BR0113634A - Antibióticos de cefalosporina e suas pró-drogas - Google Patents

Antibióticos de cefalosporina e suas pró-drogas

Info

Publication number
BR0113634A
BR0113634A BR0113634-8A BR0113634A BR0113634A BR 0113634 A BR0113634 A BR 0113634A BR 0113634 A BR0113634 A BR 0113634A BR 0113634 A BR0113634 A BR 0113634A
Authority
BR
Brazil
Prior art keywords
prodrugs
antibiotics
cephalosporin antibiotics
cefalosporin
bacteria
Prior art date
Application number
BR0113634-8A
Other languages
English (en)
Inventor
Tomasz W Glinka
Original Assignee
Tomasz W Glinka
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tomasz W Glinka filed Critical Tomasz W Glinka
Publication of BR0113634A publication Critical patent/BR0113634A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Abstract

"ANTIBIóTICOS DE CEFALOSPORINA E SUAS PRó-DROGAS". A presente invenção refere-se a novos antibióticos de cefalosporina, suas pró-drogas e sais farmacologicamente aceitáveis destes, que são ativos contra um amplo espectro de bactérias que são resistentes a antibióticos de beta-lactama clínicos atuais.
BR0113634-8A 2000-08-29 2001-08-23 Antibióticos de cefalosporina e suas pró-drogas BR0113634A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22917400P 2000-08-29 2000-08-29
PCT/US2001/026628 WO2002017854A2 (en) 2000-08-29 2001-08-23 Cephalosporin antibiotics and prodrugs thereof

Publications (1)

Publication Number Publication Date
BR0113634A true BR0113634A (pt) 2004-02-03

Family

ID=22860110

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0113634-8A BR0113634A (pt) 2000-08-29 2001-08-23 Antibióticos de cefalosporina e suas pró-drogas

Country Status (16)

Country Link
US (1) US6599893B2 (pt)
EP (1) EP1333836A4 (pt)
JP (1) JP2004507481A (pt)
CN (1) CN1471399A (pt)
AR (1) AR030503A1 (pt)
AU (2) AU2001288420B2 (pt)
BR (1) BR0113634A (pt)
CA (1) CA2420871A1 (pt)
IL (1) IL154518A0 (pt)
MX (1) MXPA03001782A (pt)
NO (1) NO20030931L (pt)
NZ (1) NZ524438A (pt)
RU (1) RU2281948C2 (pt)
TW (1) TWI283681B (pt)
WO (1) WO2002017854A2 (pt)
ZA (1) ZA200301391B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0307834D0 (en) * 2003-04-04 2003-05-14 Ta Contrast Ab Composition
CA2526875A1 (en) * 2003-04-30 2004-11-18 Trine Pharmaceuticals, Inc. Carbacephem beta-lactam antibiotics
CN101210020B (zh) * 2006-12-31 2010-11-24 山东轩竹医药科技有限公司 新型头孢菌素化合物
EA201070504A1 (ru) * 2007-10-25 2010-12-30 Эйкеоджен, Инк. КАРБАЦЕФЕМ β-ЛАКТАМОВЫЕ АНТИБИОТИКИ
EP2285381B1 (en) 2008-05-05 2015-12-16 The General Hospital Corporation Photoactivatable beta-lactamase substrates and analytical methods of using same
CN103945842A (zh) 2011-09-09 2014-07-23 丘比斯特药物股份有限公司 治疗肺内感染的方法
US8809314B1 (en) 2012-09-07 2014-08-19 Cubist Pharmacueticals, Inc. Cephalosporin compound
US8476425B1 (en) 2012-09-27 2013-07-02 Cubist Pharmaceuticals, Inc. Tazobactam arginine compositions
US20140274991A1 (en) 2013-03-15 2014-09-18 Cubist Pharmaceuticals, Inc. Ceftolozane pharmaceutical compositions
KR102329764B1 (ko) 2013-03-15 2021-11-23 머크 샤프 앤드 돔 코포레이션 세프톨로잔 항균성 조성물
US9872906B2 (en) 2013-03-15 2018-01-23 Merck Sharp & Dohme Corp. Ceftolozane antibiotic compositions
CA2910752C (en) * 2013-05-01 2021-11-23 Neoculi Pty Ltd Use of robenidine in the treatment of bacterial infection
WO2015035376A2 (en) 2013-09-09 2015-03-12 Calixa Therapeutics, Inc. Treating infections with ceftolozane/tazobactam in subjects having impaired renal function
US20150094293A1 (en) 2013-09-27 2015-04-02 Calixa Therapeutics, Inc. Solid forms of ceftolozane
AR110451A1 (es) * 2016-12-26 2019-03-27 Shionogi & Co Compuesto tricíclico que tiene sulfinilo y composición farmacéutica que lo comprende

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0009008A3 (de) * 1978-09-08 1980-05-14 Ciba-Geigy Ag Cephalosporinderivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
TW427993B (en) * 1993-09-09 2001-04-01 Fujisawa Pharmaceutical Co New cephem compounds
JPH10510258A (ja) * 1994-12-09 1998-10-06 藤沢薬品工業株式会社 セフェム化合物およびその医薬用途
MY127641A (en) * 1995-10-12 2006-12-29 Essential Therapeutics Inc Cephalosporin antibiotics
JPH09278778A (ja) * 1996-04-12 1997-10-28 Kyorin Pharmaceut Co Ltd 抗mrsaセファロスポリン化合物
US6030965A (en) * 1997-09-30 2000-02-29 Microcide Pharmaceuticals, Inc. Cephalosporin antibiotics

Also Published As

Publication number Publication date
WO2002017854A2 (en) 2002-03-07
CN1471399A (zh) 2004-01-28
ZA200301391B (en) 2004-02-20
TWI283681B (en) 2007-07-11
JP2004507481A (ja) 2004-03-11
US6599893B2 (en) 2003-07-29
CA2420871A1 (en) 2002-03-07
EP1333836A4 (en) 2004-07-07
AU2001288420B2 (en) 2006-09-28
IL154518A0 (en) 2003-09-17
MXPA03001782A (es) 2004-11-01
AR030503A1 (es) 2003-08-20
NO20030931D0 (no) 2003-02-27
US20020115650A1 (en) 2002-08-22
NO20030931L (no) 2003-04-29
NZ524438A (en) 2005-08-26
WO2002017854A3 (en) 2002-06-13
EP1333836A2 (en) 2003-08-13
RU2281948C2 (ru) 2006-08-20
AU8842001A (en) 2002-03-13

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A E 8A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2021 DE 29/09/2009.