BR0215752A - Pyanoindazoles and their use in the treatment of glaucoma - Google Patents

Pyanoindazoles and their use in the treatment of glaucoma

Info

Publication number
BR0215752A
BR0215752A BR0215752-7A BR0215752A BR0215752A BR 0215752 A BR0215752 A BR 0215752A BR 0215752 A BR0215752 A BR 0215752A BR 0215752 A BR0215752 A BR 0215752A
Authority
BR
Brazil
Prior art keywords
glaucoma
treatment
pyanoindazoles
disclosed
pyanoindoles
Prior art date
Application number
BR0215752-7A
Other languages
Portuguese (pt)
Inventor
Hwang-Hsing Chen
Jesse A Way
Bryon S Severns
Original Assignee
Alcon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alcon Inc filed Critical Alcon Inc
Publication of BR0215752A publication Critical patent/BR0215752A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

"PIRANOINDAZóIS E SEU USO NO TRATAMENTO DE GLAUCOMA". Divulgam-se piranoindazóis. Divulgam-se também métodos para a diminuição e controle de pressão intra-ocular normal ou elevada assim como um método para o tratamento de glaucoma usando composições contendo um ou mais dos compostos da invenção presente.s"Pyanoindoles and their use in the treatment of glaucoma". Pyranoindoles are disclosed. Methods for the reduction and control of normal or elevated intraocular pressure as well as a method for treating glaucoma using compositions containing one or more of the compounds of the present invention are also disclosed.

BR0215752-7A 2002-05-30 2002-12-11 Pyanoindazoles and their use in the treatment of glaucoma BR0215752A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1686102A 2002-05-30 2002-05-30
PCT/US2002/039666 WO2003101379A2 (en) 2002-05-30 2002-12-11 Pyranoindazoles and their use for the treatment of glaucoma

Publications (1)

Publication Number Publication Date
BR0215752A true BR0215752A (en) 2005-03-29

Family

ID=29709135

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0215752-7A BR0215752A (en) 2002-05-30 2002-12-11 Pyanoindazoles and their use in the treatment of glaucoma

Country Status (7)

Country Link
EP (1) EP1513521A2 (en)
JP (1) JP2005532337A (en)
AU (1) AU2002353122B2 (en)
BR (1) BR0215752A (en)
CA (1) CA2486832A1 (en)
MX (1) MXPA04011791A (en)
WO (1) WO2003101379A2 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200520760A (en) 2003-12-15 2005-07-01 Alcon Inc Substituted [1,4] oxazino [2,3-g] indazoles for the treatment of glaucoma
US7425572B2 (en) 2004-12-08 2008-09-16 Alcon, Inc. Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma
TWI667233B (en) 2013-12-19 2019-08-01 德商拜耳製藥公司 Novel indazolecarboxamides, processes for their preparation, pharmaceutical preparations comprising them and their use for producing medicaments

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1392658A4 (en) * 2001-06-01 2004-10-13 Alcon Inc Novel fused indazoles and indoles and their use for the treatment of glaucoma

Also Published As

Publication number Publication date
JP2005532337A (en) 2005-10-27
CA2486832A1 (en) 2003-12-11
AU2002353122B2 (en) 2008-01-31
AU2002353122A1 (en) 2003-12-19
WO2003101379A2 (en) 2003-12-11
EP1513521A2 (en) 2005-03-16
WO2003101379A3 (en) 2004-03-04
MXPA04011791A (en) 2005-07-26

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Legal Events

Date Code Title Description
B08F Application fees: dismissal - article 86 of industrial property law

Free format text: REFERENTE A(S) 8A ANUIDADE(S).

B08K Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87)

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2108 DE 31/05/2011.