AU2003202091A1 - Guanidine derivatives - Google Patents
Guanidine derivativesInfo
- Publication number
- AU2003202091A1 AU2003202091A1 AU2003202091A AU2003202091A AU2003202091A1 AU 2003202091 A1 AU2003202091 A1 AU 2003202091A1 AU 2003202091 A AU2003202091 A AU 2003202091A AU 2003202091 A AU2003202091 A AU 2003202091A AU 2003202091 A1 AU2003202091 A1 AU 2003202091A1
- Authority
- AU
- Australia
- Prior art keywords
- guanidine derivatives
- guanidine
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0208224.6 | 2002-04-10 | ||
GBGB0208224.6A GB0208224D0 (en) | 2002-04-10 | 2002-04-10 | Chemical compounds |
PCT/GB2003/000339 WO2003045901A2 (en) | 2002-04-10 | 2003-01-28 | Guanidine derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2003202091A1 true AU2003202091A1 (en) | 2003-06-10 |
AU2003202091A8 AU2003202091A8 (en) | 2003-06-10 |
Family
ID=9934563
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2003202091A Abandoned AU2003202091A1 (en) | 2002-04-10 | 2003-01-28 | Guanidine derivatives |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU2003202091A1 (en) |
GB (1) | GB0208224D0 (en) |
WO (1) | WO2003045901A2 (en) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2511521C (en) | 2002-12-30 | 2012-02-07 | Angiotech International Ag | Drug delivery from rapid gelling polymer composition |
US20050272723A1 (en) * | 2004-04-27 | 2005-12-08 | The Regents Of The University Of Michigan | Methods and compositions for treating diseases and conditions associated with mitochondrial function |
US20090275099A1 (en) * | 2004-04-27 | 2009-11-05 | Regents Of The University Of Michigan | Methods and compositions for treating diseases and conditions associated with mitochondrial function |
KR101562549B1 (en) | 2005-05-10 | 2015-10-23 | 인사이트 홀딩스 코포레이션 | Modulators of indoleamine 2,3-dioxygenase and methods of using the same |
TWI382974B (en) | 2005-12-20 | 2013-01-21 | Incyte Corp | N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase |
US20070203140A1 (en) * | 2006-02-09 | 2007-08-30 | Combs Andrew P | N-hydroxyguanidines as modulators of indoleamine 2,3-dioxygenase |
CL2007002650A1 (en) | 2006-09-19 | 2008-02-08 | Incyte Corp | COMPOUNDS DERIVED FROM HETEROCICLO N-HIDROXIAMINO; PHARMACEUTICAL COMPOSITION, USEFUL TO TREAT CANCER, VIRAL INFECTIONS AND NEURODEGENERATIVE DISORDERS BETWEEN OTHERS. |
US20080125470A1 (en) | 2006-09-19 | 2008-05-29 | Incyte Corporation | N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase |
PE20110308A1 (en) | 2008-07-08 | 2011-06-10 | Incyte Corp | 1,2,5-OXADIAZOLES AS INHIBITORS OF INDOLAMINE 2,3-DIOXYGENASE |
CA2780333C (en) | 2009-11-17 | 2016-05-24 | The Regents Of The University Of Michigan | 1,4-benzodiazepine-2,5-diones and related compounds with therapeutic properties |
CN103458886B (en) | 2010-12-08 | 2016-06-08 | 莱斯拉公司 | Pyriconyl guanidine F1F0-atpase inhibitor and therapeutical uses thereof |
HUE035881T2 (en) | 2010-12-08 | 2018-05-28 | Lycera Corp | Pyrazolyl guanidine f1f0-atpase inhibitors and therapeutic uses thereof |
US9169199B2 (en) | 2010-12-08 | 2015-10-27 | Lycera Corporation | Cycloalkyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof |
US9580391B2 (en) | 2012-06-08 | 2017-02-28 | Lycera Corporation | Saturated acyl guanidine for inhibition of F1F0-ATPase |
WO2013185045A1 (en) | 2012-06-08 | 2013-12-12 | Lycera Corporation | Indazole guanidine f1f0-atpase inhibitors and therapeutic uses thereof |
US9221814B2 (en) | 2012-06-08 | 2015-12-29 | Lycera Corporation | Heterocyclic guanidine F1F0-atpase inhibitors and therapeutic uses thereof |
EP3066085B1 (en) | 2013-11-08 | 2020-05-13 | Incyte Holdings Corporation | Process for the synthesis of an indoleamine 2,3-dioxygenase inhibitor |
AU2014363904B2 (en) | 2013-12-10 | 2018-10-04 | Lycera Corporation | Trifluoromethyl pyrazolyl guanidine F1Fo-ATPase inhibitors and therapeutic uses thereof |
JP2016539983A (en) | 2013-12-10 | 2016-12-22 | リセラ・コーポレイションLycera Corporation | Alkylpyrazolylguanidine F1F0-ATPase inhibitor and therapeutic use thereof |
AU2014363907B2 (en) | 2013-12-10 | 2018-10-04 | Lycera Corporation | N-substituted pyrazolyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof |
CN109970675A (en) * | 2018-05-28 | 2019-07-05 | 中国医学科学院医药生物技术研究所 | One group of thiourea compound and its preparation method and application |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6054472A (en) * | 1996-04-23 | 2000-04-25 | Vertex Pharmaceuticals, Incorporated | Inhibitors of IMPDH enzyme |
AU3128197A (en) * | 1996-05-30 | 1998-01-05 | Children's Hospital Medical Center | Guanidino derivatives as inhibitors of the cytotoxic effect of peroxynitrite |
US6420403B1 (en) * | 1998-10-29 | 2002-07-16 | Edwin J. Iwanowicz | Inhibitors of IMPDH enzyme |
EP1218353B1 (en) * | 1999-07-07 | 2007-10-17 | AstraZeneca UK Limited | Quinazoline derivatives |
-
2002
- 2002-04-10 GB GBGB0208224.6A patent/GB0208224D0/en not_active Ceased
-
2003
- 2003-01-28 WO PCT/GB2003/000339 patent/WO2003045901A2/en not_active Application Discontinuation
- 2003-01-28 AU AU2003202091A patent/AU2003202091A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
GB0208224D0 (en) | 2002-05-22 |
WO2003045901A3 (en) | 2003-07-31 |
AU2003202091A8 (en) | 2003-06-10 |
WO2003045901A2 (en) | 2003-06-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |