BR6682746D0 - Processo para a preparacao de novos derivados de ciclopentanofenantreno - Google Patents

Processo para a preparacao de novos derivados de ciclopentanofenantreno

Info

Publication number
BR6682746D0
BR6682746D0 BR182746/66A BR18274666A BR6682746D0 BR 6682746 D0 BR6682746 D0 BR 6682746D0 BR 182746/66 A BR182746/66 A BR 182746/66A BR 18274666 A BR18274666 A BR 18274666A BR 6682746 D0 BR6682746 D0 BR 6682746D0
Authority
BR
Brazil
Prior art keywords
cyclopentanofenantrene
derivatives
preparation
new
new cyclopentanofenantrene
Prior art date
Application number
BR182746/66A
Other languages
English (en)
Inventor
C Beard
A Cross
Original Assignee
Syntex Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Corp filed Critical Syntex Corp
Publication of BR6682746D0 publication Critical patent/BR6682746D0/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J75/00Processes for the preparation of steroids in general
    • FMECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F28HEAT EXCHANGE IN GENERAL
    • F28BSTEAM OR VAPOUR CONDENSERS
    • F28B1/00Condensers in which the steam or vapour is separate from the cooling medium by walls, e.g. surface condenser
    • F28B1/06Condensers in which the steam or vapour is separate from the cooling medium by walls, e.g. surface condenser using air or other gas as the cooling medium
    • FMECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F28HEAT EXCHANGE IN GENERAL
    • F28FDETAILS OF HEAT-EXCHANGE AND HEAT-TRANSFER APPARATUS, OF GENERAL APPLICATION
    • F28F13/00Arrangements for modifying heat-transfer, e.g. increasing, decreasing
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00Chemistry: molecular biology and microbiology
    • Y10S435/8215Microorganisms
    • Y10S435/911Microorganisms using fungi

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Mechanical Engineering (AREA)
  • General Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Thermal Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR182746/66A 1965-09-09 1966-09-09 Processo para a preparacao de novos derivados de ciclopentanofenantreno BR6682746D0 (pt)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US486226A US3338928A (en) 1965-09-09 1965-09-09 Fused halocyclopropyl steroids
US49909265A 1965-10-20 1965-10-20
US49909165A 1965-10-20 1965-10-20
US502376A US3338893A (en) 1965-09-09 1965-10-22 Fused halocyclopropyl steroids
US502375A US3414592A (en) 1965-09-09 1965-10-22 6, 7-halomethylene androstanes and estranes and processes for their preparation
US513548A US3357973A (en) 1965-09-09 1965-12-13 7alpha-mono-and dihalomethyl steroids
US581457A US3376292A (en) 1965-09-09 1966-09-23 16alpha, 17alpha-dihalomethylene[3, 2-c]pyrazole derivatives of the pregnane series
US601862A US3365444A (en) 1965-09-09 1966-12-15 5'-hydroxypregneno [3, 2-c] pyrazole derivatives and process for their preparation

Publications (1)

Publication Number Publication Date
BR6682746D0 true BR6682746D0 (pt) 1973-12-26

Family

ID=27575452

Family Applications (1)

Application Number Title Priority Date Filing Date
BR182746/66A BR6682746D0 (pt) 1965-09-09 1966-09-09 Processo para a preparacao de novos derivados de ciclopentanofenantreno

Country Status (10)

Country Link
US (6) US3338928A (pt)
JP (1) JPS4812739B1 (pt)
BE (1) BE686640A (pt)
BR (1) BR6682746D0 (pt)
CH (2) CH533094A (pt)
DE (2) DE1593427A1 (pt)
FR (2) FR1500247A (pt)
GB (2) GB1163736A (pt)
NL (2) NL6612635A (pt)
SE (2) SE348189B (pt)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3435057A (en) * 1966-01-03 1969-03-25 Syntex Corp 16alpha,17alpha-ethylene and substituted ethylene pregnane derivatives and process
US3431256A (en) * 1966-02-14 1969-03-04 Syntex Corp 16alpha,17alpha-ethylene and substituted ethylene pregnane derivatives and process
US3400137A (en) * 1966-02-17 1968-09-03 Syntex Corp 3-desoxy-pregnenes and -19nor-pregnenes and their preparation
US3423507A (en) * 1966-02-25 1969-01-21 Schering Corp Method of treating benign prostratic hypertrophy
DE1593501C3 (de) * 1966-04-02 1975-09-11 Schering Ag, 1000 Berlin Und 4619 Bergkamen 15,16 beta-Methylensteroide der 19-Nor-androstan-Reihe, Verfahren zu deren Herstellung sowie diese enthaltende Mittel
CH540896A (de) * 1966-04-02 1973-10-15 Schering Ag Verfahren zur Herstellung von 15,16B-Methylensteroiden
US3409610A (en) * 1966-06-27 1968-11-05 Syntex Corp 9alpha-difluoromethyl and 9alpha-trifluoromethyl pregnenes
US3438975A (en) * 1966-07-01 1969-04-15 Syntex Corp 15alpha,16alpha-methylene pregnanes and 19-nor-pregnanes
US3541082A (en) * 1966-09-26 1970-11-17 Upjohn Co Steroidal delta**16-20(alpha and beta)-hydroperoxide 21-ethers
US3444295A (en) * 1966-12-29 1969-05-13 Schering Ag Anabolic composition comprising 1,2alpha-methylene-19-nor testosterone
DE1643005C3 (de) * 1967-02-09 1975-05-22 Schering Ag, 1000 Berlin Und 4619 Bergkamen 15,16beta-Methylen-testosterone, Verfahren zu ihrer Herstellung sowie diese Steroide enthaltende Mittel
US3435056A (en) * 1967-09-13 1969-03-25 Syntex Corp Halogenated cyclopropyl and cyclopropenyl steroids and process for their preparation
US3700702A (en) * 1970-12-02 1972-10-24 Hoffmann La Roche New 15{62 ,16{62 -methylene steroids
GB1377608A (en) * 1970-12-17 1974-12-18 Glaxo Lab Ltd 3alpha-hydroxy or acyloxy pregnene-21-ethers
US3718673A (en) * 1971-02-01 1973-02-27 Du Pont Process for the preparation of 21-chloro-6,6,9alpha-trifluoro-11beta, alpha, 17alpha-trihydroxy-1,4-pregnadien-3,20-dione 16,17-ketals and selected intermediates
US3932388A (en) * 1974-04-22 1976-01-13 Schering Corporation -Azido-4,6-pregnadieno(3,2-c)pyrazoles, processes for their preparation and intermediates useful therein
DE2803187A1 (de) * 1978-01-23 1979-08-02 Schering Ag Neue kortikoide, ihre herstellung und verwendung
JPS5578308A (en) * 1978-12-07 1980-06-12 Nippon Denso Co Ltd Temperature control method
IT1149935B (it) * 1980-07-02 1986-12-10 Finchimica Srl Uso farmacologico del 6-cloro-17-idrossi 1 alfa,2 alfa-metilpregna 4,6-dien-3,20-dione
AU572589B2 (en) 1983-12-14 1988-05-12 Upjohn Company, The 11(alpha)-difluoromethyl and (e)-and (z)-11-fluoromethylene steroids

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3047566A (en) * 1958-06-13 1962-07-31 Leo Pharm Prod Ltd 6a, 6a-dihalo-6, 7-methylene steroids and method
US3299054A (en) * 1961-12-01 1967-01-17 Merck & Co Inc 4-pregneno-[3, 2-c] pyrazoles and processes of preparing them
GB1101117A (en) * 1964-02-01 1968-01-31 Ormonoterapia Richter Spa Steroidal 2ª‡-carbonylhydrazones

Also Published As

Publication number Publication date
DE1593426A1 (de) 1970-07-30
FR1500247A (fr) 1967-11-03
NL6612687A (pt) 1967-03-10
US3338893A (en) 1967-08-29
US3414592A (en) 1968-12-03
US3376292A (en) 1968-04-02
US3357973A (en) 1967-12-12
CH480315A (de) 1969-10-31
US3338928A (en) 1967-08-29
DE1593427A1 (de) 1970-07-30
NL6612635A (pt) 1967-03-10
GB1163736A (en) 1969-09-10
CH533094A (de) 1973-01-31
JPS4812739B1 (pt) 1973-04-23
SE348189B (pt) 1972-08-28
US3365444A (en) 1968-01-23
FR6651M (pt) 1969-01-27
BE686640A (pt) 1967-02-15
GB1163737A (en) 1969-09-10
SE376426B (pt) 1975-05-26

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