AU703380B2 - Stereoselective process - Google Patents
Stereoselective process Download PDFInfo
- Publication number
- AU703380B2 AU703380B2 AU12878/97A AU1287897A AU703380B2 AU 703380 B2 AU703380 B2 AU 703380B2 AU 12878/97 A AU12878/97 A AU 12878/97A AU 1287897 A AU1287897 A AU 1287897A AU 703380 B2 AU703380 B2 AU 703380B2
- Authority
- AU
- Australia
- Prior art keywords
- alkyl
- phenyl
- coor
- group
- rio
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C235/06—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
- C07D317/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Surface Acoustic Wave Elements And Circuit Networks Thereof (AREA)
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US875895P | 1995-12-12 | 1995-12-12 | |
| US60/008758 | 1995-12-12 | ||
| GB9602833 | 1996-02-13 | ||
| GBGB9602833.7A GB9602833D0 (en) | 1996-02-13 | 1996-02-13 | Stereoselective process |
| US1328896P | 1996-03-12 | 1996-03-12 | |
| US60/013288 | 1996-03-12 | ||
| GB9608928 | 1996-04-29 | ||
| GBGB9608928.9A GB9608928D0 (en) | 1996-04-29 | 1996-04-29 | Stereoselective process |
| PCT/US1996/019782 WO1997021693A1 (en) | 1995-12-12 | 1996-12-09 | Stereoselective process |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU1287897A AU1287897A (en) | 1997-07-03 |
| AU703380B2 true AU703380B2 (en) | 1999-03-25 |
Family
ID=27451397
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU12878/97A Ceased AU703380B2 (en) | 1995-12-12 | 1996-12-09 | Stereoselective process |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP0869950A1 (ja) |
| JP (1) | JP2000501737A (ja) |
| AU (1) | AU703380B2 (ja) |
| CA (1) | CA2238960A1 (ja) |
| WO (1) | WO1997021693A1 (ja) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6451827B2 (en) | 1998-05-12 | 2002-09-17 | Wyeth | 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia |
| US6699896B1 (en) | 1998-05-12 | 2004-03-02 | Wyeth | Oxazole-aryl-carboxylic acids useful in the treatment of insulin resistance and hyperglycemia |
| US6110963A (en) * | 1998-05-12 | 2000-08-29 | American Home Products Corporation | Aryl-oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia |
| US6166069A (en) * | 1998-05-12 | 2000-12-26 | American Home Products Corporation | Phenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia |
| US6232322B1 (en) | 1998-05-12 | 2001-05-15 | American Home Products Corporation | Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia |
| US6214877B1 (en) | 1998-05-12 | 2001-04-10 | John A. Butera | 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia |
| US6221902B1 (en) | 1998-05-12 | 2001-04-24 | American Home Products Corporation | Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia |
| US6310081B1 (en) | 1999-05-10 | 2001-10-30 | American Home Products Corporation | Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia |
| US7091230B2 (en) | 2001-02-09 | 2006-08-15 | Merck & Co., Inc. | 2-aryloxy-2-arylalkanoic acids for diabetes and lipid disorders |
| EP2298729A4 (en) * | 2008-06-03 | 2012-12-19 | Kaneka Corp | PROCESS FOR PRODUCING OPTICALLY ACTIVE AMINO ACID DERIVATIVE |
-
1996
- 1996-12-09 AU AU12878/97A patent/AU703380B2/en not_active Ceased
- 1996-12-09 WO PCT/US1996/019782 patent/WO1997021693A1/en not_active Application Discontinuation
- 1996-12-09 CA CA 2238960 patent/CA2238960A1/en not_active Abandoned
- 1996-12-09 JP JP09522200A patent/JP2000501737A/ja active Pending
- 1996-12-09 EP EP96943713A patent/EP0869950A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| AU1287897A (en) | 1997-07-03 |
| WO1997021693A1 (en) | 1997-06-19 |
| JP2000501737A (ja) | 2000-02-15 |
| CA2238960A1 (en) | 1997-06-19 |
| EP0869950A1 (en) | 1998-10-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |