AU4506399A - Aryl pyridinyl thiazoles - Google Patents

Aryl pyridinyl thiazoles

Info

Publication number
AU4506399A
AU4506399A AU45063/99A AU4506399A AU4506399A AU 4506399 A AU4506399 A AU 4506399A AU 45063/99 A AU45063/99 A AU 45063/99A AU 4506399 A AU4506399 A AU 4506399A AU 4506399 A AU4506399 A AU 4506399A
Authority
AU
Australia
Prior art keywords
thiazoles
pyridinyl
aryl
aryl pyridinyl
pyridinyl thiazoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU45063/99A
Inventor
Thomas Hugo Keller
Neil John Press
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9812117.1A external-priority patent/GB9812117D0/en
Priority claimed from GBGB9818653.9A external-priority patent/GB9818653D0/en
Application filed by Novartis AG filed Critical Novartis AG
Publication of AU4506399A publication Critical patent/AU4506399A/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
    • C07D213/46Oxygen atoms
    • C07D213/50Ketonic radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
AU45063/99A 1998-06-05 1999-06-03 Aryl pyridinyl thiazoles Abandoned AU4506399A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB9812117 1998-06-05
GBGB9812117.1A GB9812117D0 (en) 1998-06-05 1998-06-05 Organic compounds
GB9818653 1998-08-26
GBGB9818653.9A GB9818653D0 (en) 1998-08-26 1998-08-26 Organic compounds
PCT/EP1999/003859 WO1999064418A1 (en) 1998-06-05 1999-06-03 Aryl pyridinyl thiazoles

Publications (1)

Publication Number Publication Date
AU4506399A true AU4506399A (en) 1999-12-30

Family

ID=26313800

Family Applications (1)

Application Number Title Priority Date Filing Date
AU45063/99A Abandoned AU4506399A (en) 1998-06-05 1999-06-03 Aryl pyridinyl thiazoles

Country Status (2)

Country Link
AU (1) AU4506399A (en)
WO (1) WO1999064418A1 (en)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001010865A1 (en) * 1999-08-06 2001-02-15 Takeda Chemical Industries, Ltd. p38MAP KINASE INHIBITORS
BR0013899A (en) 1999-09-10 2003-07-08 Merck & Co Inc A compound, pharmaceutical composition, processes for treating or preventing cancer, a disease in which angiogenesis is implicated, retinal vascularization, diabetic retinopathy, age-related macular degeneration, inflammatory diseases, tyrosine-dependent disease or conditions. kinase, bone-associated pathologies, and processes for producing a pharmaceutical composition, and for reducing or preventing tissue damage following a cerebral ischemic event
EP1224185B1 (en) * 1999-10-27 2005-11-30 Novartis AG Thiazole and imidazo[4,5-b]pyridine compounds and their pharmaceutical use
DE60136530D1 (en) 2000-03-01 2008-12-24 Janssen Pharmaceutica Nv 2,4-DISUBSTITUTED THIAZOLYL DERIVATIVES
EP1268474A2 (en) * 2000-03-30 2003-01-02 Takeda Chemical Industries, Ltd. Substituted 1,3-thiazole compounds, their production and use
US7189717B2 (en) * 2000-04-26 2007-03-13 Eisai Co., Ltd. Medicinal compositions promoting bowel movement
GB0028383D0 (en) 2000-11-21 2001-01-03 Novartis Ag Organic compounds
CA2437248A1 (en) * 2001-02-02 2002-08-15 Takeda Chemical Industries, Ltd. Jnk inhibitor
CA2444487A1 (en) * 2001-05-18 2002-11-28 Endacea Inc. Methods and formulations of using a1 adenosine and p2x purinoreceptor antagonists
JP2004535437A (en) 2001-06-22 2004-11-25 メルク エンド カムパニー インコーポレーテッド Tyrosine kinase inhibitor
CA2451980C (en) 2001-08-13 2012-12-11 Janssen Pharmaceutica N.V. 2-amino-4,5-trisubstituted thiazolyl derivatives and their use against autoimmune disorders
TWI301834B (en) 2001-10-22 2008-10-11 Eisai R&D Man Co Ltd Pyrimidone compound and pharmaceutical composition including the same
JP2005510508A (en) * 2001-11-08 2005-04-21 藤沢薬品工業株式会社 Thiazolepyridazinones as adenosine antagonists
US6872724B2 (en) 2002-07-24 2005-03-29 Merck & Co., Inc. Polymorphs with tyrosine kinase activity
CA2551611C (en) 2003-12-26 2013-06-25 Kyowa Hakko Kogyo Co., Ltd. Thiazole derivatives for treating or preventing parkinson's disease
GB0401336D0 (en) * 2004-01-21 2004-02-25 Novartis Ag Organic compounds
EP1794157B1 (en) * 2004-09-22 2014-02-26 H. Lundbeck A/S 2-acylaminothiazole derivatives
NZ554385A (en) * 2004-09-22 2010-01-29 Lundbeck & Co As H 2-Acylaminothiazole derivatives having affinity for the adenosine 2A
US7674912B2 (en) 2005-04-25 2010-03-09 H. Lundbeck A/S Pro-drugs of N-thiazol-2-yl-benzamide derivatives
EP1894930A4 (en) 2005-06-23 2010-06-23 Kyowa Hakko Kirin Co Ltd Thiazole derivative
JP5121453B2 (en) 2005-08-02 2013-01-16 協和発酵キリン株式会社 Treatment and / or prevention agent for sleep disorders
EP2198710A1 (en) 2008-12-19 2010-06-23 Bayer CropScience AG Use of 5-pyridin-4yl-(1,3) thiazoles for combating phytopathogenic fungi
ES2578363B1 (en) 2015-01-22 2017-01-31 Palobiofarma, S.L. A3 adenosine receptor modulators
ES2676535B1 (en) 2017-01-20 2019-04-29 Palobiofarma Sl MODULATORS OF A3 ADENOSINE RECEIVERS
CN109293652B (en) * 2017-07-24 2021-10-22 四川科伦博泰生物医药股份有限公司 Substituted thiazole derivative and application thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0149884B1 (en) * 1983-09-09 1992-12-16 Takeda Chemical Industries, Ltd. 5-pyridyl-1,3-thiazole derivatives, their production and use
EP0308020A3 (en) * 1987-09-18 1990-12-05 Merck & Co. Inc. 5-(aryl and heteroaryl)-6-(aryl and heteroaryl)-1,2-dihydro-2-oxo 3-pyridinecarboxylic acids and derivatives thereof
EP0797575B1 (en) * 1994-12-13 2003-10-15 F. Hoffmann-La Roche Ag Imidazole derivatives as protein kinase inhibitors in particular egf-r tyrosine kinase
JPH11193281A (en) * 1997-10-27 1999-07-21 Takeda Chem Ind Ltd Adenosine a3 receptor antagonistic agent and thiazole compound

Also Published As

Publication number Publication date
WO1999064418A1 (en) 1999-12-16

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase