BR6676469D0 - Processo para preparar novos compostos cefalosporinicos tendo atividade antibiotica - Google Patents

Processo para preparar novos compostos cefalosporinicos tendo atividade antibiotica

Info

Publication number
BR6676469D0
BR6676469D0 BR176469/66A BR17646966A BR6676469D0 BR 6676469 D0 BR6676469 D0 BR 6676469D0 BR 176469/66 A BR176469/66 A BR 176469/66A BR 17646966 A BR17646966 A BR 17646966A BR 6676469 D0 BR6676469 D0 BR 6676469D0
Authority
BR
Brazil
Prior art keywords
antibiotic activity
prepare new
cephalosporin compounds
new cephalosporin
compounds
Prior art date
Application number
BR176469/66A
Other languages
English (en)
Inventor
J Spencer
C Ryan
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BR6676469D0 publication Critical patent/BR6676469D0/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/32Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by an araliphatic carboxylic acid, which is substituted on the aliphatic radical by hetero atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
BR176469/66A 1965-03-08 1966-01-17 Processo para preparar novos compostos cefalosporinicos tendo atividade antibiotica BR6676469D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43804665A 1965-03-08 1965-03-08

Publications (1)

Publication Number Publication Date
BR6676469D0 true BR6676469D0 (pt) 1973-09-06

Family

ID=23738987

Family Applications (1)

Application Number Title Priority Date Filing Date
BR176469/66A BR6676469D0 (pt) 1965-03-08 1966-01-17 Processo para preparar novos compostos cefalosporinicos tendo atividade antibiotica

Country Status (10)

Country Link
US (1) US3518260A (pt)
BE (1) BE675298A (pt)
BR (1) BR6676469D0 (pt)
CH (1) CH480368A (pt)
CY (1) CY527A (pt)
DE (1) DE1670600A1 (pt)
DK (1) DK140943B (pt)
GB (1) GB1123333A (pt)
NL (1) NL6600636A (pt)
SE (1) SE354663B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4123611A (en) * 1970-10-21 1978-10-31 President Of Osaka University N-protected amino compounds
YU39709B (en) * 1972-09-15 1985-04-30 Bristol Myers Co Process for producing cephalosporin
GB1438872A (en) * 1972-11-17 1976-06-09 Fujisawa Pharmaceutical Co 7-beta-aminoacylamino-3-substituted-3-cephem-4-carboxylic acid derivatives and preparation thereof
US3880846A (en) * 1972-12-19 1975-04-29 Squibb & Sons Inc Vinylaminoacetyl cephalosporins
FR2265391B1 (pt) * 1974-04-02 1978-11-03 Isf Spa
AT342197B (de) * 1975-02-20 1978-03-28 Ciba Geigy Ag Neues verfahren zur herstellung von 3-cephemverbindungen
US4474780A (en) * 1983-07-22 1984-10-02 Eli Lilly And Company Crystalline cephalosporin
US4490370A (en) * 1983-04-12 1984-12-25 Eli Lilly And Company Naphthylglycyl cephalosporin derivatives
US4492694A (en) * 1983-04-12 1985-01-08 Eli Lilly And Company Indolylglycyl cephalosporin derivatives
HU207285B (en) * 1989-07-27 1993-03-29 Chinoin Gyogyszer Es Vegyeszet Process for producing n-substituted phenyl-glycine derivatives
HU208110B (en) * 1989-07-27 1993-08-30 Chinoin Gyogyszer Es Vegyeszet Process for producing phenylglycine derivatives
US5908929A (en) * 1996-12-05 1999-06-01 Vitara Chemicals Limited Process for the manufacture of the antibiotic 7-(D-α-amino-α-phenylacetamido)-3-methyl-3-cephem-4-carboxylic acid (cephalexin) and pharmaceutically acceptable salts thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3252973A (en) * 1962-10-08 1966-05-24 Lilly Co Eli Acylation via carbodimides for penicillin and cephalosporin preparation
SE320074B (pt) * 1964-01-16 1970-02-02 Astra Ab

Also Published As

Publication number Publication date
DK140943B (da) 1979-12-10
BE675298A (pt) 1966-07-18
DE1670600A1 (de) 1970-08-06
US3518260A (en) 1970-06-30
NL6600636A (pt) 1966-09-09
SE354663B (pt) 1973-03-19
CH480368A (de) 1969-10-31
DK140943C (pt) 1980-05-19
GB1123333A (en) 1968-08-14
CY527A (en) 1970-02-16

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