BR1100336A - Composição farmacêutica para uso oral, e, processo para preparar a mesma - Google Patents

Composição farmacêutica para uso oral, e, processo para preparar a mesma

Info

Publication number
BR1100336A
BR1100336A BR1100336-7A BR1100336A BR1100336A BR 1100336 A BR1100336 A BR 1100336A BR 1100336 A BR1100336 A BR 1100336A BR 1100336 A BR1100336 A BR 1100336A
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
oral use
compound
formula
melting point
Prior art date
Application number
BR1100336-7A
Other languages
English (en)
Inventor
Tadashi Makino
Yoshio Mizukami
Jun-Ichi Kikuta
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=17938952&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR1100336(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Priority to BR1100336-7A priority Critical patent/BR1100336A/pt
Publication of BR1100336A publication Critical patent/BR1100336A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Plural Heterocyclic Compounds (AREA)
BR1100336-7A 1991-11-20 1997-04-23 Composição farmacêutica para uso oral, e, processo para preparar a mesma BR1100336A (pt)

Priority Applications (1)

Application Number Priority Date Filing Date Title
BR1100336-7A BR1100336A (pt) 1991-11-20 1997-04-23 Composição farmacêutica para uso oral, e, processo para preparar a mesma

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP30492491 1991-11-20
BR1100336-7A BR1100336A (pt) 1991-11-20 1997-04-23 Composição farmacêutica para uso oral, e, processo para preparar a mesma

Publications (1)

Publication Number Publication Date
BR1100336A true BR1100336A (pt) 2000-04-18

Family

ID=17938952

Family Applications (1)

Application Number Title Priority Date Filing Date
BR1100336-7A BR1100336A (pt) 1991-11-20 1997-04-23 Composição farmacêutica para uso oral, e, processo para preparar a mesma

Country Status (18)

Country Link
US (1) US5534534A (pt)
EP (3) EP0546358B1 (pt)
KR (1) KR100256633B1 (pt)
CN (1) CN1047518C (pt)
AT (2) ATE157248T1 (pt)
AU (1) AU659691B2 (pt)
BR (1) BR1100336A (pt)
CA (1) CA2083305C (pt)
DE (2) DE69221831T2 (pt)
DK (1) DK0546358T3 (pt)
ES (1) ES2104797T3 (pt)
FI (2) FI111604B (pt)
GR (1) GR3025338T3 (pt)
HU (1) HU211608A9 (pt)
MX (1) MX9206634A (pt)
NO (1) NO304408B1 (pt)
NZ (1) NZ245175A (pt)
TW (1) TW284688B (pt)

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TW284688B (pt) * 1991-11-20 1996-09-01 Takeda Pharm Industry Co Ltd
TW272942B (pt) * 1993-02-10 1996-03-21 Takeda Pharm Industry Co Ltd
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TW418204B (en) * 1997-03-28 2001-01-11 Dev Center Biotechnology Novel 1,2,4-triazine-5-ketonyl benzene derivatives and the analogs, the preparation, and the pharmaceutical compositions as angiotension II receptor antogonists
US6297239B1 (en) 1997-10-08 2001-10-02 Merck & Co., Inc. Inhibitors of prenyl-protein transferase
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US20050031683A1 (en) * 2003-08-04 2005-02-10 Ashish Kapoor Solid pharmaceutical composition
CA2542499A1 (en) * 2003-10-16 2005-04-28 Teva Pharmaceutical Industries Ltd. Preparation of candesartan cilexetil
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EP1711168A2 (en) * 2004-01-23 2006-10-18 Ranbaxy Laboratories Limited Oral pharmaceutical compositions of candesartan cilexetil
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EP1742938A1 (en) * 2004-05-05 2007-01-17 Teva Pharmaceutical Industries Ltd. Preparation of candesartan cilexetil in high purity
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EP1836195A2 (en) * 2005-01-14 2007-09-26 Teva Pharmaceutical Industries Ltd Preparation of crude candesartan cilexetil
DK1843754T3 (da) * 2005-01-26 2011-11-21 Lek Pharmaceuticals Ny farmaceutisk sammensætning indeholdende candesartan-cilexetil som lipofilt krystallinsk stof
EP1763525A2 (en) * 2005-05-10 2007-03-21 Teva Pharmaceutical Industries Ltd. Stable micronized candesartan cilexetil and methods for preparing thereof
US7815939B2 (en) * 2005-07-20 2010-10-19 Astellas Pharma Inc. Coated fine particles containing drug for intrabuccally fast disintegrating dosage forms
PE20080696A1 (es) * 2006-04-27 2008-08-04 Takeda Pharmaceutical Composicion farmaceutica solida que comprende un derivado de bencimidazol y clorhidrato de pioglitazona
CN101528262A (zh) * 2006-08-10 2009-09-09 武田药品工业株式会社 药物组合物
WO2008045006A1 (en) * 2006-10-11 2008-04-17 Fako Ilaclari A. S. Formulations of candesartan
ES2301401B1 (es) * 2006-11-28 2009-06-08 Laboratorios Liconsa S.A. Composicion farmaceutica solida estabilizada de candesartan cilexetilo.
EP1952806A1 (en) 2007-02-01 2008-08-06 Helm AG Process for the preparation of adsorbates of candesartan
DE602008002371D1 (de) * 2007-03-08 2010-10-14 Teva Pharma Pharmazeutische zusammensetzung mit candesartan-cilexetil
CL2008000868A1 (es) * 2007-03-28 2008-10-10 Takeda Pharmaceutical Composicion farmaceutica solida que comprende un compuesto derivado de benzimidazol y un agente de control de ph; metodo de estabilizacion y de mejoramiento de la disolucion; uso de un agente de control de ph.
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WO2008149338A2 (en) * 2007-06-06 2008-12-11 Dexcel Ltd. Process for forming solid oral dosage forms of angiotensin ii receptor antagonists
DE102007052070A1 (de) 2007-10-30 2009-05-07 Tiefenbacher Pharmachemikalien Alfred E. Tiefenbacher Gmbh & Co. Kg Candesartancilexetil
SI2165702T1 (sl) 2008-09-17 2012-05-31 Helm Ag Stabilni in z lahkoto raztopljeni sestavki kandesartan cileksetila pripravljeni z vlažno granulacijo
WO2010075347A2 (en) 2008-12-23 2010-07-01 Takeda Pharmaceutical Company Limited Methods of treating hypertension with at least one angiotensin ii receptor blocker and chlorthalidone
ES2364011B1 (es) 2009-11-20 2013-01-24 Gp Pharm, S.A. Cápsulas de principios activos farmacéuticos y ésteres de ácidos grasos poliinsaturados para el tratamiento de enfermedades cardiovasculares.
WO2012047538A1 (en) 2010-10-06 2012-04-12 Glaxosmithkline Llc Benzimidazole derivatives as pi3 kinase inhibitors
CN102138920A (zh) * 2011-02-24 2011-08-03 海南中济医药科技有限公司 一种含有坎地沙坦酯和氢***的药物组合物及其制备方法
CN102357095A (zh) * 2011-07-12 2012-02-22 迪沙药业集团有限公司 稳定的药物组合物
AP2014007621A0 (en) 2011-11-11 2014-05-31 Pfizer 2-Thiopyrimidinones
WO2014088123A1 (en) * 2012-12-05 2014-06-12 Sawai Pharmaceutical Co., Ltd. Candesartan cilexetil-containing preparation
PL236001B1 (pl) 2012-12-21 2020-11-30 Adamed Spolka Z Ograniczona Odpowiedzialnoscia Złożona kompozycja farmaceutyczna zawierająca kandesartan cyleksetylu oraz amlodypinę, sposób jej wytwarzania oraz jednostkowa postać dawkowania zawierająca tę kompozycję
EP2990038B1 (en) 2013-04-25 2019-11-20 Kyorin Pharmaceutical Co., Ltd. Solid pharmaceutical composition
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CN111617046A (zh) * 2020-07-09 2020-09-04 浙江诺得药业有限公司 阿齐沙坦分散片及其制备工艺
CN112957336A (zh) * 2021-03-03 2021-06-15 广州白云山天心制药股份有限公司 一种稳定的坎地沙坦酯药物固体组合物及其制备方法

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Also Published As

Publication number Publication date
KR930009606A (ko) 1993-06-21
EP1468683A3 (en) 2012-06-06
EP0782852B1 (en) 2004-09-29
CA2083305C (en) 2003-12-09
ES2104797T3 (es) 1997-10-16
EP0782852A1 (en) 1997-07-09
NZ245175A (en) 1994-07-26
DE69233424T2 (de) 2005-02-17
ATE277602T1 (de) 2004-10-15
CA2083305A1 (en) 1993-05-21
US5534534A (en) 1996-07-09
CN1047518C (zh) 1999-12-22
MX9206634A (es) 1993-05-31
CN1072338A (zh) 1993-05-26
AU659691B2 (en) 1995-05-25
ATE157248T1 (de) 1997-09-15
AU2839192A (en) 1993-05-27
NO924417L (no) 1993-05-21
FI925270A0 (fi) 1992-11-19
EP0546358B1 (en) 1997-08-27
GR3025338T3 (en) 1998-02-27
NO304408B1 (no) 1998-12-14
EP0546358A3 (pt) 1994-03-30
DK0546358T3 (da) 1998-03-09
DE69221831D1 (de) 1997-10-02
FI20030210A (fi) 2003-02-12
EP0546358A2 (en) 1993-06-16
HU211608A9 (en) 1995-12-28
TW284688B (pt) 1996-09-01
EP1468683A2 (en) 2004-10-20
NO924417D0 (no) 1992-11-16
DE69233424D1 (de) 2004-11-04
KR100256633B1 (ko) 2000-05-15
FI925270A (fi) 1993-05-21
DE69221831T2 (de) 1998-01-02
FI111604B (fi) 2003-08-29

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