BE794554A - Nouveaux derives de penicilline et de cephalusporine - Google Patents

Nouveaux derives de penicilline et de cephalusporine

Info

Publication number
BE794554A
BE794554A BE794554DA BE794554A BE 794554 A BE794554 A BE 794554A BE 794554D A BE794554D A BE 794554DA BE 794554 A BE794554 A BE 794554A
Authority
BE
Belgium
Prior art keywords
cephalusporin
penicillin
new derivatives
derivatives
new
Prior art date
Application number
Other languages
English (en)
Inventor
G A Koppel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Publication of BE794554A publication Critical patent/BE794554A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/57—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with a further substituent in position 7, e.g. cephamycines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BE794554D 1972-01-31 Nouveaux derives de penicilline et de cephalusporine BE794554A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22229372A 1972-01-31 1972-01-31
US30169472A 1972-10-27 1972-10-27

Publications (1)

Publication Number Publication Date
BE794554A true BE794554A (fr) 1973-07-26

Family

ID=26916655

Family Applications (1)

Application Number Title Priority Date Filing Date
BE794554D BE794554A (fr) 1972-01-31 Nouveaux derives de penicilline et de cephalusporine

Country Status (23)

Country Link
US (1) US3994885A (fr)
JP (2) JPS4885595A (fr)
AR (2) AR209256A1 (fr)
AT (1) AT327378B (fr)
AU (1) AU465803B2 (fr)
BE (1) BE794554A (fr)
BG (1) BG34453A3 (fr)
CA (1) CA1033718A (fr)
CH (1) CH571525A5 (fr)
CS (1) CS195262B2 (fr)
DD (1) DD103900A5 (fr)
DE (1) DE2304226C3 (fr)
ES (1) ES411163A1 (fr)
FR (1) FR2170051B1 (fr)
GB (1) GB1412886A (fr)
HU (1) HU170405B (fr)
IE (1) IE37252B1 (fr)
IL (1) IL41361A (fr)
NL (1) NL179207C (fr)
PH (1) PH12535A (fr)
SE (1) SE418184B (fr)
YU (1) YU36964B (fr)
ZA (1) ZA73407B (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU36181B (en) * 1971-11-29 1982-02-25 Merck & Co Inc Process for obtaining 7-(2-thienylacetamido)-7-methoxy-3-carbamoyloxymethyl-3-cephem-4-carboxylates
US4447602A (en) * 1971-11-29 1984-05-08 Merck & Co., Inc. Process to prepare 7-substituted cephalosporins or 6-substituted penicillins
CA1040620A (fr) * 1972-11-14 1978-10-17 Frank J. Urban Alkoxy-6 acylamidopenicillines-6 et alkoxy-7 acylamido-7 acetoxycephalosporines
DE2460477A1 (de) * 1973-12-26 1975-07-10 Yamanouchi Pharma Co Ltd Verbessertes verfahren zur herstellung von 6-alkoxy-substituierten penicillinen
US3991051A (en) * 1975-05-01 1976-11-09 E. R. Squibb & Sons, Inc. [(Oxyalkyl)thioacetyl]cephalosporin derivatives
US3989696A (en) * 1975-05-01 1976-11-02 E. R. Squibb & Sons, Inc. 3-Heterothio[(oxyalkyl)thioacetyl]cephalosporin derivatives
JPS5941999B2 (ja) 1975-07-24 1984-10-11 武田薬品工業株式会社 セフエムまたはベナム化合物の製造法
JPS5279081A (en) * 1975-12-25 1977-07-02 Yamanouchi Pharmaceut Co Ltd Preparation of novel 7-methoxycephalosporins
CA1093997A (fr) * 1975-12-25 1981-01-20 Shunichi Watanabe Procede de production de 7-methoxy cephalosporines
JPS5422391A (en) * 1977-07-21 1979-02-20 Toyama Chem Co Ltd Preparation of novel 7alpha-methoxycephalosporins
US4048163A (en) * 1976-03-22 1977-09-13 Eli Lilly And Company Process for preparation of 7-alkoxy-3-chloromethylcephems
US4048160A (en) * 1976-03-22 1977-09-13 Eli Lilly And Company Process for preparation of 7-alkoxy-3-bromomethylcephems
US4165429A (en) * 1976-06-28 1979-08-21 Yamanouchi Pharmaceutical Co., Ltd. 7α-METHOXY-CEPHALOSPORANIC ACID DERIVATIVES
US4311837A (en) * 1979-05-01 1982-01-19 Eli Lilly And Company Certain heterocyclic thiomethyl derivatives of 7-(dihalogenated phenylthioacetamido)cephalosporanic acids useful in the treatment of infections caused by _Streptococcus faecalis
DE3373475D1 (en) * 1982-12-14 1987-10-15 Beecham Group Plc Process for the preparation of beta-lactam compounds
MY129257A (en) * 1995-03-21 2007-03-30 Betz Laboratories Methods of inhibiting corrosion using halo-benzotriazoles
US5773627A (en) * 1995-03-21 1998-06-30 Betzdearborn Inc. Methods of inhibiting corrosion using halo-benzotriazoles
AR035728A1 (es) * 2001-01-16 2004-07-07 Merck & Co Inc Proceso perfeccionado para la sintesis de carbapenem
US7662955B2 (en) * 2003-03-20 2010-02-16 Orchid Chemicals And Pharmaceuticals Ltd. Process for the preparation of cefoxitin

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3780031A (en) * 1971-11-29 1973-12-18 Merck & Co Inc Process for preparing cephalosporin compounds
US3780034A (en) * 1971-11-29 1973-12-18 Merck & Co Inc Process for preparing substituted cephalosporins
US3775410A (en) * 1971-11-29 1973-11-27 B Christensen Process for preparing cephalosporin compounds
US3780037A (en) * 1971-11-29 1973-12-18 Merck & Co Inc Process for preparing cephalosporin compounds
YU36181B (en) * 1971-11-29 1982-02-25 Merck & Co Inc Process for obtaining 7-(2-thienylacetamido)-7-methoxy-3-carbamoyloxymethyl-3-cephem-4-carboxylates

Also Published As

Publication number Publication date
ES411163A1 (es) 1976-04-16
JPS6021595B2 (ja) 1985-05-28
IE37252B1 (en) 1977-06-08
NL179207B (nl) 1986-03-03
DD103900A5 (fr) 1974-02-12
HU170405B (fr) 1977-06-28
NL7301419A (fr) 1973-08-02
YU36964B (en) 1984-08-31
AR209426A1 (es) 1977-04-29
CA1033718A (fr) 1978-06-27
ATA78373A (de) 1975-04-15
AU5137373A (en) 1974-07-25
CS195262B2 (en) 1980-01-31
NL179207C (nl) 1986-08-01
IE37252L (en) 1973-07-31
BG34453A3 (en) 1983-09-15
AU465803B2 (en) 1975-10-09
JPS5745188A (en) 1982-03-13
IL41361A (en) 1979-05-31
US3994885A (en) 1976-11-30
CH571525A5 (fr) 1976-01-15
IL41361A0 (en) 1973-03-30
FR2170051B1 (fr) 1976-10-22
DE2304226B2 (de) 1979-07-19
SE418184B (sv) 1981-05-11
DE2304226C3 (de) 1980-04-03
PH12535A (en) 1979-05-17
AR209256A1 (es) 1977-04-15
DE2304226A1 (de) 1973-08-16
ZA73407B (en) 1974-09-25
JPS4885595A (fr) 1973-11-13
YU22873A (en) 1982-06-18
FR2170051A1 (fr) 1973-09-14
GB1412886A (en) 1975-11-05
AT327378B (de) 1976-01-26

Similar Documents

Publication Publication Date Title
BE771584A (fr) Nouveaux derives de phenyl-imidazolyl-alcanyle et leur obtention
BE764019A (fr) Nouveaux derives du benzo-cyclohepta-thiophene et leur preparation
BE794554A (fr) Nouveaux derives de penicilline et de cephalusporine
BE779128A (fr) Nouveaux derives de benzazine
FR2102106A1 (fr) Nouveaux derives du benzocyclobutene
BE791889A (fr) Nouveaux derives de la pyridine
FR2291200A1 (fr) Nouveaux derives g-lactone et g-hemiacetal bicycliques
BE797905A (fr) Nouveaux derives du benzodioxole
BE794377A (fr) Nouveaux derives du benzo-cyclohepta-thiophene
AR214383A1 (es) Derivados de dialquilfosfanatos
BE758766A (fr) Nouveaux derives de la morpholine et de la
BE791907A (fr) Nouveaux derives des imidazolines
BE780630A (fr) Nouveaux derives d'imidazo-pyridine
BE784235A (fr) Nouveaux derives esters oxofuryliques de la penicilline et de la cephalosporine
FI55033B (fi) Foerfarande foer framstaellning av terapeutiskt aktiva pyrazin-4-oxidderivat
BE800894A (fr) Derives de phenylcetones et leur production
AR201288A1 (es) Derivados de alfa-cianmetansulfonamidobenceno
SE385433B (sv) Av tradar bestaende netbotten
BE771115A (fr) Derives de la quinoleine et leur preparation
BE797823A (fr) Nouveaux derives du benzo-cyclohepia-thiophine
BE794159A (fr) Nouveaux composes furaniques et application de ceux-ci
BE802797A (fr) Nouveaux derives de beta-aminocetones
BE799615A (fr) Nouveaux derives de la 6alpha-methylprednisolone
BE795041A (fr) Nouveaux derives de l'amino-propane
BE748030A (fr) Nouveaux derives de la phenothiazine

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: ELI LILLY AND CY

Effective date: 19890131