BR6572768D0 - Processo para a preparacao de nucleosidas - Google Patents

Processo para a preparacao de nucleosidas

Info

Publication number
BR6572768D0
BR6572768D0 BR172768/65A BR17276865A BR6572768D0 BR 6572768 D0 BR6572768 D0 BR 6572768D0 BR 172768/65 A BR172768/65 A BR 172768/65A BR 17276865 A BR17276865 A BR 17276865A BR 6572768 D0 BR6572768 D0 BR 6572768D0
Authority
BR
Brazil
Prior art keywords
nucleosides
preparation
Prior art date
Application number
BR172768/65A
Other languages
English (en)
Inventor
T Shen
W Ruyle
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of BR6572768D0 publication Critical patent/BR6572768D0/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR172768/65A 1964-09-02 1965-08-31 Processo para a preparacao de nucleosidas BR6572768D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US394054A US3328388A (en) 1964-09-02 1964-09-02 Arabinofuranosyl pyrimidines and methods of preparing same

Publications (1)

Publication Number Publication Date
BR6572768D0 true BR6572768D0 (pt) 1973-08-07

Family

ID=23557362

Family Applications (1)

Application Number Title Priority Date Filing Date
BR172768/65A BR6572768D0 (pt) 1964-09-02 1965-08-31 Processo para a preparacao de nucleosidas

Country Status (6)

Country Link
US (1) US3328388A (pt)
BR (1) BR6572768D0 (pt)
CH (1) CH477453A (pt)
DE (1) DE1595946A1 (pt)
GB (2) GB1104999A (pt)
NL (1) NL6511420A (pt)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1030970A (en) * 1964-05-15 1966-05-25 Inst Mikrobiologii Im Akad D K Method for the preparation of 2', 3', 5'-tri-o-acyl-6-azacytidines
US3404144A (en) * 1965-12-23 1968-10-01 Research Corp 1-beta-d-arabinofuranosyl-5-fluorocytosine compounds
US3462416A (en) * 1967-01-30 1969-08-19 Upjohn Co Hydrogenated pyrimidine nucleosides and nucleotides
DE2012888C3 (de) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden
GB1386585A (en) * 1970-11-16 1975-03-12 Wellcome Found Purine sugar derivatives
DE2122991C2 (de) * 1971-05-04 1982-06-09 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von Cytosin- und 6-Azacytosinnucleosiden
US3869446A (en) * 1971-11-18 1975-03-04 Ceskoslovenska Akademie Ved Process of preparing 6-azapyrimidine ribonucleosides
US3935184A (en) * 1972-02-22 1976-01-27 Syntex (U.S.A.) Inc. Synthetic polyoxin type nucleosides
US3998807A (en) * 1972-03-03 1976-12-21 Syntex (U.S.A.) Inc. Arabinofuranosyl cytosines and methods of making
US4017606A (en) * 1973-10-04 1977-04-12 The Upjohn Company Organic compounds and process
JPS61204193A (ja) * 1985-03-05 1986-09-10 Takeda Chem Ind Ltd シトシンヌクレオシド類の製造法
US5215971A (en) * 1986-12-19 1993-06-01 Medivir Ab Antiviral pharmaceutical composition comprising 5-substituted pyrimidine nucleosides
SE8605503D0 (sv) * 1986-12-19 1986-12-19 Astra Laekemedel Ab Novel medicinal use
GB8726136D0 (en) * 1987-11-07 1987-12-09 Wellcome Found Therapeutic nucleosides
US5684164A (en) 1988-04-11 1997-11-04 Biochem Pharma Inc. Processes for preparing substituted 1,3-oxathiolanes with antiviral properties
WO2004041834A2 (en) * 2002-10-31 2004-05-21 Metabasis Therapeutics, Inc. Novel cyclic phosphate diesters of 1,3-propane-1-aryl diols and their use in preparing prodrugs
EP2883959A1 (en) 2013-12-13 2015-06-17 Plasmia Biotech, S.L. Enzymatic production of cytosinic nucleoside analogues
AU2015217221A1 (en) 2014-02-13 2016-08-11 Ligand Pharmaceuticals, Inc. Prodrug compounds and their uses
JP6262079B2 (ja) * 2014-06-02 2018-01-17 東ソー・ファインケム株式会社 4−(2,2,2−トリフルオロエトキシ)−5−(トリフルオロメチル)ピリミジン誘導体及びその製造方法
CN106687118A (zh) 2014-07-02 2017-05-17 配体药物公司 前药化合物及其用途
EP3737676B1 (en) 2018-01-09 2024-03-06 Ligand Pharmaceuticals, Inc. Acetal compounds and therapeutic uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2885396A (en) * 1957-03-21 1959-05-05 Heidelberger Charles N-glycosides of 5-fluorouracil
US2949451A (en) * 1959-04-21 1960-08-16 Hoffmann La Roche Preparation of thymidine and deoxyfluorouridine, and intermediates therefor
NL299755A (pt) * 1959-06-03
US3135737A (en) * 1960-06-30 1964-06-02 Olin Mathieson Chemical Compan 3-(hydrocarbonthio)-2-(tri-o-benzoylribofuranosyl)-as-triazin-5(2h)-ones and process therefor

Also Published As

Publication number Publication date
GB1104998A (en) 1968-03-06
NL6511420A (pt) 1966-03-03
DE1595946A1 (de) 1970-07-09
US3328388A (en) 1967-06-27
GB1104999A (en) 1968-03-06
CH477453A (de) 1969-08-31

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