1999-03-15 | Merrell Pharma Inc | Substituierte piperidine für die behandlung von allergischen krankheiten |
FR2738819B1 (fr) * | 1995-09-14 | 1997-12-05 | Sanofi Sa | Nouveaux composes antagonistes selectifs du recepteur nk3 humain, procede pour leur obtention et compositions pharmaceutiques les contenant |
GB9600235D0 (en) * | 1996-01-05 | 1996-03-06 | Pfizer Ltd | Therapeutic agents |
-
1998
- 1998-10-08 GB GBGB9821898.5A patent/GB9821898D0/en not_active Ceased
-
1999
- 1999-10-04 JP JP11283389A patent/JP3091844B2/ja not_active Expired - Fee Related
- 1999-10-06 EP EP99307878A patent/EP0992493A1/en not_active Withdrawn
- 1999-10-06 CA CA002285120A patent/CA2285120A1/en not_active Abandoned
- 1999-10-08 BR BR9904429-3A patent/BR9904429A/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CA2285120A1 (en) | 2000-04-08 |
EP0992493A1 (en) | 2000-04-12 |
JP2000119251A (ja) | 2000-04-25 |
JP3091844B2 (ja) | 2000-09-25 |
GB9821898D0 (en) | 1998-12-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES555653A0 (es) | Un procedimiento para preparar compuestos imidazoheterociclicos | |
WO2002016381A3 (en) | Composition and method for inhibiting platelet aggregation | |
BR9714787A (pt) | Compostos de 4- fenilpiperidina e processo para sua preparação | |
BR9806778A (pt) | Derivados de benzoìla substuìda por 3-heterociclila e de ácido benzóico substituìdo por 3-heterociclila, composto, composição, processos para a preparação de derivados de benzoìla substituìda por 3-heterociclila e de uma composição, e para controle de vegetação indesejável, e, uso de um derivado de benzoìla substituìda por 3-heterociclila. | |
MX9709951A (es) | Derivados de benzamida y su uso como antagonistas de vasopresina. | |
BR0308146A (pt) | Composto, composição farmacêutica, uso de um composto, e, processo para a preparação de um composto | |
BR9907300A (pt) | Inibidores do fator xa oxoaza-heterociclila substituìdos | |
EP0269574A3 (en) | Novel adenosine derivatives and pharmaceutical compositions containing them as an active ingredient | |
BR0108894A (pt) | Composição farmacêutica, compostos e processo de preparação de compostos | |
BR0111263A (pt) | Derivados de 2-aminocarbonil-9h-purina | |
BRPI0211844B8 (pt) | composto de ácido fenóxi-acético ou um de seus sais farmaceuticamente aceitáveis, e, composição farmacêutica | |
BR9812046A (pt) | Compostos, processos para a preperação do composto e para tratar um paciente humano ou animal, composição farmacêutica, e, uso de um composto | |
DE69420579D1 (de) | 9-HYDROXY-PYRIDO [1,2-a] PYRIMIDIN-4-ON-ETHER-DERIVATE | |
BR9807132A (pt) | Derivados de pirrolidina tendo atividade inibitória de fosfolipase a2 | |
BR0308145A (pt) | Composto, composição farmacêutica, uso de um composto, e, processo para a preparação de um composto | |
IE872329L (en) | New cephem compounds and processes for preparation thereof | |
GR3034769T3 (en) | Triazole antifungal agents. | |
HK1019334A1 (en) | 2-(arylphenyl) amino-imidazoline derivatives | |
BR9904429A (pt) | Heterociclos | |
BR9909086A (pt) | Derivados de piperidinila e n-amidinopiperidinila | |
DK0962457T3 (da) | Piperidoner som tachykininantagonister | |
BR9813613A (pt) | Derivado 3-(benzazol-4-il) pirimidinadiona, uso de um derivado i de 3-(benzazol-4-il) pirimidinadiona ou um sal agriculturalmente útil do mesmo, composição herbicida, processos para a preparação de composições herbicidamente ativas e de controle de vegetação indispensável, ariluréia, arilanilida, e, 2-aminofenol substituìdo, -tiofenol ou -anilina | |
TNSN97092A1 (ar) | مثبطات انزيم بروتيني فلزي وتركيبات صيدلانية تحتوي على تلك المثبتطات واستخدامها الصيدلاني وطرق ومركبات وسيطة مفيدة لتحضير التركيبات المذكورة. | |
BR9813920A (pt) | Trifluorometilbifenilil-dihalofenilazolinas como pesticidas | |
HRP20000027B1 (en) | Process for the preparation of alkoxyfuranoneamine derivatives, compounds obtained by this process, and the use of these compounds |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 5A , 6A , 7A E 8A ANUIDADES. |
|
B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1926 DE 04/12/2007. |