FI824314L
(fi)
*
|
1981-12-16 |
1983-06-17 |
Sankyo Co |
Thienopyrimidin-derivater, deras framstaellning och deras medicinska anvaendning
|
JPS60146891A
(ja)
*
|
1984-01-05 |
1985-08-02 |
Mitsubishi Chem Ind Ltd |
〔2,3−d〕チエノピリミジン誘導体およびその塩
|
JPH068292B2
(ja)
*
|
1985-05-07 |
1994-02-02 |
アルカロイダ ベギエスゼティ ギャル |
トリアゾリルキノリン誘導体
|
US4670560A
(en)
*
|
1986-04-28 |
1987-06-02 |
Ortho Pharmaceutical Corporation |
Thienopyrimidine-2,4-dione derivatives and intermediates thereof
|
EP0364598A4
(en)
*
|
1988-03-02 |
1992-01-15 |
Yoshitomi Pharmaceutical Industries, Ltd. |
3,4-dihydrothieno 2,3-d¨pyrimidine compounds and pharmaceutical application thereof
|
US5280026A
(en)
*
|
1989-05-30 |
1994-01-18 |
Smithkline Beecham Intercredit B.V. |
Thienopyrimidines
|
GB8912335D0
(en)
*
|
1989-05-30 |
1989-07-12 |
Smithkline Beckman Intercredit |
Compounds
|
DE4008726A1
(de)
*
|
1990-03-19 |
1991-09-26 |
Basf Ag |
Thieno(2,3-d)pyrimidinderivate
|
BR9101256A
(pt)
*
|
1990-03-30 |
1991-11-05 |
Dowelanco |
Composto,composicao fungicida,processo fungicida,composicao inseticida ou acaricida e processo inseticida ou acaricida
|
US5869486A
(en)
*
|
1995-02-24 |
1999-02-09 |
Ono Pharmaceutical Co., Ltd. |
Fused pyrimidines and pyriazines as pharmaceutical compounds
|
PT757984E
(pt)
*
|
1995-08-08 |
2003-02-28 |
Ono Pharmaceutical Co |
Derivados de acido hidroxamico uteis para inibir a gelatinase
|
DE19632423A1
(de)
*
|
1996-08-12 |
1998-02-19 |
Merck Patent Gmbh |
Thienopyrimidine
|
DE19650378A1
(de)
*
|
1996-12-05 |
1998-06-10 |
Basf Ag |
Neue Pyrimidylverbindungen als Pflanzenschutzmittel
|
WO1998027087A1
(fr)
*
|
1996-12-18 |
1998-06-25 |
Eli Lilly And Company |
Procede combinatoire de realisation d'echantillotheques de pyrimidines fondues
|
US20030162795A1
(en)
*
|
1998-10-22 |
2003-08-28 |
Pfizer Inc. |
Thienopyrimidine and thienopyridine derivatives useful as anticancer agents
|
US6133271A
(en)
*
|
1998-11-19 |
2000-10-17 |
Cell Pathways, Inc. |
Method for inhibiting neoplastic cells and related conditions by exposure thienopyrimidine derivatives
|
US6608053B2
(en)
*
|
2000-04-27 |
2003-08-19 |
Yamanouchi Pharmaceutical Co., Ltd. |
Fused heteroaryl derivatives
|
US6503914B1
(en)
|
2000-10-23 |
2003-01-07 |
Board Of Regents, The University Of Texas System |
Thienopyrimidine-based inhibitors of the Src family
|
WO2002088138A1
(fr)
*
|
2001-04-30 |
2002-11-07 |
Bayer Corporation |
Nouveaux thiopheno[2,3-d]pyrimidines 4-amino-5,6-substitutes
|
US6805491B2
(en)
*
|
2002-05-20 |
2004-10-19 |
Stratos International, Inc. |
Stub having an optical fiber
|
AR044743A1
(es)
*
|
2002-09-26 |
2005-10-05 |
Nihon Nohyaku Co Ltd |
Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos,
|
US7612078B2
(en)
*
|
2003-03-31 |
2009-11-03 |
Epix Delaware, Inc. |
Piperidinylamino-thieno[2,3-D] pyrimidine compounds
|
ATE511511T1
(de)
*
|
2003-03-31 |
2011-06-15 |
Trovis Pharmaceuticals Llc |
Neue piperidinylaminothienoä2,3-dü pyrimidinverbindungen
|
US20050222175A1
(en)
*
|
2004-03-31 |
2005-10-06 |
Dhanoa Dale S |
New piperidinylamino-thieno[2,3-D] pyrimidine compounds
|
GB0315950D0
(en)
|
2003-06-11 |
2003-08-13 |
Xention Discovery Ltd |
Compounds
|
US7488736B2
(en)
*
|
2004-05-17 |
2009-02-10 |
Epix Delaware, Inc. |
Thienopyridinone compounds and methods of treatment
|
GB0412467D0
(en)
*
|
2004-06-04 |
2004-07-07 |
Astrazeneca Ab |
Chemical compounds
|
GB0412986D0
(en)
|
2004-06-10 |
2004-07-14 |
Xention Discovery Ltd |
Compounds
|
KR20070057792A
(ko)
*
|
2004-07-16 |
2007-06-07 |
선에시스 파마슈티컬스 인코포레이티드 |
오로라 키나아제 저해물질로서 유용한 티에노피리미딘
|
GB0420719D0
(en)
*
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
US7598265B2
(en)
*
|
2004-09-30 |
2009-10-06 |
Epix Delaware, Inc. |
Compositions and methods for treating CNS disorders
|
US7407966B2
(en)
*
|
2004-10-07 |
2008-08-05 |
Epix Delaware, Inc. |
Thienopyridinone compounds and methods of treatment
|
US7576211B2
(en)
*
|
2004-09-30 |
2009-08-18 |
Epix Delaware, Inc. |
Synthesis of thienopyridinone compounds and related intermediates
|
CA2583259C
(fr)
*
|
2004-10-08 |
2011-08-02 |
Astellas Pharma Inc. |
Derive polycyclique aromatique de pyrimidine
|
KR101386797B1
(ko)
*
|
2004-10-21 |
2014-04-21 |
다우 아그로사이언시즈 엘엘씨 |
살진균 활성을 갖는 티에노-피리미딘 화합물
|
GB0423653D0
(en)
*
|
2004-10-25 |
2004-11-24 |
Piramed Ltd |
Pharmaceutical compounds
|
US7576212B2
(en)
|
2004-12-09 |
2009-08-18 |
Xention Limited |
Thieno[2,3-B] pyridines as potassium channel inhibitors
|
US7576080B2
(en)
*
|
2004-12-23 |
2009-08-18 |
Memory Pharmaceuticals Corporation |
Certain thienopyrimidine derivatives as phosphodiesterase 10 inhibitors
|
EP1928884B1
(fr)
*
|
2005-09-23 |
2010-01-13 |
Equispharm Co., Ltd. |
Derives de 5,6-dimethyl[2,3-di]pyrimidine, leurs procede de preparation et composition pharmaceutique les comportant pour un traitement antiviral
|
EP1937691A1
(fr)
|
2005-10-21 |
2008-07-02 |
Dow Agrosciences LLC |
Composes de thieno-pyrimidine a activite fongicide
|
US7531482B2
(en)
*
|
2005-10-21 |
2009-05-12 |
Dow Agrosciences Llc |
Thieno-pyrimidine compounds having fungicidal activity
|
WO2007056215A2
(fr)
*
|
2005-11-02 |
2007-05-18 |
Cytovia, Inc. |
N-aryl-thienopyrimidin-4-amines et analogues en tant qu'activateurs de caspases et inducteurs d'apoptose et utilisation associee
|
WO2007056214A2
(fr)
*
|
2005-11-02 |
2007-05-18 |
Cytovia, Inc |
N-alkyl-n-aryl-thienopyrimidin-4-amines et analogues en tant qu'activateurs de caspases et inducteurs d'apoptose et utilisation associee
|
US20070099941A1
(en)
*
|
2005-11-02 |
2007-05-03 |
Cytovia, Inc. |
N-arylalkyl-thienopyrimidin-4-amines and analogs as activators of caspases and inducers of apoptosis and the use thereof
|
GB0525164D0
(en)
|
2005-12-09 |
2006-01-18 |
Xention Discovery Ltd |
Compounds
|
TWI417095B
(zh)
|
2006-03-15 |
2013-12-01 |
Janssen Pharmaceuticals Inc |
1,4-二取代之3-氰基-吡啶酮衍生物及其作為mGluR2-受體之正向異位性調節劑之用途
|
AU2007243457B2
(en)
|
2006-04-26 |
2012-02-23 |
F. Hoffmann-La Roche Ag |
Pharmaceutical compounds
|
TW200801012A
(en)
|
2006-04-26 |
2008-01-01 |
Piramed Ltd |
Phosphoinositide 3-kinase inhibitor compounds and methods of use
|
US7781433B2
(en)
*
|
2006-04-26 |
2010-08-24 |
Piramed Limited |
Pharmaceutical compounds
|
KR20090018144A
(ko)
|
2006-05-22 |
2009-02-19 |
바스프 에스이 |
4-아미노-5-클로로-티에노[2,3-d]-피리미딘 화합물을 사용하는 살충 방법
|
US9487533B2
(en)
*
|
2006-12-07 |
2016-11-08 |
Genentech, Inc. |
Phosphoinositide 3-kinase inhibitor compounds and methods of use
|
MY180595A
(en)
*
|
2006-12-07 |
2020-12-03 |
Genentech Inc |
Phosphoinositide 3-kinase inhibitor compounds and methods of use
|
TW200845978A
(en)
*
|
2007-03-07 |
2008-12-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
|
TW200900065A
(en)
|
2007-03-07 |
2009-01-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
|
US7928111B2
(en)
|
2007-06-08 |
2011-04-19 |
Senomyx, Inc. |
Compounds including substituted thienopyrimidinone derivatives as ligands for modulating chemosensory receptors
|
US9603848B2
(en)
*
|
2007-06-08 |
2017-03-28 |
Senomyx, Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
US8633186B2
(en)
|
2007-06-08 |
2014-01-21 |
Senomyx Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
AU2008297877C1
(en)
*
|
2007-09-14 |
2013-11-07 |
Addex Pharma S.A. |
1,3-disubstituted-4-phenyl-1 H-pyridin-2-ones
|
CN101801951B
(zh)
|
2007-09-14 |
2013-11-13 |
杨森制药有限公司 |
1’,3’-二取代的-4-苯基-3,4,5,6-四氢-2h,1’h-[1,4’]二吡啶-2’-酮
|
EP2200985B1
(fr)
|
2007-09-14 |
2011-07-13 |
Ortho-McNeil-Janssen Pharmaceuticals, Inc. |
4-(aryl-x-phényl)-1h-pyridine-2-ones 1,3-disubstituées
|
US8354528B2
(en)
*
|
2007-10-25 |
2013-01-15 |
Genentech, Inc. |
Process for making thienopyrimidine compounds
|
GB0721095D0
(en)
*
|
2007-10-26 |
2007-12-05 |
Piramed Ltd |
Pharmaceutical compounds
|
CN101861316B
(zh)
*
|
2007-11-14 |
2013-08-21 |
奥梅-杨森制药有限公司 |
咪唑并[1,2-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途
|
CA2731800C
(fr)
|
2008-07-31 |
2018-03-20 |
Senomyx, Inc. |
Procedes et intermediaires pour la realisation d'exhausteurs de gout sucre
|
WO2010014813A2
(fr)
|
2008-07-31 |
2010-02-04 |
Senomyx, Inc. |
Compositions comprenant des édulcorants et leurs procédés de préparation
|
ES2439291T3
(es)
|
2008-09-02 |
2014-01-22 |
Janssen Pharmaceuticals, Inc. |
Derivados de 3-azabiciclo[3.1.0]hexilo como moduladores de receptores de glutamato metabotrópicos
|
JP5656848B2
(ja)
|
2008-10-16 |
2015-01-21 |
ジャンセン ファーマシューティカルズ, インコーポレイテッド. |
代謝型グルタミン酸受容体モジュレーターとしてのインドールおよびベンゾモルホリンの誘導体
|
US8691813B2
(en)
|
2008-11-28 |
2014-04-08 |
Janssen Pharmaceuticals, Inc. |
Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
|
WO2010065743A2
(fr)
*
|
2008-12-03 |
2010-06-10 |
Nanotherapeutics, Inc. |
Composés bicycliques et leurs procédés de fabrication et d'utilisation
|
MX2011011962A
(es)
|
2009-05-12 |
2012-02-28 |
Janssen Pharmaceuticals Inc |
Derivados de 1,2,4-triazolo[4,3-a]piridina y su uso como moduladores alostericos positivos de receptores de glutamato metabotropico (mglur2).
|
ME01573B
(me)
|
2009-05-12 |
2014-09-20 |
Addex Pharma Sa |
DERIVATI 1,2,4-TRIAZOLO[4,3-a]PIRIDINA I NJIHOVA UPOTREBA U TRETMANU ILI PREVENCIJI NEUROLOŠKIH I PSIHIJATRIJSKIH POREMEĆAJA
|
MY153913A
(en)
|
2009-05-12 |
2015-04-15 |
Janssen Pharmaceuticals Inc |
7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
|
JP5781066B2
(ja)
|
2009-05-27 |
2015-09-16 |
ジェネンテック, インコーポレイテッド |
p110δに対して選択的な二環式ピリミジンPI3K阻害剤化合物及び使用方法
|
WO2010136491A1
(fr)
*
|
2009-05-27 |
2010-12-02 |
F. Hoffmann-La Roche Ag |
Composés bicycliques indole-pyrimidine inhibiteurs de pi3k sélectifs pour p110 delta et leurs procédés d'utilisation
|
JP5325297B2
(ja)
*
|
2009-07-16 |
2013-10-23 |
株式会社エス・ディー・エス バイオテック |
農園芸用の有害生物防除剤としての4−(3−ブチニル)アミノピリミジン誘導体
|
WO2011014660A1
(fr)
|
2009-07-30 |
2011-02-03 |
Merial Limited |
Composés insecticides à base de 4‑amino-thiéno[2,3-d]pyrimidine et leurs méthodes d'utilisation
|
EP2488178B1
(fr)
*
|
2009-10-12 |
2016-11-16 |
F.Hoffmann-La Roche Ag |
Combinaisons d'un inhibiteur de pi3k et d'un inhibiteur de mek
|
WO2012012712A2
(fr)
*
|
2010-07-23 |
2012-01-26 |
President And Fellows Of Harvard College |
Composés renforçant l'activité protéasome tricyclique
|
US9000054B2
(en)
|
2010-08-12 |
2015-04-07 |
Senomyx, Inc. |
Method of improving stability of sweet enhancer and composition containing stabilized sweet enhancer
|
JP5852666B2
(ja)
|
2010-11-08 |
2016-02-03 |
ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド |
1,2,4−トリアゾロ[4,3−a]ピリジン誘導体およびmGluR2受容体のポジティブアロステリックモジュレーターとしてのそれらの使用
|
AU2011328195B2
(en)
|
2010-11-08 |
2015-04-02 |
Janssen Pharmaceuticals, Inc. |
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
|
US9271967B2
(en)
|
2010-11-08 |
2016-03-01 |
Janssen Pharmaceuticals, Inc. |
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
|
TWI441824B
(zh)
|
2010-12-16 |
2014-06-21 |
Hoffmann La Roche |
三環pi3k抑制劑化合物及其使用方法
|
NZ613449A
(en)
*
|
2011-01-14 |
2015-08-28 |
Sds Biotech Corp |
Agri-horticultural pest control compositions comprising 4-(3-butynyl)aminopyrimidine derivatives
|
CA2825028A1
(fr)
*
|
2011-02-09 |
2012-08-16 |
F. Hoffman-La Roche Ag |
Composes heterocycliques en tant qu'inhibiteurs de pi3 kinase
|
CN103946226A
(zh)
|
2011-07-19 |
2014-07-23 |
无限药品股份有限公司 |
杂环化合物及其应用
|
MX354835B
(es)
|
2012-08-06 |
2018-03-21 |
Senomyx Inc |
Modificador del sabor dulce.
|
JO3155B1
(ar)
|
2013-02-19 |
2017-09-20 |
Senomyx Inc |
معدِّل نكهة حلوة
|
JO3368B1
(ar)
|
2013-06-04 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
|
JO3367B1
(ar)
|
2013-09-06 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
|
PL3096790T3
(pl)
|
2014-01-21 |
2020-01-31 |
Janssen Pharmaceutica, N.V. |
Kombinacje zawierające pozytywne modulatory allosteryczne lub agonistów ortosterycznych metabotropowego receptora glutaminergicznego podtypu 2 i ich zastosowanie
|
KR20200036063A
(ko)
|
2014-01-21 |
2020-04-06 |
얀센 파마슈티카 엔.브이. |
대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
|
CN104725398B
(zh)
*
|
2015-01-29 |
2017-01-18 |
杨威 |
一种jak/stat3磷酸化抑制剂及其制备方法与用途
|
US11312690B2
(en)
*
|
2015-07-24 |
2022-04-26 |
University Of Lousville Research Foundation, Inc. |
Compounds, compositions, methods for treating diseases, and methods for preparing compounds
|
US20220117968A1
(en)
*
|
2017-07-17 |
2022-04-21 |
Saint Louis University |
Thieno[2,3-d)pyrimidines and benzofuro(3,2-d)pyrimidines as antimicrobial agents
|
MX2021001193A
(es)
|
2018-08-07 |
2021-04-28 |
Firmenich Incorporated |
2,2-dioxidos de 4-amino-1h-benzo[c][1,2,6]tiadiazina 5-sustituidos y formulaciones y usos de los mismos.
|