BR112022005449A2 - Compostos antibacterianos - Google Patents

Compostos antibacterianos

Info

Publication number
BR112022005449A2
BR112022005449A2 BR112022005449A BR112022005449A BR112022005449A2 BR 112022005449 A2 BR112022005449 A2 BR 112022005449A2 BR 112022005449 A BR112022005449 A BR 112022005449A BR 112022005449 A BR112022005449 A BR 112022005449A BR 112022005449 A2 BR112022005449 A2 BR 112022005449A2
Authority
BR
Brazil
Prior art keywords
antibacterial compounds
compounds
antibacterial
tuberculosis
medicaments
Prior art date
Application number
BR112022005449A
Other languages
English (en)
Inventor
Antonie Lamprecht Dirk
Anita Lanckacker Ellen
Maria J Lammens Godelieve
Émile Georges Guillemont Jérôme
Friedrich Walter Weidner Steffen
Original Assignee
Janssen Sciences Ireland Unlimited Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Sciences Ireland Unlimited Co filed Critical Janssen Sciences Ireland Unlimited Co
Publication of BR112022005449A2 publication Critical patent/BR112022005449A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/005Enzyme inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

compostos antibacterianos. a presente invenção refere-se aos seguintes compostos em que as partes inteiras são como definidas na descrição e em que os compostos podem ser úteis como medicamentos, por exemplo, para uso no tratamento de tuberculose (por exemplo, em combinação).
BR112022005449A 2019-09-30 2020-09-29 Compostos antibacterianos BR112022005449A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP19200377 2019-09-30
PCT/EP2020/077175 WO2021063915A1 (en) 2019-09-30 2020-09-29 Antibacterial compounds

Publications (1)

Publication Number Publication Date
BR112022005449A2 true BR112022005449A2 (pt) 2022-06-21

Family

ID=68104409

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112022005449A BR112022005449A2 (pt) 2019-09-30 2020-09-29 Compostos antibacterianos

Country Status (10)

Country Link
US (1) US20220372033A1 (pt)
EP (1) EP4038069A1 (pt)
JP (1) JP2022551823A (pt)
KR (1) KR20220075335A (pt)
CN (1) CN114466848A (pt)
AU (1) AU2020360560A1 (pt)
BR (1) BR112022005449A2 (pt)
CA (1) CA3151712A1 (pt)
MX (1) MX2022003816A (pt)
WO (1) WO2021063915A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4296674A1 (en) 2022-06-20 2023-12-27 Université Toulouse III - Paul Sabatier Innovative molecules decreasing virulence of mycobacterium for the treatment of tuberculosis

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI2301544T1 (sl) 2002-07-25 2013-01-31 Janssen Pharmaceutica, N.V. Derivati kinolina kot vmesne spojine za mikobakterijske inhibitorje
MX345762B (es) * 2010-03-18 2017-02-15 Pasteur Institut Korea Compuestos antiinfecciosos.
GB201020076D0 (en) * 2010-11-26 2011-01-12 Liverpool School Tropical Medicine Antimalarial compounds
CN105745208A (zh) * 2013-08-02 2016-07-06 韩国巴斯德研究所 一种抗感染化合物
EA201890204A1 (ru) 2015-07-02 2018-06-29 Янссен Сайенсиз Айрлэнд Юси Антибактериальные соединения
GB201522232D0 (en) * 2015-12-16 2016-01-27 Liverpool School Tropical Medicine Combination product
MA45377A (fr) 2016-06-16 2019-04-24 Janssen Sciences Ireland Unlimited Co Composés hétérocycliques en tant qu'agents antibacteriens
JP2019518050A (ja) 2016-06-16 2019-06-27 ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー 抗菌薬としての複素環式化合物
WO2018084809A1 (en) * 2016-11-02 2018-05-11 Nanyang Technological University Methods for the treatment or prevention of mycobacterial infections

Also Published As

Publication number Publication date
AU2020360560A1 (en) 2022-03-10
EP4038069A1 (en) 2022-08-10
JP2022551823A (ja) 2022-12-14
CA3151712A1 (en) 2021-04-08
WO2021063915A1 (en) 2021-04-08
CN114466848A (zh) 2022-05-10
MX2022003816A (es) 2022-05-06
US20220372033A1 (en) 2022-11-24
KR20220075335A (ko) 2022-06-08

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