BR112015000150A2 - composições farmacêuticas dissuasoras de abuso de liberação controlada - Google Patents

composições farmacêuticas dissuasoras de abuso de liberação controlada

Info

Publication number
BR112015000150A2
BR112015000150A2 BR112015000150A BR112015000150A BR112015000150A2 BR 112015000150 A2 BR112015000150 A2 BR 112015000150A2 BR 112015000150 A BR112015000150 A BR 112015000150A BR 112015000150 A BR112015000150 A BR 112015000150A BR 112015000150 A2 BR112015000150 A2 BR 112015000150A2
Authority
BR
Brazil
Prior art keywords
controlled release
pharmaceutical compositions
abuse deterrent
deterrent pharmaceutical
release abuse
Prior art date
Application number
BR112015000150A
Other languages
English (en)
Inventor
Boye George
Engslev Fischer Gina
Martin ØVERGÅRD Jan
Lindhart Karsten
Rex Olsen Martin
Skak Nikolaj
Holm Tygesen Peter
Elhauge Torben
Original Assignee
Egalet Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48703579&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112015000150(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Egalet Ltd filed Critical Egalet Ltd
Publication of BR112015000150A2 publication Critical patent/BR112015000150A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, ***e
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, ***e

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

resumo da patente de invenção para: “composições farmacêuticas dissuasoras de abuso de liberação controlada". a presente invenção se refere a composições farmacêuticas que são resistentes ao abuso e que também podem permitir liberação controlada. a presente invenção também se refere ao uso das ditas composições farmacêuticas no tratamento de dor.
BR112015000150A 2012-07-06 2013-07-01 composições farmacêuticas dissuasoras de abuso de liberação controlada BR112015000150A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261668741P 2012-07-06 2012-07-06
DKPA201270405 2012-07-06
PCT/EP2013/063851 WO2014006004A1 (en) 2012-07-06 2013-07-01 Abuse deterrent pharmaceutical compositions for controlled release

Publications (1)

Publication Number Publication Date
BR112015000150A2 true BR112015000150A2 (pt) 2017-06-27

Family

ID=48703579

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015000150A BR112015000150A2 (pt) 2012-07-06 2013-07-01 composições farmacêuticas dissuasoras de abuso de liberação controlada

Country Status (13)

Country Link
US (3) US9549899B2 (pt)
EP (1) EP2877161A1 (pt)
JP (1) JP2015521988A (pt)
KR (1) KR20150059167A (pt)
CN (1) CN104684548A (pt)
AU (1) AU2013285988A1 (pt)
BR (1) BR112015000150A2 (pt)
CA (1) CA2877183A1 (pt)
EA (1) EA201590165A1 (pt)
HK (1) HK1210599A1 (pt)
MX (1) MX2014015880A (pt)
NZ (1) NZ704011A (pt)
WO (1) WO2014006004A1 (pt)

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US20210322321A1 (en) * 2018-10-19 2021-10-21 Temple University-Of The Commonwealth System Of Higher Education Tamper-resistant drug dosage forms and methods of making and use thereof
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US20140220126A1 (en) 2014-08-07
US9044402B2 (en) 2015-06-02
US20140010873A1 (en) 2014-01-09
US20170333354A9 (en) 2017-11-23
HK1210599A1 (en) 2016-04-29
EP2877161A1 (en) 2015-06-03
NZ704011A (en) 2016-04-29
KR20150059167A (ko) 2015-05-29
JP2015521988A (ja) 2015-08-03
US9549899B2 (en) 2017-01-24
US20170181974A1 (en) 2017-06-29
CN104684548A (zh) 2015-06-03
EA201590165A1 (ru) 2015-08-31
AU2013285988A1 (en) 2015-02-12
CA2877183A1 (en) 2014-01-09
WO2014006004A1 (en) 2014-01-09

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